KR20020082136A - 선택적 ｐｄｅ10 억제제의 치료 용도 - Google Patents
선택적 ｐｄｅ10 억제제의 치료 용도 Download PDFInfo
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- KR20020082136A KR20020082136A KR1020020021667A KR20020021667A KR20020082136A KR 20020082136 A KR20020082136 A KR 20020082136A KR 1020020021667 A KR1020020021667 A KR 1020020021667A KR 20020021667 A KR20020021667 A KR 20020021667A KR 20020082136 A KR20020082136 A KR 20020082136A
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| DE10130151A1 (de) * | 2001-06-22 | 2003-01-02 | Bayer Ag | Neue Verwendung für PDE 10A-Inhibitoren |
| DE10230604A1 (de) * | 2002-07-08 | 2004-01-29 | Bayer Ag | Heterocyclisch substituierte Imidazotriazine |
| US20060110783A1 (en) * | 2002-11-08 | 2006-05-25 | Bayer Healthcare Ag | Diagnostics and therapeutics for diseases associated with human phosphodiesterase 10a (pde10a) |
| EP1562588A4 (en) * | 2002-11-15 | 2007-10-31 | Merck & Co Inc | USE OF PDE4 INHIBITORS AS ADDITIONAL TREATMENT IN PSYCHIATRICAL DISEASES |
| US8338420B1 (en) | 2002-12-04 | 2012-12-25 | Mitsubishi Tanabe Pharma Corporation | Treatment of Parkinson's disease and enhancement of dopamine signal using PDE 10 inhibitor |
| MXPA05013553A (es) * | 2003-06-30 | 2006-03-09 | Altana Pharma Ag | Pirrolodihidroisoquinolinas como inhibidores de pde10. |
| EP1641457B1 (en) * | 2003-06-30 | 2009-08-05 | Nycomed GmbH | Pyrrolo-dihydroisoquinoline derivatives as pde10 inhibitors |
| BRPI0511854A (pt) * | 2004-06-07 | 2008-01-15 | Pfizer Prod Inc | inibição de fosfodiestearase 10 como tratamento para condições relacionados com a obesidade e relacionadas a sìndrome metabólica |
| US7576080B2 (en) * | 2004-12-23 | 2009-08-18 | Memory Pharmaceuticals Corporation | Certain thienopyrimidine derivatives as phosphodiesterase 10 inhibitors |
| DE602006006544D1 (de) * | 2005-01-12 | 2009-06-10 | Nycomed Gmbh | Neue pyrrolodihydroisochinoline als pde10-inhibitoren |
| EP1940819A1 (en) * | 2005-08-16 | 2008-07-09 | Memory Pharmaceuticals Corporation | Phosphodiesterase 10 inhibitors |
| TW200815436A (en) * | 2006-05-30 | 2008-04-01 | Elbion Ag | 4-amino-pyrido[3,2-e]pyrazines, their use as inhibitors of phosphodiesterase 10, and processes for preparing them |
| TW200817400A (en) | 2006-05-30 | 2008-04-16 | Elbion Ag | Pyrido [3,2-e] pyrazines, their use as inhibitors of phosphodiesterase 10, and processes for preparing them |
| US20100056791A1 (en) * | 2006-09-01 | 2010-03-04 | Yasushi Kohno | Pyrazolopyridine carboxamide derivative and phosphodiesterase (pde) inhibitor containing the same |
| CA2661992A1 (en) * | 2006-09-06 | 2008-03-13 | Kyorin Pharmaceutical Co., Ltd. | Pyrazolopyridine derivative and phosphodiesterase (pde) inhibitor containing the same as active ingredient |
| US7786139B2 (en) * | 2006-11-21 | 2010-08-31 | Omeros Corporation | PDE10 inhibitors and related compositions and methods |
| US7858620B2 (en) | 2007-09-19 | 2010-12-28 | H. Lundbeck A/S | Cyanoisoquinoline |
| EP2348018A4 (en) | 2008-09-25 | 2012-04-25 | Kyorin Seiyaku Kk | HETEROCYCLIC BIARYL DERIVATIVE AND PDE INHIBITOR CONTAINING ACTIVE SUBSTANCE |
| EP2351748A4 (en) | 2008-10-09 | 2012-03-21 | Kyorin Seiyaku Kk | ISOCHINOLINE DERIVATIVES AND THESE PDE INHIBITORS CONTAINING ACTIVE SUBSTANCE |
| PT2443105E (pt) | 2009-06-19 | 2015-01-14 | Lundbeck & Co As H | Novo derivado de fenilimidazole como inibidor da enzima pde10a |
| TWI481607B (zh) | 2009-12-17 | 2015-04-21 | Lundbeck & Co As H | 作為ｐｄｅ１０ａ酵素抑制劑的２－芳基咪唑衍生物 |
| TWI487705B (zh) | 2009-12-17 | 2015-06-11 | Lundbeck & Co As H | 作為ｐｄｅ１０ａ酵素抑制劑之雜芳香族芳基三唑衍生物 |
| TW201200516A (en) | 2009-12-17 | 2012-01-01 | Lundbeck & Co As H | Phenylimidazole derivatives comprising an ethynylene linker as PDE10A enzyme inhibitors |
| TWI485151B (zh) | 2009-12-17 | 2015-05-21 | Lundbeck & Co As H | 作為ｐｄｅ１０ａ酵素抑制劑之雜芳香族苯基咪唑衍生物 |
| PH12012501643A1 (en) | 2010-02-26 | 2017-07-19 | Mitsubishi Tanabe Pharma Corp | Pyrazolopyrimidine compounds and their use as pde 10 inhibitors |
| TW201215607A (en) | 2010-07-02 | 2012-04-16 | Lundbeck & Co As H | Aryl-and heteroarylamid derivatives as PDE10A enzyme inhibitor |
| TW201206935A (en) | 2010-07-16 | 2012-02-16 | Lundbeck & Co As H | Triazolo-and pyrazoloquinazoline derivatives as PDE10A enzyme inhibitor |
| JO3089B1 (ar) | 2010-11-19 | 2017-03-15 | H Lundbeck As | مشتقات ايميدازول كمثبطات لانزيمات pde10a |
| WO2013127817A1 (en) | 2012-02-27 | 2013-09-06 | H. Lundbeck A/S | Imidazole derivatives as pde10a enzyme inhibitors |
| US10154988B2 (en) | 2012-11-14 | 2018-12-18 | The Johns Hopkins University | Methods and compositions for treating schizophrenia |
| TR201904614T4 (en) | 2013-02-27 | 2019-05-21 | Mochida Pharm Co Ltd | Novel pyrazole derivative. |
| US10039764B2 (en) | 2013-07-12 | 2018-08-07 | University Of South Alabama | Treatment and diagnosis of cancer and precancerous conditions using PDE10A inhibitors and methods to measure PDE10A expression |
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2002
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- 2002-04-17 EP EP02252729A patent/EP1250923A3/en not_active Withdrawn
- 2002-04-18 AU AU34409/02A patent/AU3440902A/en not_active Abandoned
- 2002-04-18 CA CA002382326A patent/CA2382326A1/en not_active Abandoned
- 2002-04-19 HU HU0201310A patent/HUP0201310A3/hu unknown
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- 2002-04-19 JP JP2002117635A patent/JP3839343B2/ja not_active Expired - Fee Related
- 2002-04-19 US US10/126,113 patent/US20030008806A1/en not_active Abandoned
- 2002-04-19 KR KR1020020021667A patent/KR20020082136A/ko not_active Ceased
- 2002-04-19 PL PL02353535A patent/PL353535A1/xx not_active Application Discontinuation
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| US5556862A (en) * | 1993-12-28 | 1996-09-17 | Nippon Zoki Pharmaceutical Co., Ltd. | Pharmaceutical compositions containing isoquinoline derivatives |
| WO1995019173A1 (en) * | 1994-01-14 | 1995-07-20 | EGIS Gyógyszergyár Rt. | Pharmaceutical compositions |
| EP0755685A1 (en) * | 1994-04-15 | 1997-01-29 | Meiji Seika Kaisha Ltd. | Medicinal composition for treating tardive dyskinesia and utilization thereof |
| KR970061253A (ko) * | 1996-02-28 | 1997-09-12 | 정명식 | 이소퀴놀린 화합물을 함유하는 항우울제 |
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Also Published As
| Publication number | Publication date |
|---|---|
| ZA200203123B (en) | 2003-10-20 |
| PL353535A1 (en) | 2002-10-21 |
| HUP0201310A2 (hu) | 2003-02-28 |
| CN1382490A (zh) | 2002-12-04 |
| EP1250923A2 (en) | 2002-10-23 |
| AU3440902A (en) | 2002-10-24 |
| CN1840181A (zh) | 2006-10-04 |
| JP2002363103A (ja) | 2002-12-18 |
| HUP0201310A3 (en) | 2008-10-28 |
| US20030008806A1 (en) | 2003-01-09 |
| HU0201310D0 (enExample) | 2002-06-29 |
| JP3839343B2 (ja) | 2006-11-01 |
| CA2382326A1 (en) | 2002-10-20 |
| KR20060002003A (ko) | 2006-01-06 |
| HK1048070A1 (zh) | 2003-03-21 |
| EP1250923A3 (en) | 2003-01-15 |
| NZ518478A (en) | 2004-04-30 |
| IL149106A0 (en) | 2002-11-10 |
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