KR102051449B1 - 결핵균 유래의 4'-포스포판테테이닐 트랜스퍼레이즈 효소 저해물질 및 이를 유효성분으로 함유하는 결핵의 예방 또는 치료용 약학적 조성물 - Google Patents
결핵균 유래의 4'-포스포판테테이닐 트랜스퍼레이즈 효소 저해물질 및 이를 유효성분으로 함유하는 결핵의 예방 또는 치료용 약학적 조성물 Download PDFInfo
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- KR102051449B1 KR102051449B1 KR1020170014330A KR20170014330A KR102051449B1 KR 102051449 B1 KR102051449 B1 KR 102051449B1 KR 1020170014330 A KR1020170014330 A KR 1020170014330A KR 20170014330 A KR20170014330 A KR 20170014330A KR 102051449 B1 KR102051449 B1 KR 102051449B1
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- KR
- South Korea
- Prior art keywords
- tuberculosis
- pharmaceutical composition
- active ingredient
- compound
- phosphopantetheinyl transferase
- Prior art date
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- A23L33/00—Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
- A23L33/10—Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof using additives
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4196—1,2,4-Triazoles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/428—Thiazoles condensed with carbocyclic rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D263/57—Aryl or substituted aryl radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
- C07D277/66—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2 with aromatic rings or ring systems directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
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- A23V—INDEXING SCHEME RELATING TO FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES AND LACTIC OR PROPIONIC ACID BACTERIA USED IN FOODSTUFFS OR FOOD PREPARATION
- A23V2002/00—Food compositions, function of food ingredients or processes for food or foodstuffs
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23V—INDEXING SCHEME RELATING TO FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES AND LACTIC OR PROPIONIC ACID BACTERIA USED IN FOODSTUFFS OR FOOD PREPARATION
- A23V2200/00—Function of food ingredients
- A23V2200/30—Foods, ingredients or supplements having a functional effect on health
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- Y10S514/924—
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- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
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- Engineering & Computer Science (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR1020170014330A KR102051449B1 (ko) | 2017-02-01 | 2017-02-01 | 결핵균 유래의 4'-포스포판테테이닐 트랜스퍼레이즈 효소 저해물질 및 이를 유효성분으로 함유하는 결핵의 예방 또는 치료용 약학적 조성물 |
| PCT/KR2018/001262 WO2018143638A1 (fr) | 2017-02-01 | 2018-01-30 | Inhibiteur d'enzyme de 4'-phosphopantéthéinyl transférase dérivé de mycobacterium tuberculosis et composition pharmaceutique le contenant en tant que principe actif pour la prévention ou le traitement de la tuberculose |
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| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR1020170014330A KR102051449B1 (ko) | 2017-02-01 | 2017-02-01 | 결핵균 유래의 4'-포스포판테테이닐 트랜스퍼레이즈 효소 저해물질 및 이를 유효성분으로 함유하는 결핵의 예방 또는 치료용 약학적 조성물 |
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| Publication Number | Publication Date |
|---|---|
| KR20180089684A KR20180089684A (ko) | 2018-08-09 |
| KR102051449B1 true KR102051449B1 (ko) | 2019-12-03 |
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| KR1020170014330A KR102051449B1 (ko) | 2017-02-01 | 2017-02-01 | 결핵균 유래의 4'-포스포판테테이닐 트랜스퍼레이즈 효소 저해물질 및 이를 유효성분으로 함유하는 결핵의 예방 또는 치료용 약학적 조성물 |
Country Status (2)
| Country | Link |
|---|---|
| KR (1) | KR102051449B1 (fr) |
| WO (1) | WO2018143638A1 (fr) |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20130041005A1 (en) * | 2011-05-13 | 2013-02-14 | Tragex Pharma | Pharmaceutical compositions comprising neuropilin inhibitors, and their use for the prevention and/or treatment of angiogenic disorders and cancers |
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2017
- 2017-02-01 KR KR1020170014330A patent/KR102051449B1/ko active IP Right Grant
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2018
- 2018-01-30 WO PCT/KR2018/001262 patent/WO2018143638A1/fr active Application Filing
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20130041005A1 (en) * | 2011-05-13 | 2013-02-14 | Tragex Pharma | Pharmaceutical compositions comprising neuropilin inhibitors, and their use for the prevention and/or treatment of angiogenic disorders and cancers |
Non-Patent Citations (4)
| Title |
|---|
| Chemical Abstract Compound, STN express. RN 347332-12-1 (2001.07.22)* |
| Chemical Abstract Compound, STN express. RN 428447-05-6 (2002.06.11)* |
| Chemical Abstract Compound, STN express. RN 639055-48-4 (2004.01.19)* |
| PARK, S. W. 등, Chemistry & Biology, 2015, 22권, 제1호, 페이지 76-86* |
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| Publication number | Publication date |
|---|---|
| KR20180089684A (ko) | 2018-08-09 |
| WO2018143638A1 (fr) | 2018-08-09 |
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