KR101702159B1 - (4―페닐―피페리딘―1―일)―[5―(1h―피라졸―4―일)―티오펜―3―일]―메탄온 화합물 및 그의 용도 - Google Patents

(4―페닐―피페리딘―1―일)―[5―(1h―피라졸―4―일)―티오펜―3―일]―메탄온 화합물 및 그의 용도 Download PDF

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KR101702159B1
KR101702159B1 KR1020127006255A KR20127006255A KR101702159B1 KR 101702159 B1 KR101702159 B1 KR 101702159B1 KR 1020127006255 A KR1020127006255 A KR 1020127006255A KR 20127006255 A KR20127006255 A KR 20127006255A KR 101702159 B1 KR101702159 B1 KR 101702159B1
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스캇 피터 웹스터
조나단 로버트 세클
브라이언 로버트 워커
피터 왈드
토마스 데이빗 팔린
하젤 조안 다이크
트레보얼 로버트 페리얼
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더 유니버시티 오브 에든버러
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KR1020127006255A 2009-09-16 2010-09-14 (4―페닐―피페리딘―1―일)―[5―(1h―피라졸―4―일)―티오펜―3―일]―메탄온 화합물 및 그의 용도 Expired - Fee Related KR101702159B1 (ko)

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Application Number Priority Date Filing Date Title
US24282509P 2009-09-16 2009-09-16
US61/242,825 2009-09-16
PCT/GB2010/001732 WO2011033255A1 (en) 2009-09-16 2010-09-14 (4-phenyl-piperidin-1-yl)-[5-1h-pyrazol-4yl)-thiophen-3-yl]-methanone compounds and their use

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KR20120093161A KR20120093161A (ko) 2012-08-22
KR101702159B1 true KR101702159B1 (ko) 2017-02-02

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US (1) US8642621B2 (enExample)
EP (1) EP2477983B1 (enExample)
JP (1) JP5779181B2 (enExample)
KR (1) KR101702159B1 (enExample)
AU (1) AU2010297068B2 (enExample)
CA (1) CA2772504C (enExample)
DK (1) DK2477983T3 (enExample)
ES (1) ES2540547T3 (enExample)
IL (1) IL218315A (enExample)
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GB0724251D0 (en) 2007-12-12 2008-02-06 Univ Edinburgh Therapeutic compounds and their use
GB0804685D0 (en) 2008-03-13 2008-04-16 Univ Edinburgh Therapeutic compounds and their use
DK2477983T3 (en) 2009-09-16 2015-06-29 Univ Edinburgh (4-phenyl-piperidin-1-yl) - [5-1H-pyrazol-4-yl) -thiophene-3-yl] -METHANONFORBINDELSER AND THEIR USE
BR112012027640B1 (pt) 2010-04-29 2021-08-03 The University Of Edinburgh Composto, composição farmacêutica, e, métodos de preparar uma composição farmacêutica, de inibir a função da 11beta-hidroxiesteroide desidrogenase do tipo 1
CA2900309A1 (fr) * 2013-02-14 2014-08-21 Galderma Research & Development Procede de synthese de 4-piperidin-4-yl-benzene-1,3-diol et de ses sels et nouveau compose 4-(2,4-dihydroxy-phenyl)-4-hydroxy-piperidine-1-carboxylate de tert-butyle
US9944644B2 (en) 2013-03-14 2018-04-17 The Trustees Of Columbia University In The City Of New York Octahydropyrrolopyrroles their preparation and use
US10273243B2 (en) 2013-03-14 2019-04-30 The Trustees Of Columbia University In The City Of New York 4-phenylpiperidines, their preparation and use
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