LT2498756T - Neratinibo maleato tablečių sudėtis - Google Patents

Neratinibo maleato tablečių sudėtis

Info

Publication number
LT2498756T
LT2498756T LT10779339T LT10779339T LT2498756T LT 2498756 T LT2498756 T LT 2498756T LT 10779339 T LT10779339 T LT 10779339T LT 10779339 T LT10779339 T LT 10779339T LT 2498756 T LT2498756 T LT 2498756T
Authority
LT
Lithuania
Prior art keywords
tablet formulations
neratinib maleate
neratinib
maleate
formulations
Prior art date
Application number
LT10779339T
Other languages
English (en)
Inventor
Muhammad Ashraf
Krishnendu Ghosh
Chimanlall Goolcharran
Mainuddin Mahmud
Arwinder Singh Nagi
Original Assignee
Wyeth Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43478191&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LT2498756(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth Llc filed Critical Wyeth Llc
Publication of LT2498756T publication Critical patent/LT2498756T/lt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
LT10779339T 2009-11-09 2010-11-02 Neratinibo maleato tablečių sudėtis LT2498756T (lt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25940309P 2009-11-09 2009-11-09
PCT/IB2010/054964 WO2011055303A1 (en) 2009-11-09 2010-11-02 Tablet formulations of neratinib maleate

Publications (1)

Publication Number Publication Date
LT2498756T true LT2498756T (lt) 2019-12-10

Family

ID=43478191

Family Applications (1)

Application Number Title Priority Date Filing Date
LT10779339T LT2498756T (lt) 2009-11-09 2010-11-02 Neratinibo maleato tablečių sudėtis

Country Status (21)

Country Link
US (2) US8518446B2 (lt)
EP (3) EP3566697A1 (lt)
JP (3) JP5835883B2 (lt)
CN (2) CN102724970B (lt)
AR (2) AR078952A1 (lt)
AU (1) AU2010316683B2 (lt)
CA (1) CA2780428C (lt)
CY (1) CY1122330T1 (lt)
DK (1) DK2498756T4 (lt)
ES (1) ES2757882T5 (lt)
FI (1) FI2498756T4 (lt)
HR (1) HRP20192026T4 (lt)
HU (1) HUE046606T2 (lt)
LT (1) LT2498756T (lt)
NZ (1) NZ599763A (lt)
PL (1) PL2498756T5 (lt)
PT (1) PT2498756T (lt)
RS (1) RS59599B2 (lt)
SI (1) SI2498756T2 (lt)
TW (1) TWI466690B (lt)
WO (1) WO2011055303A1 (lt)

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CN104337782A (zh) * 2013-08-02 2015-02-11 山东新时代药业有限公司 一种甲磺酸伊马替尼片剂
EA201992707A1 (ru) 2013-11-18 2020-06-30 Глобал Блад Терапьютикс, Инк. Соединения и их применения для модуляции гемоглобина
WO2015112850A2 (en) * 2014-01-23 2015-07-30 Wenle Xia Use of psoralen derivatives and combination therapy for treatment of cell proliferation disorders
AP2016009261A0 (en) 2014-02-07 2016-06-30 Global Blood Therapeutics Inc Crystalline polymorphs of the free base of 2-hydroxy-6-((2-(1-isopropyl-1h-pyrazol-5-yl)pyridin-3-yl)methoxy)benzaldehyde
US10244991B2 (en) 2014-02-17 2019-04-02 Children's National Medical Center Method and system for providing recommendation for optimal execution of surgical procedures
MX2017001177A (es) * 2014-07-25 2017-05-01 Novartis Ag Formulacion en forma de tableta de 2-fluor-n-metil-4-[7-(quinolin- 6-ylmetil) imidazo[1,2,b] [1,2,4]triazin-2-il]benzamida.
KR102305932B1 (ko) 2015-06-29 2021-09-28 플로로놀 인코퍼레이티드 갈조류의 고체 약제학적 조성물
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CN106913529B (zh) * 2015-12-24 2020-12-04 江苏恒瑞医药股份有限公司 一种来那替尼或其可药用盐药物组合物的制备方法
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JP2020518565A (ja) * 2017-04-28 2020-06-25 アサナ バイオサイエンシズ，リミティド ライアビリティ カンパニー アトピー性皮膚炎の治療及び原薬の安定性を向上するための製剤、方法、キット、及び剤形
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Also Published As

Publication number Publication date
EP3566697A1 (en) 2019-11-13
AU2010316683A1 (en) 2012-05-24
NZ599763A (en) 2014-06-27
JP2017075192A (ja) 2017-04-20
US20110111018A1 (en) 2011-05-12
DK2498756T4 (da) 2023-03-20
US20140004184A1 (en) 2014-01-02
DK2498756T3 (da) 2019-11-25
RS59599B1 (sr) 2020-01-31
US8518446B2 (en) 2013-08-27
CN103893140B (zh) 2016-06-01
AR078952A1 (es) 2011-12-14
HRP20192026T4 (hr) 2023-03-31
CN102724970B (zh) 2014-06-25
HUE046606T2 (hu) 2020-03-30
ES2757882T5 (es) 2023-05-10
HRP20192026T1 (hr) 2020-02-07
RS59599B2 (sr) 2023-03-31
PL2498756T5 (pl) 2023-04-17
AU2010316683B2 (en) 2015-10-08
PL2498756T3 (pl) 2020-03-31
SI2498756T2 (sl) 2023-04-28
CA2780428A1 (en) 2011-05-12
JP5835883B2 (ja) 2015-12-24
SI2498756T1 (sl) 2020-01-31
TWI466690B (zh) 2015-01-01
PT2498756T (pt) 2019-11-26
CA2780428C (en) 2018-02-13
CY1122330T1 (el) 2021-01-27
EP2498756B1 (en) 2019-09-04
JP2011098964A (ja) 2011-05-19
CN103893140A (zh) 2014-07-02
CN102724970A (zh) 2012-10-10
EP2498756B2 (en) 2023-02-15
EP4066821A1 (en) 2022-10-05
WO2011055303A1 (en) 2011-05-12
FI2498756T4 (fi) 2023-03-22
JP2015091882A (ja) 2015-05-14
TW201138774A (en) 2011-11-16
EP2498756A1 (en) 2012-09-19
AR114143A2 (es) 2020-07-29
US8790708B2 (en) 2014-07-29
ES2757882T3 (es) 2020-04-30

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