JPWO2023207283A5 - - Google Patents

Info

Publication number
JPWO2023207283A5
JPWO2023207283A5 JP2024563976A JP2024563976A JPWO2023207283A5 JP WO2023207283 A5 JPWO2023207283 A5 JP WO2023207283A5 JP 2024563976 A JP2024563976 A JP 2024563976A JP 2024563976 A JP2024563976 A JP 2024563976A JP WO2023207283 A5 JPWO2023207283 A5 JP WO2023207283A5
Authority
JP
Japan
Prior art keywords
group
alkyl
compound
independently selected
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024563976A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025517106A (ja
JP2025517106A5 (https=
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2023/077272 external-priority patent/WO2023207283A1/en
Publication of JP2025517106A publication Critical patent/JP2025517106A/ja
Publication of JPWO2023207283A5 publication Critical patent/JPWO2023207283A5/ja
Publication of JP2025517106A5 publication Critical patent/JP2025517106A5/ja
Pending legal-status Critical Current

Links

JP2024563976A 2022-04-28 2023-02-20 Parp1阻害剤としての化合物 Pending JP2025517106A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CNPCT/CN2022/089986 2022-04-28
CN2022089986 2022-04-28
PCT/CN2023/077272 WO2023207283A1 (en) 2022-04-28 2023-02-20 Compounds as parp1 inhibitiors

Publications (3)

Publication Number Publication Date
JP2025517106A JP2025517106A (ja) 2025-06-03
JPWO2023207283A5 true JPWO2023207283A5 (https=) 2026-02-27
JP2025517106A5 JP2025517106A5 (https=) 2026-02-27

Family

ID=88517229

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024563976A Pending JP2025517106A (ja) 2022-04-28 2023-02-20 Parp1阻害剤としての化合物

Country Status (6)

Country Link
US (1) US20250289814A1 (https=)
EP (1) EP4514795A4 (https=)
JP (1) JP2025517106A (https=)
KR (1) KR20250033148A (https=)
CN (1) CN119487027A (https=)
WO (1) WO2023207283A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2023209820B2 (en) 2022-01-21 2024-10-10 Xinthera, Inc. Parp1 inhibitors and uses thereof
KR20240161147A (ko) 2022-03-14 2024-11-12 슬랩 파마슈티컬스 엘엘씨 다중 사이클릭 화합물
FI4497438T3 (fi) 2022-04-28 2025-10-20 Xinthera Inc Trisyklisiä parp1:n estäjiä ja niiden käyttötapoja
TW202416977A (zh) * 2022-09-30 2024-05-01 大陸商中國醫藥研究開發中心有限公司 含氮雜環類化合物及其醫藥用途
US20250129051A1 (en) * 2023-10-23 2025-04-24 Gilead Sciences, Inc. Parp1 inhibitors and uses thereof

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUP9903758A3 (en) * 1996-05-29 2000-07-28 Warner Lambert Co Benzoxazinone dopamine d4 receptor antagonists and pharmaceutical compositions containing the same
GB0227240D0 (en) * 2002-11-21 2002-12-31 Glaxo Group Ltd Compounds
RU2007101544A (ru) * 2004-06-17 2008-08-10 Уайт (Us) Антагонисты рецепторов высвобождающего гонадотропин гормона
US8404713B2 (en) * 2007-10-26 2013-03-26 Janssen Pharmaceutica Nv Quinolinone derivatives as PARP inhibitors
AR070221A1 (es) * 2008-01-23 2010-03-25 Astrazeneca Ab Derivados de ftalazinona inhibidores de polimerasas, composiciones farmaceuticas que los contienen y usos de los mismos para prevenir y/o tratar tumores cancerigenos,lesiones isquemicas y otras enfermedades asociadas.
WO2010111626A2 (en) * 2009-03-27 2010-09-30 Takeda Pharmaceutical Company Limited Poly (adp-ribose) polymerase (parp) inhibitors
MX2022000711A (es) * 2019-07-19 2022-02-23 Astrazeneca Ab Inhibidores de parp1.
TW202309025A (zh) * 2021-04-19 2023-03-01 美商辛瑟拉股份有限公司 Parp1抑制劑及其用途
WO2022228387A1 (en) * 2021-04-26 2022-11-03 Fochon Biosciences, Ltd. Compounds as parp inhibitors
US20230159525A1 (en) * 2021-10-01 2023-05-25 Xinthera, Inc. Azetidine and pyrrolidine parp1 inhibitors and uses thereof
TW202416977A (zh) * 2022-09-30 2024-05-01 大陸商中國醫藥研究開發中心有限公司 含氮雜環類化合物及其醫藥用途

Similar Documents

Publication Publication Date Title
EP2799437B1 (en) Quinoline and cinnoline derivatives and use thereof
TWI296524B (en) Angiogenesis inhibitors
CN104736155B (zh) 双环化合物作为激酶的抑制剂
JPWO2021013735A5 (https=)
EP2253625A1 (en) Pyridazinones, the preparation and the use thereof
JP2011509301A5 (https=)
EP2990057B1 (en) Pai-1 inhibitor for use in enhancing the antitumor effect of an antitumor agent in a patient
EP3710456B1 (en) Macrocyclic indole derivatives
US10752612B2 (en) PLK4 inhibitors
JP2007508238A5 (https=)
EP4331614A1 (en) Use of medicament in treatment of tumor disease
KR102038401B1 (ko) 키나아제 억제제의 제조 및 응용
JP2011509302A5 (https=)
CN104230952B (zh) 含有嘧啶骨架的化合物及其制备方法和用途
KR20180118745A (ko) 소라페닙 또는 레고라페닙과 트록사시타빈의 포스포라미데이트 전구약물의 병용 요법
US20210395242A1 (en) Heterocyclic compounds as ahr modulators
CN111763215A (zh) 一种具有含氮杂环结构的化合物及其制备方法和用途
CN111217815B (zh) 含有喋啶酮骨架的化合物及其制备方法和应用
JPWO2023207283A5 (https=)
JP2017137323A (ja) 新規抗がん剤
JPH07252147A (ja) クマリン誘導体を含有する薬剤
CN114790207A (zh) 作为pi3k/mtor抑制剂的被取代的吡啶基取代的稠合喹啉化合物
WO2025087460A1 (zh) 一种吡啶并吡唑衍生物药物组合物及其应用
JPWO2020045461A1 (ja) ピラゾロ[3,4−d]ピリミジン化合物を有効成分とする治療剤
CN112442014B (zh) Pdgfr激酶抑制剂及其用途