KR20060125812A - 니코틴성 아세틸콜린 수용체 리간드 - Google Patents
니코틴성 아세틸콜린 수용체 리간드 Download PDFInfo
- Publication number
- KR20060125812A KR20060125812A KR1020067012361A KR20067012361A KR20060125812A KR 20060125812 A KR20060125812 A KR 20060125812A KR 1020067012361 A KR1020067012361 A KR 1020067012361A KR 20067012361 A KR20067012361 A KR 20067012361A KR 20060125812 A KR20060125812 A KR 20060125812A
- Authority
- KR
- South Korea
- Prior art keywords
- disease
- oxygen
- sulfur
- disorder
- atoms
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 0 *=C(NC1C(CC2)CCN2C1)[Al]*[Al] Chemical compound *=C(NC1C(CC2)CCN2C1)[Al]*[Al] 0.000 description 1
- UGMNQKTZCMYUTJ-UHFFFAOYSA-N COC(c([s]c(-c1cccnc1)c1)c1F)=O Chemical compound COC(c([s]c(-c1cccnc1)c1)c1F)=O UGMNQKTZCMYUTJ-UHFFFAOYSA-N 0.000 description 1
- CBDZTEBMHMCYCY-UHFFFAOYSA-N OC(c(cc(cc1)-c2ccccc2)c1F)=O Chemical compound OC(c(cc(cc1)-c2ccccc2)c1F)=O CBDZTEBMHMCYCY-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Neurology (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US53171203P | 2003-12-22 | 2003-12-22 | |
| US60/531,712 | 2003-12-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20060125812A true KR20060125812A (ko) | 2006-12-06 |
Family
ID=34710246
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020067012361A Withdrawn KR20060125812A (ko) | 2003-12-22 | 2004-12-20 | 니코틴성 아세틸콜린 수용체 리간드 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20070270458A1 (https=) |
| EP (1) | EP1699786A1 (https=) |
| JP (1) | JP2007515478A (https=) |
| KR (1) | KR20060125812A (https=) |
| CN (1) | CN1914201A (https=) |
| AU (1) | AU2004303737A1 (https=) |
| BR (1) | BRPI0417927A (https=) |
| CA (1) | CA2550844A1 (https=) |
| IL (1) | IL176071A0 (https=) |
| MX (1) | MXPA06007026A (https=) |
| NO (1) | NO20063356L (https=) |
| SG (1) | SG149052A1 (https=) |
| WO (1) | WO2005061494A1 (https=) |
| ZA (1) | ZA200605074B (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE20130775A1 (es) | 2010-05-27 | 2013-07-21 | Targacept Inc | Antagonistas no competitivos de receptores nicotinicos |
| WO2012007500A2 (de) | 2010-07-15 | 2012-01-19 | Bayer Cropscience Ag | Neue heterocyclische verbindungen als schädlingsbekämpfungsmittel |
| WO2021174174A1 (en) * | 2020-02-28 | 2021-09-02 | Remix Therapeutics Inc. | Thiophenyl derivatives useful for modulating nucleic acid splicing |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2529548A1 (fr) * | 1982-07-02 | 1984-01-06 | Delalande Sa | Nouveaux derives de l'amino-3 quinuclidine, leur procede et leur application en therapeutique |
| DE3852145T2 (de) * | 1987-02-18 | 1995-04-06 | Beecham Group Plc | Indolderivate, Verfahren zu deren Herstellung und pharmazeutische Präparate, die diese enthalten. |
| SE0000540D0 (sv) * | 2000-02-18 | 2000-02-18 | Astrazeneca Ab | New compounds |
| WO2002017358A2 (en) * | 2000-08-21 | 2002-02-28 | Pharmacia & Upjohn Company | Quinuclidine-substituted heteroaryl moieties for treatment of disease (nicotinic acetylcholine receptor antagonists) |
| US6599916B2 (en) * | 2000-08-21 | 2003-07-29 | Pharmacia & Upjohn Company | Quinuclidine-substituted heteroaryl moieties for treatment of disease |
| EP1311505A2 (en) * | 2000-08-21 | 2003-05-21 | PHARMACIA & UPJOHN COMPANY | Quinuclidine-substituted heteroaryl moieties for treatment of disease ( nicotinic acetylcholine receptor ligands ) |
| DE10156719A1 (de) * | 2001-11-19 | 2003-05-28 | Bayer Ag | Heteroarylcarbonsäureamide |
-
2004
- 2004-12-20 MX MXPA06007026A patent/MXPA06007026A/es unknown
- 2004-12-20 CN CNA2004800412932A patent/CN1914201A/zh active Pending
- 2004-12-20 JP JP2006546908A patent/JP2007515478A/ja not_active Abandoned
- 2004-12-20 BR BRPI0417927-7A patent/BRPI0417927A/pt not_active IP Right Cessation
- 2004-12-20 AU AU2004303737A patent/AU2004303737A1/en not_active Abandoned
- 2004-12-20 WO PCT/SE2004/001940 patent/WO2005061494A1/en not_active Ceased
- 2004-12-20 EP EP04809113A patent/EP1699786A1/en not_active Withdrawn
- 2004-12-20 US US10/583,582 patent/US20070270458A1/en not_active Abandoned
- 2004-12-20 KR KR1020067012361A patent/KR20060125812A/ko not_active Withdrawn
- 2004-12-20 CA CA002550844A patent/CA2550844A1/en not_active Abandoned
- 2004-12-20 SG SG200809495-5A patent/SG149052A1/en unknown
-
2006
- 2006-05-31 IL IL176071A patent/IL176071A0/en unknown
- 2006-06-20 ZA ZA200605074A patent/ZA200605074B/en unknown
- 2006-07-19 NO NO20063356A patent/NO20063356L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CN1914201A (zh) | 2007-02-14 |
| AU2004303737A1 (en) | 2005-07-07 |
| CA2550844A1 (en) | 2005-07-07 |
| BRPI0417927A (pt) | 2007-04-17 |
| SG149052A1 (en) | 2009-01-29 |
| WO2005061494A1 (en) | 2005-07-07 |
| ZA200605074B (en) | 2007-05-30 |
| US20070270458A1 (en) | 2007-11-22 |
| IL176071A0 (en) | 2006-10-05 |
| JP2007515478A (ja) | 2007-06-14 |
| MXPA06007026A (es) | 2006-08-31 |
| EP1699786A1 (en) | 2006-09-13 |
| NO20063356L (no) | 2006-09-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PA0105 | International application |
Patent event date: 20060621 Patent event code: PA01051R01D Comment text: International Patent Application |
|
| PG1501 | Laying open of application | ||
| PC1203 | Withdrawal of no request for examination | ||
| WITN | Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid |