MA49754A - Méthodes de traitement de symptômes de gastroparésie au moyen de velusetrag - Google Patents

Méthodes de traitement de symptômes de gastroparésie au moyen de velusetrag

Info

Publication number
MA49754A
MA49754A MA049754A MA49754A MA49754A MA 49754 A MA49754 A MA 49754A MA 049754 A MA049754 A MA 049754A MA 49754 A MA49754 A MA 49754A MA 49754 A MA49754 A MA 49754A
Authority
MA
Morocco
Prior art keywords
gastroparesia
velusetrag
methods
treating symptoms
symptoms
Prior art date
Application number
MA049754A
Other languages
English (en)
Other versions
MA49754B1 (fr
Inventor
Christopher Noel Barnes
Maria Grimaldi
Cecilia Renzulli
Giuseppe Claudio Viscomi
Original Assignee
Alfasigma Spa
Theravance Biopharma R&D Ip Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alfasigma Spa, Theravance Biopharma R&D Ip Llc filed Critical Alfasigma Spa
Publication of MA49754A publication Critical patent/MA49754A/fr
Publication of MA49754B1 publication Critical patent/MA49754B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/47042-Quinolinones, e.g. carbostyril
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Otolaryngology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicinal Preparation (AREA)
MA49754A 2017-07-31 2018-07-30 Méthodes de traitement de symptômes de gastroparésie au moyen de velusetrag MA49754B1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762539229P 2017-07-31 2017-07-31
EP18756041.2A EP3661518B1 (fr) 2017-07-31 2018-07-30 Méthodes de traitement de symptômes de gastroparésie au moyen de velusetrag
PCT/US2018/044337 WO2019027881A1 (fr) 2017-07-31 2018-07-30 Méthodes de traitement de symptômes de gastroparésie au moyen de velusetrag

Publications (2)

Publication Number Publication Date
MA49754A true MA49754A (fr) 2020-06-10
MA49754B1 MA49754B1 (fr) 2024-10-31

Family

ID=63245036

Family Applications (1)

Application Number Title Priority Date Filing Date
MA49754A MA49754B1 (fr) 2017-07-31 2018-07-30 Méthodes de traitement de symptômes de gastroparésie au moyen de velusetrag

Country Status (30)

Country Link
US (1) US11642339B2 (fr)
EP (1) EP3661518B1 (fr)
JP (2) JP7431721B2 (fr)
KR (1) KR102692887B1 (fr)
CN (1) CN110996961A (fr)
AU (1) AU2018309667B2 (fr)
BR (1) BR112020000482A2 (fr)
CA (1) CA3069989C (fr)
CL (1) CL2019003598A1 (fr)
DK (1) DK3661518T3 (fr)
EA (1) EA202090416A1 (fr)
ES (1) ES2991549T3 (fr)
FI (1) FI3661518T3 (fr)
HR (1) HRP20241359T1 (fr)
HU (1) HUE068595T2 (fr)
IL (1) IL272023B2 (fr)
LT (1) LT3661518T (fr)
MA (1) MA49754B1 (fr)
MD (1) MD3661518T2 (fr)
MX (1) MX2020001217A (fr)
PL (1) PL3661518T3 (fr)
PT (1) PT3661518T (fr)
RS (1) RS66049B1 (fr)
SG (1) SG11201912266QA (fr)
SI (1) SI3661518T1 (fr)
SM (1) SMT202400447T1 (fr)
TW (1) TW201909896A (fr)
UA (1) UA125596C2 (fr)
WO (1) WO2019027881A1 (fr)
ZA (1) ZA201908495B (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL319356A (en) 2022-09-20 2025-05-01 Alfasigma Spa Velostrag for use in the treatment of chronic pseudointestinal obstruction (CIPO)

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8309575B2 (en) 2004-04-07 2012-11-13 Theravance, Inc. Quinolinone-carboxamide compounds as 5-HT4 receptor agonists
TWI351282B (en) 2004-04-07 2011-11-01 Theravance Inc Quinolinone-carboxamide compounds as 5-ht4 recepto
US7728006B2 (en) 2004-04-07 2010-06-01 Theravance, Inc. Quinolinone-carboxamide compounds as 5-HT4 receptor agonists
TWI377206B (en) * 2005-04-06 2012-11-21 Theravance Inc Crystalline form of a quinolinone-carboxamide compound
CA2637214C (fr) 2006-02-16 2014-04-22 Theravance, Inc. Procede pour preparer des intermediaires 8-azabicylo[3.2.1]octan-3-one de composes agonistes du recepteur 5-ht4
HRP20180018T1 (hr) 2009-04-13 2018-02-09 Theravance Biopharma R&D Ip, Llc Kombinacija agonista receptora 5-ht 4 i inhibitora acetilkolinesteraze za liječenje kognitivnog poremećaja
CA2845039A1 (fr) * 2011-08-18 2013-02-21 Shire Ag Combinaisons d'un agoniste de recepteur 5-ht4 et d'un inhibiteur de pde4 pour utilisation en therapie
MX356317B (es) * 2011-08-25 2018-05-23 Evoke Pharma Inc Tratamiento de síntomas asociados a gastroparesia femenina.

Also Published As

Publication number Publication date
US11642339B2 (en) 2023-05-09
HUE068595T2 (hu) 2025-01-28
PL3661518T3 (pl) 2024-11-18
JP7529952B2 (ja) 2024-08-07
UA125596C2 (uk) 2022-04-27
MD3661518T2 (ro) 2024-12-31
JP7431721B2 (ja) 2024-02-15
CL2019003598A1 (es) 2020-09-21
KR102692887B1 (ko) 2024-08-08
EA202090416A1 (ru) 2020-05-25
HRP20241359T1 (hr) 2025-01-31
CA3069989A1 (fr) 2019-02-07
US20190030022A1 (en) 2019-01-31
AU2018309667B2 (en) 2024-08-01
FI3661518T3 (fi) 2024-10-10
ZA201908495B (en) 2021-04-28
CA3069989C (fr) 2025-05-06
AU2018309667A1 (en) 2020-02-06
DK3661518T3 (da) 2024-10-07
LT3661518T (lt) 2024-10-25
MA49754B1 (fr) 2024-10-31
EP3661518A1 (fr) 2020-06-10
SG11201912266QA (en) 2020-01-30
SMT202400447T1 (it) 2024-11-15
TW201909896A (zh) 2019-03-16
JP2020529415A (ja) 2020-10-08
MX2020001217A (es) 2020-03-24
RS66049B1 (sr) 2024-11-29
IL272023A (en) 2020-03-31
WO2019027881A1 (fr) 2019-02-07
PT3661518T (pt) 2024-11-04
ES2991549T3 (es) 2024-12-04
IL272023B1 (en) 2024-08-01
SI3661518T1 (sl) 2025-01-31
BR112020000482A2 (pt) 2020-07-21
CN110996961A (zh) 2020-04-10
IL272023B2 (en) 2024-12-01
JP2022169720A (ja) 2022-11-09
KR20200035986A (ko) 2020-04-06
EP3661518B1 (fr) 2024-08-28

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