KR840005457A - 5-옥소-2,3,6,7-테트라히드로-5H-티아졸로(3,2-a) 피리미딘 유도체류의 제조방법 - Google Patents
5-옥소-2,3,6,7-테트라히드로-5H-티아졸로(3,2-a) 피리미딘 유도체류의 제조방법 Download PDFInfo
- Publication number
- KR840005457A KR840005457A KR1019830003385A KR830003385A KR840005457A KR 840005457 A KR840005457 A KR 840005457A KR 1019830003385 A KR1019830003385 A KR 1019830003385A KR 830003385 A KR830003385 A KR 830003385A KR 840005457 A KR840005457 A KR 840005457A
- Authority
- KR
- South Korea
- Prior art keywords
- group
- carbon atoms
- solvent
- crops
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 238000000034 method Methods 0.000 title claims 5
- GINHPDWLEHHRNI-UHFFFAOYSA-N 2,3,6,7-tetrahydro-[1,3]thiazolo[3,2-a]pyrimidin-5-one Chemical class O=C1CCN=C2SCCN12 GINHPDWLEHHRNI-UHFFFAOYSA-N 0.000 title 1
- 125000004432 carbon atom Chemical group C* 0.000 claims 9
- 125000000217 alkyl group Polymers 0.000 claims 4
- KWYUFKZDYYNOTN-UHFFFAOYSA-M Potassium hydroxide Chemical compound [OH-].[K+] KWYUFKZDYYNOTN-UHFFFAOYSA-M 0.000 claims 3
- 125000003545 alkoxy group Chemical group 0.000 claims 3
- 150000001875 compounds Chemical class 0.000 claims 3
- 125000005843 halogen group Chemical group 0.000 claims 3
- 239000000203 mixture Substances 0.000 claims 3
- 239000002904 solvent Substances 0.000 claims 3
- CQOALHPQGSYSNO-UHFFFAOYSA-N 5h-1,3-thiazol-2-imine Chemical compound N=C1SCC=N1 CQOALHPQGSYSNO-UHFFFAOYSA-N 0.000 claims 2
- RTZKZFJDLAIYFH-UHFFFAOYSA-N Diethyl ether Chemical compound CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 claims 2
- 239000002253 acid Substances 0.000 claims 2
- 239000004480 active ingredient Substances 0.000 claims 2
- 239000002585 base Substances 0.000 claims 2
- 229910052801 chlorine Inorganic materials 0.000 claims 2
- 125000001309 chloro group Chemical group Cl* 0.000 claims 2
- 125000004093 cyano group Chemical group *C#N 0.000 claims 2
- 230000003287 optical effect Effects 0.000 claims 2
- HEMHJVSKTPXQMS-UHFFFAOYSA-M sodium hydroxide Inorganic materials [OH-].[Na+] HEMHJVSKTPXQMS-UHFFFAOYSA-M 0.000 claims 2
- 125000001424 substituent group Chemical group 0.000 claims 2
- VJVCQKOMUMNIGE-UHFFFAOYSA-N 1,3-thiazolidin-2-amine Chemical compound NC1NCCS1 VJVCQKOMUMNIGE-UHFFFAOYSA-N 0.000 claims 1
- NGNBDVOYPDDBFK-UHFFFAOYSA-N 2-[2,4-di(pentan-2-yl)phenoxy]acetyl chloride Chemical compound CCCC(C)C1=CC=C(OCC(Cl)=O)C(C(C)CCC)=C1 NGNBDVOYPDDBFK-UHFFFAOYSA-N 0.000 claims 1
- REGFWZVTTFGQOJ-UHFFFAOYSA-N 4,5-dihydro-1,3-thiazol-2-amine Chemical group NC1=NCCS1 REGFWZVTTFGQOJ-UHFFFAOYSA-N 0.000 claims 1
- 229940126062 Compound A Drugs 0.000 claims 1
- 229920000742 Cotton Polymers 0.000 claims 1
- 241000219146 Gossypium Species 0.000 claims 1
- 244000020551 Helianthus annuus Species 0.000 claims 1
- 235000003222 Helianthus annuus Nutrition 0.000 claims 1
- NLDMNSXOCDLTTB-UHFFFAOYSA-N Heterophylliin A Natural products O1C2COC(=O)C3=CC(O)=C(O)C(O)=C3C3=C(O)C(O)=C(O)C=C3C(=O)OC2C(OC(=O)C=2C=C(O)C(O)=C(O)C=2)C(O)C1OC(=O)C1=CC(O)=C(O)C(O)=C1 NLDMNSXOCDLTTB-UHFFFAOYSA-N 0.000 claims 1
- DGAQECJNVWCQMB-PUAWFVPOSA-M Ilexoside XXIX Chemical group C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)OS(=O)(=O)[O-])C)C)[C@@H]2[C@]1(C)O)C)C(=O)O[C@H]6[C@@H]([C@H]([C@@H]([C@H](O6)CO)O)O)O.[Na+] DGAQECJNVWCQMB-PUAWFVPOSA-M 0.000 claims 1
- 240000007594 Oryza sativa Species 0.000 claims 1
- 235000007164 Oryza sativa Nutrition 0.000 claims 1
- 240000008042 Zea mays Species 0.000 claims 1
- 235000005824 Zea mays ssp. parviglumis Nutrition 0.000 claims 1
- 235000002017 Zea mays subsp mays Nutrition 0.000 claims 1
- -1 acetamino groups Chemical group 0.000 claims 1
- 239000000654 additive Substances 0.000 claims 1
- 230000000996 additive effect Effects 0.000 claims 1
- 229910052783 alkali metal Inorganic materials 0.000 claims 1
- 150000001340 alkali metals Chemical class 0.000 claims 1
- 125000003282 alkyl amino group Chemical group 0.000 claims 1
- 125000005530 alkylenedioxy group Chemical group 0.000 claims 1
- 125000003277 amino group Chemical group 0.000 claims 1
- 150000008064 anhydrides Chemical class 0.000 claims 1
- 229910052799 carbon Inorganic materials 0.000 claims 1
- 239000000969 carrier Substances 0.000 claims 1
- 235000005822 corn Nutrition 0.000 claims 1
- 125000004663 dialkyl amino group Chemical group 0.000 claims 1
- 230000002363 herbicidal effect Effects 0.000 claims 1
- 239000004009 herbicide Substances 0.000 claims 1
- 239000012442 inert solvent Substances 0.000 claims 1
- 150000007529 inorganic bases Chemical class 0.000 claims 1
- 239000007788 liquid Substances 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 1
- 231100001184 nonphytotoxic Toxicity 0.000 claims 1
- 150000007530 organic bases Chemical class 0.000 claims 1
- 239000003960 organic solvent Substances 0.000 claims 1
- 229940083082 pyrimidine derivative acting on arteriolar smooth muscle Drugs 0.000 claims 1
- 150000003230 pyrimidines Chemical class 0.000 claims 1
- 239000011541 reaction mixture Substances 0.000 claims 1
- 235000009566 rice Nutrition 0.000 claims 1
- 239000007787 solid Substances 0.000 claims 1
- 125000000547 substituted alkyl group Chemical group 0.000 claims 1
- 239000004094 surface-active agent Substances 0.000 claims 1
- 238000009333 weeding Methods 0.000 claims 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8213048 | 1982-07-23 | ||
| FR8213048A FR2530636A1 (fr) | 1982-07-23 | 1982-07-23 | Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR840005457A true KR840005457A (ko) | 1984-11-12 |
Family
ID=9276336
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1019830003385A Abandoned KR840005457A (ko) | 1982-07-23 | 1983-07-22 | 5-옥소-2,3,6,7-테트라히드로-5H-티아졸로(3,2-a) 피리미딘 유도체류의 제조방법 |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP0102908A1 (enExample) |
| JP (1) | JPS5933291A (enExample) |
| KR (1) | KR840005457A (enExample) |
| AU (1) | AU1713483A (enExample) |
| BR (1) | BR8303925A (enExample) |
| DK (1) | DK337583A (enExample) |
| FR (1) | FR2530636A1 (enExample) |
| GR (1) | GR78632B (enExample) |
| IL (1) | IL69140A0 (enExample) |
| MA (1) | MA19850A1 (enExample) |
| OA (1) | OA07502A (enExample) |
| PL (1) | PL243128A1 (enExample) |
| PT (1) | PT77074B (enExample) |
| ZA (1) | ZA835338B (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5749017B2 (ja) | 2008-01-22 | 2015-07-15 | ダウ アグロサイエンシィズ エルエルシー | ５−フルオロピリミジン誘導体 |
| UA106889C2 (uk) | 2009-08-07 | 2014-10-27 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні n1-ацил-5-фторпіримідинону |
| ES2471371T3 (es) | 2009-08-07 | 2014-06-26 | Dow Agrosciences Llc | Derivados de N1-sulfonil-5-fluoropirimidinona |
| UA107671C2 (en) | 2009-08-07 | 2015-02-10 | Dow Agrosciences Llc | N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives |
| UA112284C2 (uk) | 2009-08-07 | 2016-08-25 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні 5-фторпіримідинону |
| JP5781090B2 (ja) * | 2010-01-07 | 2015-09-16 | ダウ アグロサイエンシィズ エルエルシー | チアゾロ［５，４−ｄ］ピリミジン及び農薬としてのそれらの使用 |
| JP6128658B2 (ja) | 2011-08-17 | 2017-05-17 | アダマ・マクテシム・リミテッド | ５−フルオロ−４−イミノ−３−（置換）−３，４−ジヒドロピリミジン−２−（１ｈ）−オン誘導体 |
| JP6258969B2 (ja) | 2012-12-28 | 2018-01-10 | アダマ・マクテシム・リミテッド | Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキサミド誘導体 |
| DK2938194T3 (da) | 2012-12-28 | 2020-01-02 | Adama Makhteshim Ltd | N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater |
| EP3689142A1 (en) | 2012-12-28 | 2020-08-05 | Adama Makhteshim Ltd. | 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives |
| CN112094262A (zh) | 2012-12-31 | 2020-12-18 | 阿达玛马克西姆股份有限公司 | 作为杀真菌剂的化合物 |
| CN103044460B (zh) * | 2013-01-30 | 2015-02-25 | 石家庄学院 | 3,5,7-三苯基-5H-噻唑并[3,2-a]嘧啶类衍生物及应用 |
| WO2015103144A1 (en) | 2013-12-31 | 2015-07-09 | Dow Agrosciences Llc | 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation |
| CR20160345A (es) | 2013-12-31 | 2017-02-21 | Adama Makhteshim Ltd | Mezclas fungicidas sinérgicas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona e inhibidor(es) de la biosíntesis de esteroles para el control fúngico |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL129375B1 (en) * | 1980-07-24 | 1984-05-31 | Rhone Poulenc Ind | Process for preparing novel derivatives of 2,3,6,7-tetrahydro-thiazole-/3,2-a/-pyrimidin-5-one |
-
1982
- 1982-07-23 FR FR8213048A patent/FR2530636A1/fr not_active Withdrawn
-
1983
- 1983-07-01 IL IL69140A patent/IL69140A0/xx unknown
- 1983-07-04 EP EP83420112A patent/EP0102908A1/fr not_active Withdrawn
- 1983-07-19 GR GR71968A patent/GR78632B/el unknown
- 1983-07-21 OA OA58069A patent/OA07502A/xx unknown
- 1983-07-21 PL PL24312883A patent/PL243128A1/xx unknown
- 1983-07-21 ZA ZA835338A patent/ZA835338B/xx unknown
- 1983-07-21 PT PT77074A patent/PT77074B/pt unknown
- 1983-07-21 AU AU17134/83A patent/AU1713483A/en not_active Abandoned
- 1983-07-21 JP JP58133540A patent/JPS5933291A/ja active Pending
- 1983-07-22 MA MA20071A patent/MA19850A1/fr unknown
- 1983-07-22 BR BR8303925A patent/BR8303925A/pt unknown
- 1983-07-22 KR KR1019830003385A patent/KR840005457A/ko not_active Abandoned
- 1983-07-22 DK DK337583A patent/DK337583A/da not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| ZA835338B (en) | 1984-03-28 |
| OA07502A (fr) | 1985-03-31 |
| FR2530636A1 (fr) | 1984-01-27 |
| JPS5933291A (ja) | 1984-02-23 |
| DK337583D0 (da) | 1983-07-22 |
| BR8303925A (pt) | 1984-02-28 |
| PL243128A1 (en) | 1984-07-16 |
| GR78632B (enExample) | 1984-09-27 |
| PT77074A (fr) | 1983-08-01 |
| IL69140A0 (en) | 1983-11-30 |
| EP0102908A1 (fr) | 1984-03-14 |
| AU1713483A (en) | 1984-01-26 |
| DK337583A (da) | 1984-01-24 |
| MA19850A1 (fr) | 1984-04-01 |
| PT77074B (fr) | 1986-04-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PA0109 | Patent application |
Patent event code: PA01091R01D Comment text: Patent Application Patent event date: 19830722 |
|
| PG1501 | Laying open of application | ||
| PC1902 | Submission of document of abandonment before decision of registration | ||
| SUBM | Surrender of laid-open application requested |