KR20120042766A - 지방산 아마이드 가수분해효소 억제제로서의 이속사졸린 - Google Patents

지방산 아마이드 가수분해효소 억제제로서의 이속사졸린 Download PDF

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KR20120042766A
KR20120042766A KR1020117030377A KR20117030377A KR20120042766A KR 20120042766 A KR20120042766 A KR 20120042766A KR 1020117030377 A KR1020117030377 A KR 1020117030377A KR 20117030377 A KR20117030377 A KR 20117030377A KR 20120042766 A KR20120042766 A KR 20120042766A
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South Korea
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alkyl
certain embodiments
aryl
independently
alkenyl
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Korean (ko)
Inventor
마크 엘 벤크
알프레도 씨 카스트로
로렌스 케이 찬
캐서린 에이 에반스
루이스 그레니어
마이클 제이 그로간
이브스 르블랑
타오 리우
스테판 페루소
다니엘 에이 스나이더
토마스 티 티비츠
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인피니티 파마슈티칼스, 인코포레이티드
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Publication of KR20120042766A publication Critical patent/KR20120042766A/ko
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Reproductive Health (AREA)
  • Dermatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pulmonology (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Pregnancy & Childbirth (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Otolaryngology (AREA)
  • Child & Adolescent Psychology (AREA)
KR1020117030377A 2009-05-18 2010-05-18 지방산 아마이드 가수분해효소 억제제로서의 이속사졸린 Withdrawn KR20120042766A (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US17928309P 2009-05-18 2009-05-18
US17928009P 2009-05-18 2009-05-18
US17928509P 2009-05-18 2009-05-18
US61/179,283 2009-05-18
US61/179,280 2009-05-18
US61/179,285 2009-05-18

Publications (1)

Publication Number Publication Date
KR20120042766A true KR20120042766A (ko) 2012-05-03

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Country Status (16)

Country Link
EP (1) EP2432771A4 (https=)
JP (1) JP2012527467A (https=)
KR (1) KR20120042766A (https=)
CN (1) CN102459202B (https=)
AR (1) AR076687A1 (https=)
AU (1) AU2010249674A1 (https=)
BR (1) BRPI1011049A2 (https=)
CA (1) CA2762527A1 (https=)
IL (1) IL216420A0 (https=)
MX (1) MX2011012263A (https=)
NZ (2) NZ596585A (https=)
RU (1) RU2539595C2 (https=)
SG (2) SG176168A1 (https=)
TW (1) TW201043620A (https=)
WO (1) WO2010135360A1 (https=)
ZA (1) ZA201108657B (https=)

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JP5373613B2 (ja) 2006-10-16 2013-12-18 バイオノミクス リミテッド 新規な抗不安薬化合物
US8927551B2 (en) 2009-05-18 2015-01-06 Infinity Pharmaceuticals, Inc. Isoxazolines as inhibitors of fatty acid amide hydrolase
US9149465B2 (en) 2009-05-18 2015-10-06 Infinity Pharmaceuticals, Inc. Isoxazolines as inhibitors of fatty acid amide hydrolase
WO2011085216A2 (en) 2010-01-08 2011-07-14 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating parkinson's disease and restless legs syndrome
WO2011123719A2 (en) 2010-03-31 2011-10-06 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating abdominal, visceral and pelvic pain
CA2828780A1 (en) 2011-03-02 2012-09-07 Bionomics Limited Novel small-molecules as therapeutics
EP2707367B1 (en) 2011-05-12 2019-10-09 Bionomics Limited Methods for preparing naphthyridines
WO2018112843A1 (en) 2016-12-22 2018-06-28 Merck Sharp & Dohme Corp. Heteroaryl piperidine ether allosteric modulators of the m4 muscarinic acetylcholine receptor
CA3072420A1 (en) * 2017-08-10 2019-02-14 Taisho Pharmaceutical Co., Ltd. Pyridine compound substituted with azole
US10485790B1 (en) 2018-09-13 2019-11-26 Syneurx International (Taiwan) Corp. Salts of cycloserine compounds and applications thereof
WO2020081572A1 (en) * 2018-10-15 2020-04-23 Dana-Farber Cancer Institute, Inc. Transcriptional enhanced associate domain (tead) transcription factor inhibitors and uses thereof
CN110016142B (zh) * 2019-04-30 2021-08-03 合肥工业大学 一种含嘧啶硼酸结构的硅油及其制备方法
WO2020243423A1 (en) 2019-05-31 2020-12-03 Ikena Oncology, Inc. Tead inhibitors and uses thereof
KR20220030222A (ko) 2019-05-31 2022-03-10 이케나 온콜로지, 인코포레이티드 Tead 억제제 및 이의 용도
KR20230145066A (ko) 2021-02-11 2023-10-17 바스프 에스이 치환된 이속사졸린 유도체
EP4043444A1 (en) 2021-02-11 2022-08-17 Basf Se Substituted isoxazoline derivatives
CN116888101A (zh) * 2021-02-11 2023-10-13 巴斯夫欧洲公司 取代的异噁唑啉衍生物
JP2024539280A (ja) 2021-10-25 2024-10-28 カイメラ セラピューティクス， インコーポレイテッド Ｔｙｋ２分解剤およびそれらの使用
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NZ619076A (en) 2015-07-31
MX2011012263A (es) 2012-01-30
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SG176168A1 (en) 2011-12-29
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TW201043620A (en) 2010-12-16
CN102459202A (zh) 2012-05-16
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NZ596585A (en) 2014-01-31
BRPI1011049A2 (pt) 2019-09-24
CN102459202B (zh) 2015-11-25
JP2012527467A (ja) 2012-11-08
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