KR101702159B1 - (4―페닐―피페리딘―1―일)―[5―(1h―피라졸―4―일)―티오펜―3―일]―메탄온 화합물 및 그의 용도 - Google Patents

(4―페닐―피페리딘―1―일)―[5―(1h―피라졸―4―일)―티오펜―3―일]―메탄온 화합물 및 그의 용도 Download PDF

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KR101702159B1
KR101702159B1 KR1020127006255A KR20127006255A KR101702159B1 KR 101702159 B1 KR101702159 B1 KR 101702159B1 KR 1020127006255 A KR1020127006255 A KR 1020127006255A KR 20127006255 A KR20127006255 A KR 20127006255A KR 101702159 B1 KR101702159 B1 KR 101702159B1
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스캇 피터 웹스터
조나단 로버트 세클
브라이언 로버트 워커
피터 왈드
토마스 데이빗 팔린
하젤 조안 다이크
트레보얼 로버트 페리얼
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더 유니버시티 오브 에든버러
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KR1020127006255A 2009-09-16 2010-09-14 (4―페닐―피페리딘―1―일)―[5―(1h―피라졸―4―일)―티오펜―3―일]―메탄온 화합물 및 그의 용도 Expired - Fee Related KR101702159B1 (ko)

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US24282509P 2009-09-16 2009-09-16
US61/242,825 2009-09-16
PCT/GB2010/001732 WO2011033255A1 (en) 2009-09-16 2010-09-14 (4-phenyl-piperidin-1-yl)-[5-1h-pyrazol-4yl)-thiophen-3-yl]-methanone compounds and their use

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KR20120093161A KR20120093161A (ko) 2012-08-22
KR101702159B1 true KR101702159B1 (ko) 2017-02-02

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US (1) US8642621B2 (enExample)
EP (1) EP2477983B1 (enExample)
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AU (1) AU2010297068B2 (enExample)
CA (1) CA2772504C (enExample)
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ES (1) ES2540547T3 (enExample)
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GB0724251D0 (en) 2007-12-12 2008-02-06 Univ Edinburgh Therapeutic compounds and their use
GB0804685D0 (en) 2008-03-13 2008-04-16 Univ Edinburgh Therapeutic compounds and their use
US8642621B2 (en) 2009-09-16 2014-02-04 The University Of Edinburgh (4-phenyl-piperidin-1-yl)-[5-(1H-pyrazol-4-yl)-thiophen-3-yl]-methanone compounds and their use
CN102947295B (zh) * 2010-04-29 2016-01-20 爱丁堡大学 作为11β-HSD1抑制剂的3,3-二取代的-(8-氮杂双环[3.2.1]辛烷-8-基)-[5-(1H-吡唑-4基)-噻吩-3-基]-甲酮
US9650337B2 (en) 2013-02-14 2017-05-16 Galderma Research & Development Method of synthesising 4-piperidin-4-yl-benzene-1,3-diol and the salts of same and novel compound tert-butyl 4-(2,4-dihydroxy-phenyl)-4-hydroxy-piperidine-1-carboxylate
EP2968303B1 (en) 2013-03-14 2018-07-04 The Trustees of Columbia University in the City of New York Octahydrocyclopentapyrroles, their preparation and use
WO2014151936A1 (en) 2013-03-14 2014-09-25 The Trustees Of Columbia University In The City Of New York Octahydropyrrolopyrroles, their preparation and use
US10273243B2 (en) 2013-03-14 2019-04-30 The Trustees Of Columbia University In The City Of New York 4-phenylpiperidines, their preparation and use
WO2014151959A1 (en) 2013-03-14 2014-09-25 The Trustees Of Columbia University In The City Of New York N-alkyl-2-phenoxyethanamines, their preparation and use
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