KR860002528A - GnRH 길항물질 VI의 제법 - Google Patents

GnRH 길항물질 VI의 제법 Download PDF

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Publication number
KR860002528A
KR860002528A KR1019850006506A KR850006506A KR860002528A KR 860002528 A KR860002528 A KR 860002528A KR 1019850006506 A KR1019850006506 A KR 1019850006506A KR 850006506 A KR850006506 A KR 850006506A KR 860002528 A KR860002528 A KR 860002528A
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KR
South Korea
Prior art keywords
phe
arg
trp
gly
pro
Prior art date
Application number
KR1019850006506A
Other languages
English (en)
Korean (ko)
Inventor
워어커 베일 쥬니어(외 1) 윌리
Original Assignee
델버어드 어니스트 그랜즈
더 솔크 인스티튜트 훠 바이올로지칼 스터디이즈
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 델버어드 어니스트 그랜즈, 더 솔크 인스티튜트 훠 바이올로지칼 스터디이즈 filed Critical 델버어드 어니스트 그랜즈
Publication of KR860002528A publication Critical patent/KR860002528A/ko

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/13—Luteinizing hormone-releasing hormone; related peptides

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Endocrinology (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
KR1019850006506A 1984-09-07 1985-09-06 GnRH 길항물질 VI의 제법 KR860002528A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/648,637 US4565804A (en) 1984-09-07 1984-09-07 GnRH Antagonists VI
US648,637 1984-09-07

Publications (1)

Publication Number Publication Date
KR860002528A true KR860002528A (ko) 1986-04-26

Family

ID=24601597

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019850006506A KR860002528A (ko) 1984-09-07 1985-09-06 GnRH 길항물질 VI의 제법

Country Status (12)

Country Link
US (1) US4565804A (US07816562-20101019-C00012.png)
EP (1) EP0175506A3 (US07816562-20101019-C00012.png)
JP (1) JPS6187695A (US07816562-20101019-C00012.png)
KR (1) KR860002528A (US07816562-20101019-C00012.png)
AU (1) AU4687985A (US07816562-20101019-C00012.png)
DD (1) DD248365A5 (US07816562-20101019-C00012.png)
DK (1) DK407985A (US07816562-20101019-C00012.png)
ES (1) ES8900167A1 (US07816562-20101019-C00012.png)
GR (1) GR852148B (US07816562-20101019-C00012.png)
HU (1) HUT40144A (US07816562-20101019-C00012.png)
PH (1) PH21284A (US07816562-20101019-C00012.png)
ZA (1) ZA856449B (US07816562-20101019-C00012.png)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU193093B (en) * 1985-04-16 1987-08-28 Innofinance Process for stimulating sexual activity of birds and domestic mammalians and process for producing spermatocytes for their propagation
US4705778A (en) * 1985-10-22 1987-11-10 Sri International Orally active LHRH analogs
US4888427A (en) * 1987-04-07 1989-12-19 University Of Florida Amino acids containing dihydropyridine ring systems for site-specific delivery of peptides to the brain
US5079366A (en) * 1987-04-07 1992-01-07 University Of Florida Quarternary pyridinium salts
US4800191A (en) * 1987-07-17 1989-01-24 Schally Andrew Victor LHRH antagonists
US4935491A (en) * 1987-08-24 1990-06-19 Board Of Regents, The University Of Texas System Effective antagonists of the luteinizing hormone releasing hormone which release negligible histamine
US5171835A (en) * 1988-10-21 1992-12-15 The Administrators Of The Tulane Educational Fund LHRH antagonists
US5068221A (en) * 1989-05-09 1991-11-26 Mathias John R Treatment of motility disorders with a gnrh analog
US5084443A (en) * 1989-12-04 1992-01-28 Biomeasure, Inc. Promoting expression of acetylcholine receptors with lhrh antagonist
US5064939A (en) * 1990-02-06 1991-11-12 The Salk Institute For Biological Studies Cyclic gnrh antagonists
US5434136A (en) * 1990-12-14 1995-07-18 Mathias; John R. Treatment of motility disorders with a GNRH analog
US5656727A (en) * 1992-09-15 1997-08-12 The Administrators Of The Tulane Educational Fund Antagonists of LHRH
US5480969A (en) * 1992-09-15 1996-01-02 The Administrators Of The Tulane Educational Fund Antagonists of LHRH
DE4305225A1 (de) * 1993-02-19 1994-08-25 Asta Medica Ag Neues Herstellverfahren für Cetrorelix Lyophilisat
US6828415B2 (en) 1993-02-19 2004-12-07 Zentaris Gmbh Oligopeptide lyophilisate, their preparation and use
US5696230A (en) * 1994-08-31 1997-12-09 The Board Of Regents Of The University Of Nebraska High-affinity response-selective C-terminal analogs of C5a anaphylatoxin
US5843901A (en) 1995-06-07 1998-12-01 Advanced Research & Technology Institute LHRH antagonist peptides
EP0882736A1 (en) * 1997-06-02 1998-12-09 Laboratoire Theramex S.A. LH-RH peptide analogues, their uses and pharmaceutical compositions containing them
CA2322444A1 (en) 1998-03-05 1999-09-10 Agouron Pharmaceuticals, Inc. Non-peptide gnrh agents
US6455499B1 (en) 1999-02-23 2002-09-24 Indiana University Foundation Methods for treating disorders associated with LHRH activity
DE10024451A1 (de) * 2000-05-18 2001-11-29 Asta Medica Ag Pharmazeutische Darreichungsform für Peptide, Verfahren zu deren Herstellung und Verwendung
US6598784B2 (en) * 2000-12-20 2003-07-29 Meadwestvaco Packaging Syatens, Llc Beverage carton with strap type carrying handle
US7491702B2 (en) 2001-04-18 2009-02-17 The Open University Polypeptides related to amyloid precursor protein, pharmaceutical compositions thereof, and methods of treatment using the same
EP2316849A2 (en) * 2001-04-18 2011-05-04 The Open University Polypeptides comprising RER, derivatives and uses thereof
US7622446B2 (en) 2001-04-18 2009-11-24 The Open University Polypeptides, derivatives and uses thereof
SI2078032T1 (sl) 2006-10-24 2017-12-29 Repros Therapeutics Inc. Sestave in postopki za zaviranje proliferacije endometrija
WO2018177746A1 (en) 2017-03-31 2018-10-04 Institut National De La Sante Et De La Recherche Medicale (Inserm) A gnrh antagonist for use in the treatment of a women affected with polycystic ovary syndrome

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4234571A (en) * 1979-06-11 1980-11-18 Syntex (U.S.A.) Inc. Nonapeptide and decapeptide derivatives of luteinizing hormone releasing hormone
US4317815A (en) * 1979-06-13 1982-03-02 Coy David Howard LH-RH Antagonists
US4341767A (en) * 1980-10-06 1982-07-27 Syntex Inc. Nonapeptide and decapeptide analogs of LHRH, useful as LHRH antagonists
AU9102582A (en) * 1981-12-10 1983-06-16 David Howard Coy Lh-rh antagonists
US4481190A (en) * 1982-12-21 1984-11-06 Syntex (U.S.A.) Inc. Nonapeptide and decapeptide analogs of LHRH useful as LHRH antagonists
US4444759A (en) * 1982-07-26 1984-04-24 The Salk Institute For Biological Studies GnRH Antagonists II
EP0145032B1 (en) * 1983-08-16 1987-11-04 Akzo N.V. Lh- rh antagonists

Also Published As

Publication number Publication date
ZA856449B (en) 1986-04-30
ES546761A0 (es) 1988-04-16
DD248365A5 (de) 1987-08-05
EP0175506A3 (en) 1987-10-14
DK407985D0 (da) 1985-09-06
EP0175506A2 (en) 1986-03-26
HUT40144A (en) 1986-11-28
PH21284A (en) 1987-09-28
AU4687985A (en) 1986-03-13
ES8900167A1 (es) 1988-04-16
JPS6187695A (ja) 1986-05-06
GR852148B (US07816562-20101019-C00012.png) 1986-01-08
US4565804A (en) 1986-01-21
DK407985A (da) 1986-04-09

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A201 Request for examination
E902 Notification of reason for refusal
E601 Decision to refuse application