MA49754A - Méthodes de traitement de symptômes de gastroparésie au moyen de velusetrag - Google Patents

Méthodes de traitement de symptômes de gastroparésie au moyen de velusetrag

Info

Publication number
MA49754A
MA49754A MA049754A MA49754A MA49754A MA 49754 A MA49754 A MA 49754A MA 049754 A MA049754 A MA 049754A MA 49754 A MA49754 A MA 49754A MA 49754 A MA49754 A MA 49754A
Authority
MA
Morocco
Prior art keywords
gastroparesia
velusetrag
methods
treating symptoms
symptoms
Prior art date
Application number
MA049754A
Other languages
English (en)
Inventor
Christopher Noel Barnes
Maria Grimaldi
Cecilia Renzulli
Giuseppe Claudio Viscomi
Original Assignee
Alfasigma Spa
Theravance Biopharma R&D Ip Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alfasigma Spa, Theravance Biopharma R&D Ip Llc filed Critical Alfasigma Spa
Publication of MA49754A publication Critical patent/MA49754A/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/47042-Quinolinones, e.g. carbostyril
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
MA049754A 2017-07-31 2018-07-30 Méthodes de traitement de symptômes de gastroparésie au moyen de velusetrag MA49754A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201762539229P 2017-07-31 2017-07-31

Publications (1)

Publication Number Publication Date
MA49754A true MA49754A (fr) 2020-06-10

Family

ID=63245036

Family Applications (1)

Application Number Title Priority Date Filing Date
MA049754A MA49754A (fr) 2017-07-31 2018-07-30 Méthodes de traitement de symptômes de gastroparésie au moyen de velusetrag

Country Status (18)

Country Link
US (1) US11642339B2 (fr)
EP (1) EP3661518B1 (fr)
JP (2) JP7431721B2 (fr)
KR (1) KR102692887B1 (fr)
CN (1) CN110996961A (fr)
AU (1) AU2018309667B2 (fr)
BR (1) BR112020000482A2 (fr)
CA (1) CA3069989A1 (fr)
CL (1) CL2019003598A1 (fr)
EA (1) EA202090416A1 (fr)
IL (1) IL272023B1 (fr)
MA (1) MA49754A (fr)
MX (1) MX2020001217A (fr)
SG (1) SG11201912266QA (fr)
TW (1) TW201909896A (fr)
UA (1) UA125596C2 (fr)
WO (1) WO2019027881A1 (fr)
ZA (1) ZA201908495B (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2024061960A1 (fr) 2022-09-20 2024-03-28 Alfasigma S.P.A. Velusetrag destiné à être utilisé dans le traitement de la pseudo-obstruction intestinale chronique (poic)

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7728006B2 (en) 2004-04-07 2010-06-01 Theravance, Inc. Quinolinone-carboxamide compounds as 5-HT4 receptor agonists
US8309575B2 (en) 2004-04-07 2012-11-13 Theravance, Inc. Quinolinone-carboxamide compounds as 5-HT4 receptor agonists
TWI351282B (en) 2004-04-07 2011-11-01 Theravance Inc Quinolinone-carboxamide compounds as 5-ht4 recepto
TWI377206B (en) * 2005-04-06 2012-11-21 Theravance Inc Crystalline form of a quinolinone-carboxamide compound
CN101384588B (zh) 2006-02-16 2011-08-31 施万制药 制备5-ht4受体激动剂化合物的中间体的方法
AU2010236734B2 (en) 2009-04-13 2015-06-11 Theravance Biopharma R&D Ip, Llc 5-HT4 receptor agonist compounds for treatment of cognitive disorders
US20130045988A1 (en) * 2011-08-18 2013-02-21 Shire Ag Combination therapy
PT2747561T (pt) * 2011-08-25 2018-09-28 Evoke Pharma Inc Tratamento de sintomas associados com a gastroparesia feminina

Also Published As

Publication number Publication date
SG11201912266QA (en) 2020-01-30
TW201909896A (zh) 2019-03-16
IL272023B1 (en) 2024-08-01
CL2019003598A1 (es) 2020-09-21
JP2022169720A (ja) 2022-11-09
AU2018309667A1 (en) 2020-02-06
BR112020000482A2 (pt) 2020-07-21
KR102692887B1 (ko) 2024-08-08
AU2018309667B2 (en) 2024-08-01
KR20200035986A (ko) 2020-04-06
IL272023A (en) 2020-03-31
US20190030022A1 (en) 2019-01-31
ZA201908495B (en) 2021-04-28
EA202090416A1 (ru) 2020-05-25
CA3069989A1 (fr) 2019-02-07
US11642339B2 (en) 2023-05-09
WO2019027881A1 (fr) 2019-02-07
UA125596C2 (uk) 2022-04-27
JP2020529415A (ja) 2020-10-08
JP7431721B2 (ja) 2024-02-15
MX2020001217A (es) 2020-03-24
CN110996961A (zh) 2020-04-10
EP3661518B1 (fr) 2024-08-28
EP3661518A1 (fr) 2020-06-10
JP7529952B2 (ja) 2024-08-07

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