KR20010089253A - 시클릭 에스터 또는 아마이드 유도체 - Google Patents

시클릭 에스터 또는 아마이드 유도체 Download PDF

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Publication number
KR20010089253A
KR20010089253A KR1020017003246A KR20017003246A KR20010089253A KR 20010089253 A KR20010089253 A KR 20010089253A KR 1020017003246 A KR1020017003246 A KR 1020017003246A KR 20017003246 A KR20017003246 A KR 20017003246A KR 20010089253 A KR20010089253 A KR 20010089253A
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KR
South Korea
Prior art keywords
compound
group
individually
substituted
fkbp
Prior art date
Application number
KR1020017003246A
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English (en)
Korean (ko)
Inventor
그레고리에스 해밀턴
데이비드씨 림버그
Original Assignee
다니엘 피. 맥컬럼
지피아이 엔아이엘 홀딩스, 인코포레이티드
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by 다니엘 피. 맥컬럼, 지피아이 엔아이엘 홀딩스, 인코포레이티드 filed Critical 다니엘 피. 맥컬럼
Publication of KR20010089253A publication Critical patent/KR20010089253A/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
KR1020017003246A 1998-09-21 1999-09-17 시클릭 에스터 또는 아마이드 유도체 KR20010089253A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US09/157,566 US6462072B1 (en) 1998-09-21 1998-09-21 Cyclic ester or amide derivatives
US09/157,566 1998-09-21
PCT/US1999/021290 WO2000017161A1 (en) 1998-09-21 1999-09-17 Cyclic ester or amide derivatives

Publications (1)

Publication Number Publication Date
KR20010089253A true KR20010089253A (ko) 2001-09-29

Family

ID=22564303

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020017003246A KR20010089253A (ko) 1998-09-21 1999-09-17 시클릭 에스터 또는 아마이드 유도체

Country Status (11)

Country Link
US (1) US6462072B1 (US06462072-20021008-C00001.png)
EP (1) EP1115703A1 (US06462072-20021008-C00001.png)
JP (1) JP2002526474A (US06462072-20021008-C00001.png)
KR (1) KR20010089253A (US06462072-20021008-C00001.png)
CN (1) CN1323294A (US06462072-20021008-C00001.png)
AU (1) AU6390599A (US06462072-20021008-C00001.png)
CA (1) CA2341036A1 (US06462072-20021008-C00001.png)
HU (1) HUP0103565A3 (US06462072-20021008-C00001.png)
IL (1) IL141552A0 (US06462072-20021008-C00001.png)
WO (1) WO2000017161A1 (US06462072-20021008-C00001.png)
ZA (1) ZA200101934B (US06462072-20021008-C00001.png)

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EP1434774A1 (en) 2001-10-10 2004-07-07 Sugen, Inc. 3-(4-substituted heterocyclyl)-pyrrol-2-ylmethylidene)-2-indolinone derivatives as protein kinase inhibitors
US20060063828A1 (en) * 2004-06-28 2006-03-23 Weingarten M D 1,2-Bis-(substituted-phenyl)-2-propen-1-ones and pharmaceutical compositions thereof

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Also Published As

Publication number Publication date
IL141552A0 (en) 2002-03-10
HUP0103565A3 (en) 2002-02-28
JP2002526474A (ja) 2002-08-20
ZA200101934B (en) 2002-09-18
WO2000017161A1 (en) 2000-03-30
HUP0103565A2 (hu) 2002-01-28
US6462072B1 (en) 2002-10-08
AU6390599A (en) 2000-04-10
CA2341036A1 (en) 2000-03-30
EP1115703A1 (en) 2001-07-18
CN1323294A (zh) 2001-11-21

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