LU78113A1 - Nouveaux acides 5-alkoxyimidazo(1,2-a)quinoleine-2-carboxyliques et leurs derives et composition pharmaceutique les contenant ainsi qu'un procede pour leur preparation - Google Patents

Nouveaux acides 5-alkoxyimidazo(1,2-a)quinoleine-2-carboxyliques et leurs derives et composition pharmaceutique les contenant ainsi qu'un procede pour leur preparation

Info

Publication number
LU78113A1
LU78113A1 LU78113A LU78113A LU78113A1 LU 78113 A1 LU78113 A1 LU 78113A1 LU 78113 A LU78113 A LU 78113A LU 78113 A LU78113 A LU 78113A LU 78113 A1 LU78113 A1 LU 78113A1
Authority
LU
Luxembourg
Prior art keywords
alkoxyimidazo
quinoleine
derivatives
preparation
new
Prior art date
Application number
LU78113A
Other languages
English (en)
French (fr)
Inventor
S Kadin
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of LU78113A1 publication Critical patent/LU78113A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
LU78113A 1976-09-13 1977-09-12 Nouveaux acides 5-alkoxyimidazo(1,2-a)quinoleine-2-carboxyliques et leurs derives et composition pharmaceutique les contenant ainsi qu'un procede pour leur preparation LU78113A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/722,429 US4075343A (en) 1976-09-13 1976-09-13 Anti-allergenic 5-alkoxyimidazo[1,2-A]quinoline-2-carboxylic acids and derivatives thereof

Publications (1)

Publication Number Publication Date
LU78113A1 true LU78113A1 (fr) 1979-05-23

Family

ID=24901795

Family Applications (1)

Application Number Title Priority Date Filing Date
LU78113A LU78113A1 (fr) 1976-09-13 1977-09-12 Nouveaux acides 5-alkoxyimidazo(1,2-a)quinoleine-2-carboxyliques et leurs derives et composition pharmaceutique les contenant ainsi qu'un procede pour leur preparation

Country Status (10)

Country Link
US (1) US4075343A (da)
JP (1) JPS5334800A (da)
BE (1) BE858605A (da)
DE (1) DE2740588A1 (da)
DK (1) DK149108C (da)
FR (1) FR2364213A1 (da)
GB (1) GB1542778A (da)
IE (1) IE45744B1 (da)
LU (1) LU78113A1 (da)
NL (1) NL171058C (da)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1596652A (en) * 1977-01-20 1981-08-26 Roussel Lab Ltd Imidazo (1,2-a) quinoline-2-carboxylic acid and derivatives
SE439308B (sv) * 1978-08-02 1985-06-10 Roussel Uclaf Imidazo(1,2-a)kinoxaliner och farmaceutiska kompositioner derav
SE441449B (sv) * 1979-02-09 1985-10-07 Roussel Uclaf Heterocykliska derivat och farmaceutiska kompositioner innehallande dessa derivat
FR2448541A1 (fr) * 1979-02-09 1980-09-05 Roussel Uclaf Nouveaux derives de l'oxoimidazoquinoxaline et leurs sels, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
DE3147276A1 (de) * 1981-11-28 1983-06-09 Boehringer Mannheim Gmbh, 6800 Mannheim Verfahren zur herstellung von indolderivaten, deren verwendung als wertvolle zwischenprodukte und neue 4-hydroxyindole
JPS61236965A (ja) * 1985-04-12 1986-10-22 Nissan Motor Co Ltd 中空カムシヤフト
JPS6297721A (ja) * 1985-10-22 1987-05-07 Nissan Motor Co Ltd カムシヤフトの製造方法
JPS61168319U (da) * 1986-03-14 1986-10-18
CA2021338C (en) * 1989-07-18 1996-07-16 Fumio Suzuki Imidazoquinolone derivatives
US5804686A (en) * 1996-01-19 1998-09-08 Neurogen Corporation fused pyrrolecarboxamides; a new class of GABA brain receptor ligands
US6211365B1 (en) 1996-01-19 2001-04-03 Neurogen Corporation Fused pyrrolecarboxamides; a new class of GABA brain receptor ligands
AU2218997A (en) 1996-03-22 1997-10-10 Neurogen Corporation Certain fused pyrrolecarboxamides as gaba brain receptor ligands
WO1997037999A1 (en) * 1996-04-04 1997-10-16 University Of Nebraska Board Of Regents Synthetic triple helix-forming compounds
US5723462A (en) * 1996-04-26 1998-03-03 Neurogen Corporation Certain fused pyrrolecarboxamides a new class of GABA brain receptor ligands
US20050014939A1 (en) * 1999-08-31 2005-01-20 Neurogen Corporation Fused pyrrolecarboxamides: GABA brain receptor ligands
EA200200188A1 (ru) 1999-08-31 2002-08-29 Нейроген Корпорейшн Конденсированные пирролкарбоксамиды: лиганды для гамк-мозговых рецепторов
HUP0105406A3 (en) * 2001-12-21 2003-12-29 Sanofi Aventis Imidazo[1,2-a]quinolin derivatives, process for their preparation, pharmaceutical compositions thereof and intermediates
US6989392B2 (en) * 2002-06-18 2006-01-24 Abbott Laboratories 2-Aminoquinolines as melanin concentrating hormone receptor antagonists
HUP0203976A3 (en) * 2002-11-15 2004-08-30 Sanofi Aventis Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them
CA2636043A1 (en) * 2006-01-23 2007-08-02 Amira Pharmaceuticals, Inc. Tricyclic inhibitors of 5-lipoxygenase
PE20200296A1 (es) * 2017-07-14 2020-02-06 Innate Tumor Immunity Inc Moduladores de nlrp3
CN108794485B (zh) * 2018-04-28 2020-04-24 北京施安泰医药技术开发有限公司 一类toll样受体调节剂、其药物组合物、制备方法与用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2421693A (en) * 1944-09-16 1947-06-03 Gen Aniline & Film Corp Imidazolone color formers
US3454579A (en) * 1967-08-17 1969-07-08 American Cyanamid Co Imidazo(1,5-a)quinolin-1-one and thione derivatives
GB1278272A (en) * 1969-02-19 1972-06-21 Pfizer Ltd Substituted hexahydro-imidazoquinolines
GB1347493A (en) * 1971-02-11 1974-02-27 Aspro Nicholas Ltd Benzazine derivatives
CA1033731A (en) * 1974-04-01 1978-06-27 Saul B. Kadin Process for preparing 1-oxo-1h-6-hydroxypyrimido (1,2-a)quinoline-2-carboxylic acids and derivatives
GB1484615A (en) * 1974-11-23 1977-09-01 Lepetit Spa Tricyclic n-containing derivatives

Also Published As

Publication number Publication date
DK405477A (da) 1978-03-14
NL7709442A (nl) 1978-03-15
FR2364213B1 (da) 1980-10-24
DK149108C (da) 1986-06-09
JPS5334800A (en) 1978-03-31
JPS5526143B2 (da) 1980-07-11
DE2740588A1 (de) 1978-03-16
NL171058B (nl) 1982-09-01
US4075343A (en) 1978-02-21
IE45744B1 (en) 1982-11-17
BE858605A (fr) 1978-03-13
FR2364213A1 (fr) 1978-04-07
DK149108B (da) 1986-01-27
IE45744L (en) 1978-03-13
NL171058C (nl) 1983-02-01
GB1542778A (en) 1979-03-28

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