KR100442718B1 - 1-(4-히드록시페닐)-2-(4-히드록시-4-페닐피페리딘-1-일)-1-프로판올의 메실레이트 염 삼수화물의제조 방법 - Google Patents

1-(4-히드록시페닐)-2-(4-히드록시-4-페닐피페리딘-1-일)-1-프로판올의 메실레이트 염 삼수화물의제조 방법 Download PDF

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KR100442718B1
KR100442718B1 KR10-2001-0023208A KR20010023208A KR100442718B1 KR 100442718 B1 KR100442718 B1 KR 100442718B1 KR 20010023208 A KR20010023208 A KR 20010023208A KR 100442718 B1 KR100442718 B1 KR 100442718B1
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South Korea
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formula
hydroxy
hydroxyphenyl
phenylpiperidin
propanol
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Korean (ko)
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KR20010098960A (ko
Inventor
죠셉 필립 레인빌
테리 진 쥬니어. 시나이
스탠리 왈터 왈린스키
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화이자 프로덕츠 인크.
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
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KR10-2001-0023208A 2000-04-28 2001-04-28 1-(4-히드록시페닐)-2-(4-히드록시-4-페닐피페리딘-1-일)-1-프로판올의 메실레이트 염 삼수화물의제조 방법 Expired - Fee Related KR100442718B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US20067300P 2000-04-28 2000-04-28
US60/200,673 2000-04-28

Publications (2)

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KR20010098960A KR20010098960A (ko) 2001-11-08
KR100442718B1 true KR100442718B1 (ko) 2004-08-02

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US (1) US6645986B2 (enExample)
EP (2) EP1151995B1 (enExample)
JP (2) JP3615496B2 (enExample)
KR (1) KR100442718B1 (enExample)
CN (2) CN1590373A (enExample)
AR (1) AR028376A1 (enExample)
AT (1) ATE277014T1 (enExample)
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Families Citing this family (4)

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Publication number Priority date Publication date Assignee Title
ATE319087T1 (de) * 2000-06-21 2006-03-15 Bioarray Solutions Ltd Multianalytische molekularanalyse durch verwendung anwendungsspezifischer zufallspartikelarrays
US6743921B2 (en) 2002-01-24 2004-06-01 Dsm Catalytica Pharmaceuticals, Inc. Process for the preparation of nonracemic syn-1-(4-hydroxy-phenyl)-2-(4-hydroxy-4-phenyl-piperidin-1-yl)-1-propanol compounds
EP1697543B1 (en) * 2003-11-21 2014-08-20 ANP Technologies, Inc. Asymmetrically branched polymer conjugates and microarray assays
EP1877553B1 (en) 2005-05-02 2011-01-19 ANP Technologies, Inc. Polymer conjugate enhanced bioassays

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6008233A (en) * 1995-08-11 1999-12-28 Pfizer Inc (1S,2S)-1-(4-hydroxyphenyl)-2-(4-hydroxy-4-phenylipiperidin-1-yl)-1-propanolmethanesulfonate trihydrate

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5272160A (en) * 1989-05-17 1993-12-21 Pfizer Inc 2-piperidino-1-alkanol derivatives as antiischemic agents

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6008233A (en) * 1995-08-11 1999-12-28 Pfizer Inc (1S,2S)-1-(4-hydroxyphenyl)-2-(4-hydroxy-4-phenylipiperidin-1-yl)-1-propanolmethanesulfonate trihydrate

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AU781436B2 (en) 2005-05-26
EP1477479A1 (en) 2004-11-17
US20020016465A1 (en) 2002-02-07
JP2001354651A (ja) 2001-12-25
ID30006A (id) 2001-11-01
BR0101630A (pt) 2001-12-04
ATE277014T1 (de) 2004-10-15
HUP0101723A2 (hu) 2002-02-28
TW200505858A (en) 2005-02-16
US6645986B2 (en) 2003-11-11
IN191027B (enExample) 2003-09-13
HU0101723D0 (en) 2001-07-30
YU27701A (sh) 2003-04-30
EP1151995A1 (en) 2001-11-07
AU3889601A (en) 2001-11-01
SI1151995T1 (en) 2004-12-31
HUP0101723A3 (en) 2003-03-28
EP1151995B1 (en) 2004-09-22
DE60105689D1 (de) 2004-10-28
RU2203888C2 (ru) 2003-05-10
ZA200103320B (en) 2002-10-24
CN1590373A (zh) 2005-03-09
ES2227071T3 (es) 2005-04-01
CN1321638A (zh) 2001-11-14
PL347298A1 (en) 2001-11-05
AR028376A1 (es) 2003-05-07
CA2345582C (en) 2006-05-30
JP2004196823A (ja) 2004-07-15
TR200402696T4 (tr) 2004-11-22
CN1210262C (zh) 2005-07-13
DE60105689T2 (de) 2005-11-10
HK1040246B (zh) 2005-10-28
KR20010098960A (ko) 2001-11-08
CA2345582A1 (en) 2001-10-28
HK1040246A1 (en) 2002-05-31
CZ20011471A3 (cs) 2002-02-13
IL142705A0 (en) 2002-03-10
JP3615496B2 (ja) 2005-02-02
PT1151995E (pt) 2004-11-30
DK1151995T3 (da) 2004-12-13

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