JPWO2024043334A5 - - Google Patents
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- Publication number
- JPWO2024043334A5 JPWO2024043334A5 JP2024542889A JP2024542889A JPWO2024043334A5 JP WO2024043334 A5 JPWO2024043334 A5 JP WO2024043334A5 JP 2024542889 A JP2024542889 A JP 2024542889A JP 2024542889 A JP2024542889 A JP 2024542889A JP WO2024043334 A5 JPWO2024043334 A5 JP WO2024043334A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- optionally substituted
- amino
- piperazin
- ethan
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022135257 | 2022-08-26 | ||
| PCT/JP2023/030733 WO2024043334A1 (ja) | 2022-08-26 | 2023-08-25 | 新規なピペラジン誘導体又はその塩及び医薬組成物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPWO2024043334A1 JPWO2024043334A1 (https=) | 2024-02-29 |
| JPWO2024043334A5 true JPWO2024043334A5 (https=) | 2025-05-09 |
Family
ID=90013519
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024542889A Pending JPWO2024043334A1 (https=) | 2022-08-26 | 2023-08-25 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20250326744A1 (https=) |
| EP (1) | EP4578849A4 (https=) |
| JP (1) | JPWO2024043334A1 (https=) |
| CN (1) | CN119816484A (https=) |
| AU (1) | AU2023331216A1 (https=) |
| WO (1) | WO2024043334A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2025178125A1 (ja) * | 2024-02-22 | 2025-08-28 | 富士フイルム株式会社 | 新規なピペラジン誘導体又はその塩 |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH09241241A (ja) * | 1996-03-08 | 1997-09-16 | Roussel Morishita Kk | N−(1−置換−4−ピペリジル)ベンズアミド誘導体 |
| US20050009843A1 (en) * | 2001-04-26 | 2005-01-13 | Kiyoshi Nakayama | Medicine for inhibiting drug elimination pump |
| US6689782B2 (en) * | 2001-07-16 | 2004-02-10 | Essential Therapeutics, Inc. | Fungal efflux pump inhibitors |
| CN1158270C (zh) * | 2001-09-26 | 2004-07-21 | 四川大学 | 具有钙离子拮抗作用的双哌嗪类衍生物 |
| JP2005162726A (ja) * | 2003-01-24 | 2005-06-23 | Tanabe Seiyaku Co Ltd | ピラゾロピリミジン化合物およびその製法 |
| US7851474B2 (en) * | 2005-08-02 | 2010-12-14 | Neurogen Corporation | Dipiperazinyl ketones and related analogues |
| KR20080061613A (ko) * | 2006-12-28 | 2008-07-03 | (주) 비엔씨바이오팜 | 2-(메틸티오)피리미딘 유도체, 그 제조방법 및 이를포함하는 항바이러스용 약학적 조성물 |
| CN101070308B (zh) * | 2007-06-19 | 2011-05-04 | 天津药物研究院 | 异噁唑啉衍生物及其用途 |
| CN101361741B (zh) * | 2008-09-22 | 2011-07-27 | 天津药物研究院 | 异噁唑啉类衍生物抗肿瘤新用途 |
| CN104610160A (zh) * | 2013-11-04 | 2015-05-13 | 南京大学 | 含哌嗪环的5-硝基咪唑类衍生物及其制备与在抗菌药物中的应用 |
| MX2021004191A (es) * | 2018-10-15 | 2021-05-27 | Nurix Therapeutics Inc | Compuestos bifuncionales para degradar la tirosina cinasa de bruton (btk) mediante la trayectoria de ubiquitina proteosoma. |
| WO2021113557A1 (en) * | 2019-12-04 | 2021-06-10 | Nurix Therapeutics, Inc. | Bifunctional compounds for degrading btk via ubiquitin proteosome pathway |
| CN113527227B (zh) * | 2020-04-15 | 2024-06-21 | 四川弘远药业有限公司 | 一种卡利拉嗪的制备方法 |
| WO2022047008A1 (en) * | 2020-08-26 | 2022-03-03 | Tarveda Therapeutics, Inc. | Hsp90-binding conjugates and formulations thereof |
| CN112358466B (zh) * | 2020-10-10 | 2021-10-26 | 广东省微生物研究所(广东省微生物分析检测中心) | 1,2,4-三唑-诺氟沙星杂合体及其制备方法和应用 |
| CN112592339B (zh) * | 2020-12-22 | 2022-06-07 | 广东省微生物研究所(广东省微生物分析检测中心) | 1,3,4-恶二唑-2(3h)-硫酮-诺氟沙星杂合体及其制备方法和应用 |
| WO2023055952A1 (en) * | 2021-09-29 | 2023-04-06 | C4 Therapeutics, Inc. | Neurotrophic tyrosine receptor kinase (ntrk) degrading compounds |
-
2023
- 2023-08-25 EP EP23857442.0A patent/EP4578849A4/en active Pending
- 2023-08-25 CN CN202380062202.6A patent/CN119816484A/zh active Pending
- 2023-08-25 AU AU2023331216A patent/AU2023331216A1/en active Pending
- 2023-08-25 JP JP2024542889A patent/JPWO2024043334A1/ja active Pending
- 2023-08-25 WO PCT/JP2023/030733 patent/WO2024043334A1/ja not_active Ceased
-
2025
- 2025-02-24 US US19/061,542 patent/US20250326744A1/en active Pending
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