MC1576A1 - Derives d'imidazole - Google Patents

Derives d'imidazole

Info

Publication number
MC1576A1
MC1576A1 MC841699A MC1693A MC1576A1 MC 1576 A1 MC1576 A1 MC 1576A1 MC 841699 A MC841699 A MC 841699A MC 1693 A MC1693 A MC 1693A MC 1576 A1 MC1576 A1 MC 1576A1
Authority
MC
Monaco
Prior art keywords
compound
formula
amino
lower alkoxy
acid
Prior art date
Application number
MC841699A
Other languages
English (en)
French (fr)
Inventor
Colin-Henry Cashin
Noel-Allan Roberts
Brian-Peter Tong
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838304182A external-priority patent/GB8304182D0/en
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MC1576A1 publication Critical patent/MC1576A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Dental Preparations (AREA)
  • Liquid Crystal Substances (AREA)
MC841699A 1983-02-15 1984-02-13 Derives d'imidazole MC1576A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB838304182A GB8304182D0 (en) 1983-02-15 1983-02-15 Pharmaceutical preparations
GB838329238A GB8329238D0 (en) 1983-02-15 1983-11-02 Pharmaceutical preparations

Publications (1)

Publication Number Publication Date
MC1576A1 true MC1576A1 (fr) 1985-02-04

Family

ID=26285246

Family Applications (1)

Application Number Title Priority Date Filing Date
MC841699A MC1576A1 (fr) 1983-02-15 1984-02-13 Derives d'imidazole

Country Status (11)

Country Link
US (1) US4612324A (cs)
EP (1) EP0118787A1 (cs)
AU (1) AU2428784A (cs)
DK (1) DK36584A (cs)
ES (1) ES529714A0 (cs)
FI (1) FI840389A7 (cs)
GR (1) GR79542B (cs)
IL (1) IL70912A0 (cs)
MC (1) MC1576A1 (cs)
NO (1) NO840545L (cs)
PT (1) PT78102B (cs)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ238688A (en) * 1990-06-28 1992-05-26 Smithkline Beecham Corp Substituted histidines: pharmaceutical compositions, preparation and uses thereof
IL95038A (en) * 1990-07-11 1995-10-31 Bromine Compounds Ltd Preparation of d-histidine and derivatives thereof by asymmetric transformation of l-histidine
US5741807A (en) * 1996-09-27 1998-04-21 Cytos Pharmaceuticals, L.P. Histidine compositions and methods for treating or preventing infectious and non-infectious diarrheas

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA698066A (en) * 1964-11-17 Merck And Co. Histidine derivatives
US2616828A (en) * 1951-04-30 1952-11-04 Levintow Leon Method of enzymatic resolution of amino acids
US3855238A (en) * 1970-10-14 1974-12-17 Eastman Kodak Co Process for preparing n-tertiary-butoxycarbonyl amino acids

Also Published As

Publication number Publication date
EP0118787A1 (de) 1984-09-19
ES8506643A1 (es) 1985-08-01
IL70912A0 (en) 1984-05-31
PT78102A (en) 1984-03-01
AU2428784A (en) 1984-08-23
FI840389L (fi) 1984-08-16
ES529714A0 (es) 1985-08-01
NO840545L (no) 1984-08-16
PT78102B (en) 1986-07-17
FI840389A0 (fi) 1984-01-31
US4612324A (en) 1986-09-16
DK36584D0 (da) 1984-01-26
GR79542B (cs) 1984-10-30
DK36584A (da) 1984-08-16
FI840389A7 (fi) 1984-08-16

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