KR870003090A - 아니솔 유도체 - Google Patents

아니솔 유도체 Download PDF

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Publication number
KR870003090A
KR870003090A KR1019860007443A KR860007443A KR870003090A KR 870003090 A KR870003090 A KR 870003090A KR 1019860007443 A KR1019860007443 A KR 1019860007443A KR 860007443 A KR860007443 A KR 860007443A KR 870003090 A KR870003090 A KR 870003090A
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KR
South Korea
Prior art keywords
derivative according
methoxy
methylenedioxyphenyl
anisole derivative
alkyl group
Prior art date
Application number
KR1019860007443A
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English (en)
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KR900000966B1 (ko
Inventor
요시하루 모리따
나오시 이마끼
하사오 다까야나기
유끼 다꾸마
다다시 시라사까
Original Assignee
와꼬야마 쇼에이
미쓰비시 케미칼 인더스트리스 아메리카 인코오포레이티드
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Application filed by 와꼬야마 쇼에이, 미쓰비시 케미칼 인더스트리스 아메리카 인코오포레이티드 filed Critical 와꼬야마 쇼에이
Publication of KR870003090A publication Critical patent/KR870003090A/ko
Application granted granted Critical
Publication of KR900000966B1 publication Critical patent/KR900000966B1/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/64—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

내용 없음

Description

아니솔 유도체
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (13)

  1. 하기 일반식(Ⅰ)으로 나타내지는 아니솔 유도체 ;
    상기식중 A-D는 이하에 정의하는 바와 같다.
    (1) A, B 및 C가 각각 수소원자인 경우, D는 -OH, 할로겐원자, -CO2R1(식중 R1은 저급알킬기이다) -SO2R2(식중 R2는 저급알킬기이다)
    (2) A 및 C가 각각 수소원자이고 B가 -OH인 경우, D는 -CO2R3(식중 R3는 저급알킬기이다)이며 ;
    (3) A가 수소원자이고 B 및 C가 함께 옥소기 = O를 형성하는 경우, D는 -CO2R4(식중 R4는 저급알킬기이다)이고 ; 및
    (4) B 및 C가 각각 수소원자이고 D가 할로겐원자인 경우, A는 -CHO이다.
  2. 제1항에 있어서, 각각의 R1-R4가 탄소수 1-5의 저급알킬기인 아니솔 유도체.
  3. 제2항에 있어서, 각각의 R1-R4가 탄소수 1-3의 저급알킬기인 아니솔 유도체.
  4. 제1항에 있어서, 2-(3-메톡시-4,5-메틸렌디옥시페닐)에틸알코올인 아니솔 유도체.
  5. 제1항에 있어서, 2-(3-메톡시-4,5-메틸렌디옥시페닐)에틸메탄술포네이트인 아니솔 유도체.
  6. 제1항에 있어서, 2-(3-메톡시-4,5-메틸렌디옥시페닐)에틸클로라이드인 아니솔 유도체.
  7. 제1항에 있어서, 2-(3-메톡시-4,5-메틸렌디옥시페닐)에틸브로마이드인 아니솔 유도체.
  8. 제1항에 있어서, 2-(3-메톡시-4,5-메틸렌디옥시페닐)에틸요오다이드인 아니솔 유도체.
  9. 제1항에 있어서, N-[2-(3-메톡시-4,5-메틸렌디옥시페닐)에틸]프탈이미드인 아니솔 유도체.
  10. 제1항에 있어서, 메틸3-(3-메톡시-4,5-메틸렌디옥시페닐)프로피오네이트인 아니솔 유도체.
  11. 제1항에 있어서, 메틸 3-히드록시-3-(3-메톡시-4,5-메틸렌디옥시페닐)프로피오네이트인 아니솔 유도체.
  12. 제1항에 있어서, 메틸 3-메톡시-4,5-메틸렌디옥시 벤조일 아세테이트인 아니솔 유도체.
  13. 제1항에 있어서, 2-(2-포르밀-3-메톡시-4,5-메틸렌디옥시페닐)에틸클로라이드인 아니솔 유도체.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019860007443A 1985-09-06 1986-09-05 아니솔 유도체 KR900000966B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP60197189A JPS6256484A (ja) 1985-09-06 1985-09-06 アニソ−ル誘導体
US60-197189 1985-09-06
JP197189/85 1985-09-06

Publications (2)

Publication Number Publication Date
KR870003090A true KR870003090A (ko) 1987-04-15
KR900000966B1 KR900000966B1 (ko) 1990-02-23

Family

ID=16370286

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019860007443A KR900000966B1 (ko) 1985-09-06 1986-09-05 아니솔 유도체

Country Status (6)

Country Link
US (1) US4746747A (ko)
EP (1) EP0219371B1 (ko)
JP (1) JPS6256484A (ko)
KR (1) KR900000966B1 (ko)
CA (1) CA1285571C (ko)
DE (1) DE3666818D1 (ko)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102653542B (zh) * 2011-03-02 2014-12-17 沈阳药科大学 那可丁的合成方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA733984A (en) * 1966-05-10 Merck And Co. Croweacic acid derivatives
US3922285A (en) * 1971-03-26 1975-11-25 Hoffmann La Roche Process for the methylenation of catechols

Also Published As

Publication number Publication date
EP0219371A2 (en) 1987-04-22
KR900000966B1 (ko) 1990-02-23
DE3666818D1 (de) 1989-12-14
EP0219371B1 (en) 1989-11-08
CA1285571C (en) 1991-07-02
JPS6256484A (ja) 1987-03-12
EP0219371A3 (en) 1987-11-25
US4746747A (en) 1988-05-24

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