KR102575344B1 - 항-섬유화 요법을 투여하는 방법 - Google Patents

항-섬유화 요법을 투여하는 방법 Download PDF

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Publication number
KR102575344B1
KR102575344B1 KR1020227034429A KR20227034429A KR102575344B1 KR 102575344 B1 KR102575344 B1 KR 102575344B1 KR 1020227034429 A KR1020227034429 A KR 1020227034429A KR 20227034429 A KR20227034429 A KR 20227034429A KR 102575344 B1 KR102575344 B1 KR 102575344B1
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KR20220139450A (ko
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린 판
도로시 쓰윙 청
제프리 마크 해리스
인디아나 스트롬붐
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제넨테크, 인크.
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4355—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having oxygen as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1020227034429A 2016-11-30 2017-11-29 항-섬유화 요법을 투여하는 방법 Active KR102575344B1 (ko)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1020237029765A KR20230129628A (ko) 2016-11-30 2017-11-29 항-섬유화 요법을 투여하는 방법

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US201662428163P 2016-11-30 2016-11-30
US62/428,163 2016-11-30
US201662432425P 2016-12-09 2016-12-09
US62/432,425 2016-12-09
KR1020197013644A KR20190089862A (ko) 2016-11-30 2017-11-29 항-섬유화 요법을 투여하는 방법
PCT/US2017/063549 WO2018102323A1 (en) 2016-11-30 2017-11-29 Methods of administering anti-fibrotic therapy

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020197013644A Division KR20190089862A (ko) 2016-11-30 2017-11-29 항-섬유화 요법을 투여하는 방법

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020237029765A Division KR20230129628A (ko) 2016-11-30 2017-11-29 항-섬유화 요법을 투여하는 방법

Publications (2)

Publication Number Publication Date
KR20220139450A KR20220139450A (ko) 2022-10-14
KR102575344B1 true KR102575344B1 (ko) 2023-09-06

Family

ID=60655162

Family Applications (3)

Application Number Title Priority Date Filing Date
KR1020227034429A Active KR102575344B1 (ko) 2016-11-30 2017-11-29 항-섬유화 요법을 투여하는 방법
KR1020237029765A Ceased KR20230129628A (ko) 2016-11-30 2017-11-29 항-섬유화 요법을 투여하는 방법
KR1020197013644A Ceased KR20190089862A (ko) 2016-11-30 2017-11-29 항-섬유화 요법을 투여하는 방법

Family Applications After (2)

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KR1020237029765A Ceased KR20230129628A (ko) 2016-11-30 2017-11-29 항-섬유화 요법을 투여하는 방법
KR1020197013644A Ceased KR20190089862A (ko) 2016-11-30 2017-11-29 항-섬유화 요법을 투여하는 방법

Country Status (11)

Country Link
US (3) US11207304B2 (https=)
EP (2) EP3548025A1 (https=)
JP (3) JP2020502054A (https=)
KR (3) KR102575344B1 (https=)
CN (1) CN110087651A (https=)
AU (3) AU2017366881A1 (https=)
CA (2) CA3247781A1 (https=)
IL (3) IL299447A (https=)
MX (3) MX2019006143A (https=)
TW (3) TWI826361B (https=)
WO (1) WO2018102323A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102575344B1 (ko) 2016-11-30 2023-09-06 제넨테크, 인크. 항-섬유화 요법을 투여하는 방법
CN114129517A (zh) * 2020-09-03 2022-03-04 苏州爱科百发生物医药技术有限公司 一种ak3287制剂及其制备方法和应用

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015153683A1 (en) 2014-04-02 2015-10-08 Intermune, Inc. Anti-fibrotic pyridinones

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR092742A1 (es) * 2012-10-02 2015-04-29 Intermune Inc Piridinonas antifibroticas
KR102575344B1 (ko) 2016-11-30 2023-09-06 제넨테크, 인크. 항-섬유화 요법을 투여하는 방법

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015153683A1 (en) 2014-04-02 2015-10-08 Intermune, Inc. Anti-fibrotic pyridinones

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
British Journal of Clinical Pharmacology, 20(6), 621-628, 1989.

Also Published As

Publication number Publication date
TWI826361B (zh) 2023-12-21
EP3548025A1 (en) 2019-10-09
US12310951B2 (en) 2025-05-27
WO2018102323A1 (en) 2018-06-07
JP2023139157A (ja) 2023-10-03
KR20190089862A (ko) 2019-07-31
MX2019006143A (es) 2019-10-17
US20240197693A1 (en) 2024-06-20
JP7495951B2 (ja) 2024-06-05
AU2023263548B2 (en) 2025-10-16
KR20220139450A (ko) 2022-10-14
EP4470624A3 (en) 2025-01-08
MX2020011766A (es) 2020-11-24
TW201825093A (zh) 2018-07-16
TW202539656A (zh) 2025-10-16
EP4470624A2 (en) 2024-12-04
KR20230129628A (ko) 2023-09-08
AU2023263548A1 (en) 2023-11-30
CA3247781A1 (en) 2025-07-09
TWI891129B (zh) 2025-07-21
TW202412795A (zh) 2024-04-01
IL289544A (en) 2022-03-01
US20190321344A1 (en) 2019-10-24
CA3045455A1 (en) 2018-06-07
IL299447A (en) 2023-02-01
CN110087651A (zh) 2019-08-02
IL289544B2 (en) 2023-06-01
MX2023003924A (es) 2023-04-26
AU2025238129A1 (en) 2025-10-23
US11925624B2 (en) 2024-03-12
JP2022058873A (ja) 2022-04-12
AU2017366881A1 (en) 2019-05-30
US11207304B2 (en) 2021-12-28
IL266480A (en) 2019-07-31
US20220184046A1 (en) 2022-06-16
JP2020502054A (ja) 2020-01-23

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