KR20250005055A - 아스피린 및 기타 nsaid의 고 침투성 전구약물을 이용한 심혈관 질환의 예방 또는 치료 - Google Patents
아스피린 및 기타 nsaid의 고 침투성 전구약물을 이용한 심혈관 질환의 예방 또는 치료 Download PDFInfo
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- KR20250005055A KR20250005055A KR1020247027368A KR20247027368A KR20250005055A KR 20250005055 A KR20250005055 A KR 20250005055A KR 1020247027368 A KR1020247027368 A KR 1020247027368A KR 20247027368 A KR20247027368 A KR 20247027368A KR 20250005055 A KR20250005055 A KR 20250005055A
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- substituted
- unsubstituted
- acid
- diethylamino
- ethyl
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Cardiology (AREA)
- Dermatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2022/072270 | 2022-01-17 | ||
| CN2022072270 | 2022-01-17 | ||
| PCT/CN2023/071973 WO2023134732A1 (en) | 2022-01-17 | 2023-01-12 | Prevention or treatment of cardiovascular diseases with high penetration prodrugs of aspirin and other nsaids |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20250005055A true KR20250005055A (ko) | 2025-01-09 |
Family
ID=87280122
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020247027368A Pending KR20250005055A (ko) | 2022-01-17 | 2023-01-12 | 아스피린 및 기타 nsaid의 고 침투성 전구약물을 이용한 심혈관 질환의 예방 또는 치료 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20250099491A1 (https=) |
| EP (1) | EP4465993A4 (https=) |
| JP (1) | JP2025504447A (https=) |
| KR (1) | KR20250005055A (https=) |
| CN (1) | CN118632699A (https=) |
| AU (1) | AU2023206720A1 (https=) |
| CA (1) | CA3252370A1 (https=) |
| IL (1) | IL314290A (https=) |
| TW (1) | TW202339711A (https=) |
| WO (1) | WO2023134732A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN118373749A (zh) * | 2024-04-29 | 2024-07-23 | 四川施成收生态科技有限公司 | 一种含有2-羟基苯甲酸-2-（二乙氨基）乙酯结构的化合物制备及应用 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH399486A (fr) * | 1962-10-02 | 1965-09-30 | Biosedra Lab | Procédé de préparation de nouvelles salicylamides |
| CA2656858C (en) * | 2006-07-09 | 2016-01-19 | Techfields Biochem Co. Ltd | Positively charged water-soluble prodrugs of acetylsalicylic acid |
| CN101500983B (zh) * | 2006-07-26 | 2015-09-16 | 于崇曦 | 具有快速皮肤穿透速度的带正电荷的水溶性二氟尼柳及相关化合物的前药 |
| CN111012914A (zh) * | 2012-01-18 | 2020-04-17 | 苏州泰飞尔医药有限公司 | 治疗肺部疾病的高穿透力前药组合物和医药组合物 |
| CN112521305B (zh) * | 2013-03-15 | 2023-04-25 | 苏州泰飞尔医药有限公司 | 治疗帕金森疾病的新型高穿透力药物及其药物组合物 |
-
2023
- 2023-01-12 AU AU2023206720A patent/AU2023206720A1/en active Pending
- 2023-01-12 JP JP2024542395A patent/JP2025504447A/ja active Pending
- 2023-01-12 CA CA3252370A patent/CA3252370A1/en active Pending
- 2023-01-12 KR KR1020247027368A patent/KR20250005055A/ko active Pending
- 2023-01-12 US US18/729,497 patent/US20250099491A1/en active Pending
- 2023-01-12 CN CN202380017401.5A patent/CN118632699A/zh active Pending
- 2023-01-12 IL IL314290A patent/IL314290A/en unknown
- 2023-01-12 WO PCT/CN2023/071973 patent/WO2023134732A1/en not_active Ceased
- 2023-01-12 EP EP23740073.4A patent/EP4465993A4/en active Pending
- 2023-01-16 TW TW112101788A patent/TW202339711A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2025504447A (ja) | 2025-02-12 |
| US20250099491A1 (en) | 2025-03-27 |
| WO2023134732A1 (en) | 2023-07-20 |
| TW202339711A (zh) | 2023-10-16 |
| EP4465993A4 (en) | 2026-01-07 |
| WO2023134732A9 (en) | 2024-08-08 |
| EP4465993A1 (en) | 2024-11-27 |
| AU2023206720A1 (en) | 2024-08-29 |
| IL314290A (en) | 2024-09-01 |
| CN118632699A (zh) | 2024-09-10 |
| CA3252370A1 (en) | 2023-07-20 |
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