LV13346B - Pharmaceutical tablets containing tibolone and a coating - Google Patents

Pharmaceutical tablets containing tibolone and a coating Download PDF

Info

Publication number
LV13346B
LV13346B LVP-05-72A LV050072A LV13346B LV 13346 B LV13346 B LV 13346B LV 050072 A LV050072 A LV 050072A LV 13346 B LV13346 B LV 13346B
Authority
LV
Latvia
Prior art keywords
coating
sugar
tablets
tibolone
film
Prior art date
Application number
LVP-05-72A
Other languages
English (en)
Inventor
Haan Pieter De
Lare Cornelis Elisabeth Jo Van
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of LV13346B publication Critical patent/LV13346B/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/282—Organic compounds, e.g. fats
    • A61K9/2826—Sugars or sugar alcohols, e.g. sucrose; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • A61K31/569—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone substituted in position 17 alpha, e.g. ethisterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846—Poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Preparation (AREA)

Claims (10)

  1. LV 13346 IZGUDROJUMA FORMULA 1. Ar apvalku apgādāta, stabilizēta farmaceitiska tablete, kas satur tibolonu daudzumā no 0,1 līdz 10 masas%.
  2. 2. Tablete saskaņā ar 1. punktu, pie kam apvalks ir plēves apvalks, cukura apvalks, cukura plēves apvalks vai “ietinamais” apvalks. 10
  3. 3. Tablete saskaņā ar 2. punktu, pie kam apvalks ir cukura apvalks vai cukura plēves apvalks.
  4. 4. Tablete saskaņā ar 1. vai 2. punktu, pie kam plēves apvalks satur celulozes 15 ēteri, vinilpolimēru vai želatīnu.
  5. 5. Tablete saskaņā ar 3. punktu, pie kam cukurs satur saharozi.
  6. 6. Tablete saskaņā ar jebkuru punktu no 1. līdz 5. punktam, pie kam apvalks 20 satur plastifikatoru, kas izvēlēts no grupas, kas sastāv no glicerīna, propilēnglikola un polietilēnglikola.
  7. 7. Apvalka izmantošana farmaceitiskas tabletes, kas satur tibolonu daudzumā no 0,1 līdz 10 masas%, stabilizēšanai. 25
  8. 8. Izmantošana saskaņā ar 7. punktu, pie kam apvalks ir plēves apvalks, cukura apvalks, cukura plēves apvalks vai “ietinamais” apvalks.
  9. 9. Izmantošana saskaņā ar 8. punktu, pie kam plēves apvalks satur celulozes 30 ēteri, vinilpolimēru vai želatīnu.
  10. 10. Izmantošana saskaņā ar 9. punktu, pie kam cukurs satur saharozi.
LVP-05-72A 2002-11-20 2005-06-17 Pharmaceutical tablets containing tibolone and a coating LV13346B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US42774002P 2002-11-20 2002-11-20
EP02079920 2002-11-20

Publications (1)

Publication Number Publication Date
LV13346B true LV13346B (en) 2005-12-20

Family

ID=32327854

Family Applications (1)

Application Number Title Priority Date Filing Date
LVP-05-72A LV13346B (en) 2002-11-20 2005-06-17 Pharmaceutical tablets containing tibolone and a coating

Country Status (11)

Country Link
US (1) US20060051420A1 (lv)
KR (1) KR20050085024A (lv)
AR (1) AR042083A1 (lv)
CL (1) CL2003002385A1 (lv)
CO (1) CO5590891A2 (lv)
EC (1) ECSP055811A (lv)
HR (1) HRP20050430A2 (lv)
IS (1) IS7821A (lv)
LV (1) LV13346B (lv)
NO (1) NO20052305L (lv)
PE (1) PE20040839A1 (lv)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2602730T3 (es) * 2003-09-24 2017-02-22 Novartis Consumer Health S.A. Comprimidos de diclofenaco revestidos

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3751277A (en) * 1971-03-24 1973-08-07 Dow Chemical Co Tablet coating process and composition
ATE180669T1 (de) * 1993-03-05 1999-06-15 Akzo Nobel Nv Verwendung von pregnanderivaten zur behandlung von tumoren
WO1995006462A1 (en) * 1993-08-30 1995-03-09 Warner-Lambert Company Tablet coating based on a melt-spun mixture of a saccharide and apolymer

Also Published As

Publication number Publication date
ECSP055811A (es) 2005-08-11
NO20052305L (no) 2005-06-07
PE20040839A1 (es) 2004-11-17
US20060051420A1 (en) 2006-03-09
IS7821A (is) 2005-04-25
CL2003002385A1 (es) 2005-01-14
HRP20050430A2 (en) 2005-06-30
AR042083A1 (es) 2005-06-08
CO5590891A2 (es) 2005-12-30
KR20050085024A (ko) 2005-08-29

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