MD4202B1 - Process for production of carbomethoxy derivatives of spiro[cyclopropane-oxindoles] - Google Patents
Process for production of carbomethoxy derivatives of spiro[cyclopropane-oxindoles]Info
- Publication number
- MD4202B1 MD4202B1 MD20120031A MD20120031A MD4202B1 MD 4202 B1 MD4202 B1 MD 4202B1 MD 20120031 A MD20120031 A MD 20120031A MD 20120031 A MD20120031 A MD 20120031A MD 4202 B1 MD4202 B1 MD 4202B1
- Authority
- MD
- Moldova
- Prior art keywords
- oxindoles
- cyclopropane
- spiro
- carbomethoxy
- derivatives
- Prior art date
Links
Landscapes
- Indole Compounds (AREA)
Abstract
The invention relates to the synthesis of spiro[cyclopropane-oxindoles] functionalized with the carbomethoxy group, which can serve as precursors in the synthesis of substances with anti-HIV activity.The process involves the reaction of cyclopropanation of diazoisatins with methyl acrylate, used both as reagent and solvent at its boiling point.The proposed process allows of carrying out the reaction in a shorter time with high yields, without the use of catalysts and inert atmosphere.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
MDA20120031A MD4202C1 (en) | 2012-03-21 | 2012-03-21 | Process for production of carbomethoxy derivatives of spiro[cyclopropane-oxindoles] |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
MDA20120031A MD4202C1 (en) | 2012-03-21 | 2012-03-21 | Process for production of carbomethoxy derivatives of spiro[cyclopropane-oxindoles] |
Publications (2)
Publication Number | Publication Date |
---|---|
MD4202B1 true MD4202B1 (en) | 2013-02-28 |
MD4202C1 MD4202C1 (en) | 2013-09-30 |
Family
ID=47831223
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MDA20120031A MD4202C1 (en) | 2012-03-21 | 2012-03-21 | Process for production of carbomethoxy derivatives of spiro[cyclopropane-oxindoles] |
Country Status (1)
Country | Link |
---|---|
MD (1) | MD4202C1 (en) |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS57102863A (en) * | 1980-12-16 | 1982-06-26 | Takeda Chem Ind Ltd | Spiroindolinone and its preparation |
FR2740136B1 (en) * | 1995-10-24 | 1998-01-09 | Sanofi Sa | INDOLIN-2-ONE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
US7205328B2 (en) * | 2002-10-21 | 2007-04-17 | Irm Llc | Oxindoles with anti-HIV activity |
US7370333B2 (en) * | 2003-06-02 | 2008-05-06 | Microsoft Corporation | Efficient processing of a convoy workflow scenario in a message driven process |
US7309787B2 (en) * | 2005-07-13 | 2007-12-18 | Allergan, Inc. | Kinase inhibitors |
-
2012
- 2012-03-21 MD MDA20120031A patent/MD4202C1/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
MD4202C1 (en) | 2013-09-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG4A | Patent for invention issued | ||
KA4A | Patent for invention lapsed due to non-payment of fees (with right of restoration) | ||
MM4A | Patent for invention definitely lapsed due to non-payment of fees |