CA3247781A1 - METHODS OF ADMINISTRATING ANTIFIBROTIC THERAPY - Google Patents

METHODS OF ADMINISTRATING ANTIFIBROTIC THERAPY

Info

Publication number
CA3247781A1
CA3247781A1 CA3247781A CA3247781A CA3247781A1 CA 3247781 A1 CA3247781 A1 CA 3247781A1 CA 3247781 A CA3247781 A CA 3247781A CA 3247781 A CA3247781 A CA 3247781A CA 3247781 A1 CA3247781 A1 CA 3247781A1
Authority
CA
Canada
Prior art keywords
compound
subject
therapy
dose
food
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CA3247781A
Other languages
English (en)
French (fr)
Inventor
Lin Pan
Dorothy Sze-Wing Cheung
Jeffrey Mark Harris
Indiana Strombom
Original Assignee
Genentech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Genentech Inc filed Critical Genentech Inc
Publication of CA3247781A1 publication Critical patent/CA3247781A1/en
Pending legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4355Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having oxygen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CA3247781A 2016-11-30 2017-11-29 METHODS OF ADMINISTRATING ANTIFIBROTIC THERAPY Pending CA3247781A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201662428163P 2016-11-30 2016-11-30
US62/428,163 2016-11-30
US201662432425P 2016-12-09 2016-12-09
US62/432,425 2016-12-09
CA3045455A CA3045455A1 (en) 2016-11-30 2017-11-29 Methods of administering anti-fibrotic therapy

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CA3045455A Division CA3045455A1 (en) 2016-11-30 2017-11-29 Methods of administering anti-fibrotic therapy

Publications (1)

Publication Number Publication Date
CA3247781A1 true CA3247781A1 (en) 2025-07-09

Family

ID=60655162

Family Applications (2)

Application Number Title Priority Date Filing Date
CA3247781A Pending CA3247781A1 (en) 2016-11-30 2017-11-29 METHODS OF ADMINISTRATING ANTIFIBROTIC THERAPY
CA3045455A Pending CA3045455A1 (en) 2016-11-30 2017-11-29 Methods of administering anti-fibrotic therapy

Family Applications After (1)

Application Number Title Priority Date Filing Date
CA3045455A Pending CA3045455A1 (en) 2016-11-30 2017-11-29 Methods of administering anti-fibrotic therapy

Country Status (11)

Country Link
US (3) US11207304B2 (https=)
EP (2) EP4470624A3 (https=)
JP (3) JP2020502054A (https=)
KR (3) KR20230129628A (https=)
CN (1) CN110087651A (https=)
AU (3) AU2017366881A1 (https=)
CA (2) CA3247781A1 (https=)
IL (3) IL299447A (https=)
MX (3) MX2019006143A (https=)
TW (3) TW202539656A (https=)
WO (1) WO2018102323A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11207304B2 (en) 2016-11-30 2021-12-28 Genentech, Inc. Methods of administering anti-fibrotic therapy
CN114129517A (zh) * 2020-09-03 2022-03-04 苏州爱科百发生物医药技术有限公司 一种ak3287制剂及其制备方法和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR092742A1 (es) 2012-10-02 2015-04-29 Intermune Inc Piridinonas antifibroticas
MX382781B (es) 2014-04-02 2025-03-13 Intermune Inc Piridinonas anti-fibroticas.
US11207304B2 (en) 2016-11-30 2021-12-28 Genentech, Inc. Methods of administering anti-fibrotic therapy

Also Published As

Publication number Publication date
TW202412795A (zh) 2024-04-01
US11925624B2 (en) 2024-03-12
JP2023139157A (ja) 2023-10-03
IL266480A (en) 2019-07-31
TWI826361B (zh) 2023-12-21
IL289544A (en) 2022-03-01
IL299447A (en) 2023-02-01
CA3045455A1 (en) 2018-06-07
AU2023263548B2 (en) 2025-10-16
KR20190089862A (ko) 2019-07-31
CN110087651A (zh) 2019-08-02
AU2017366881A1 (en) 2019-05-30
AU2025238129A1 (en) 2025-10-23
JP2022058873A (ja) 2022-04-12
JP2020502054A (ja) 2020-01-23
MX2020011766A (es) 2020-11-24
IL289544B2 (en) 2023-06-01
US20240197693A1 (en) 2024-06-20
KR20230129628A (ko) 2023-09-08
KR20220139450A (ko) 2022-10-14
EP4470624A2 (en) 2024-12-04
TW201825093A (zh) 2018-07-16
EP4470624A3 (en) 2025-01-08
US11207304B2 (en) 2021-12-28
TW202539656A (zh) 2025-10-16
JP7495951B2 (ja) 2024-06-05
MX2023003924A (es) 2023-04-26
TWI891129B (zh) 2025-07-21
US12310951B2 (en) 2025-05-27
KR102575344B1 (ko) 2023-09-06
AU2023263548A1 (en) 2023-11-30
US20220184046A1 (en) 2022-06-16
WO2018102323A1 (en) 2018-06-07
US20190321344A1 (en) 2019-10-24
MX2019006143A (es) 2019-10-17
EP3548025A1 (en) 2019-10-09

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US12310951B2 (en) Methods of administering anti-fibrotic therapy
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