KR102890891B1 - 지질 합성의 헤테로사이클릭 조절인자 - Google Patents

지질 합성의 헤테로사이클릭 조절인자

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Publication number
KR102890891B1
KR102890891B1 KR1020247007294A KR20247007294A KR102890891B1 KR 102890891 B1 KR102890891 B1 KR 102890891B1 KR 1020247007294 A KR1020247007294 A KR 1020247007294A KR 20247007294 A KR20247007294 A KR 20247007294A KR 102890891 B1 KR102890891 B1 KR 102890891B1
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South Korea
Prior art keywords
alkyl
halogen
cycloalkyl
straight
membered heterocycle
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KR1020247007294A
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English (en)
Korean (ko)
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KR20240036703A (ko
Inventor
더글라스 아이. 버클리
그레고리 듀크
앨런 에스. 와그먼
마크 에반칙
로버트 에스. 맥도웰
Original Assignee
새지메트 바이오사이언시스, 인코포레이티드
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Priority claimed from US15/349,960 external-priority patent/US20170119786A1/en
Application filed by 새지메트 바이오사이언시스, 인코포레이티드 filed Critical 새지메트 바이오사이언시스, 인코포레이티드
Priority to KR1020257039033A priority Critical patent/KR20250169632A/ko
Publication of KR20240036703A publication Critical patent/KR20240036703A/ko
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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