JPWO2023140329A5 - - Google Patents

Download PDF

Info

Publication number
JPWO2023140329A5
JPWO2023140329A5 JP2023575297A JP2023575297A JPWO2023140329A5 JP WO2023140329 A5 JPWO2023140329 A5 JP WO2023140329A5 JP 2023575297 A JP2023575297 A JP 2023575297A JP 2023575297 A JP2023575297 A JP 2023575297A JP WO2023140329 A5 JPWO2023140329 A5 JP WO2023140329A5
Authority
JP
Japan
Prior art keywords
cancer
active ingredient
pharmaceutical composition
mutant
protein
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2023575297A
Other languages
English (en)
Japanese (ja)
Other versions
JP7540104B2 (ja
JPWO2023140329A1 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/JP2023/001552 external-priority patent/WO2023140329A1/ja
Publication of JPWO2023140329A1 publication Critical patent/JPWO2023140329A1/ja
Publication of JPWO2023140329A5 publication Critical patent/JPWO2023140329A5/ja
Priority to JP2024135111A priority Critical patent/JP2024161461A/ja
Application granted granted Critical
Publication of JP7540104B2 publication Critical patent/JP7540104B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023575297A 2022-01-21 2023-01-19 がんの治療または予防用医薬 Active JP7540104B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024135111A JP2024161461A (ja) 2022-01-21 2024-08-13 がんの治療または予防用医薬

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2022008247 2022-01-21
JP2022008247 2022-01-21
EP22196417.4 2022-09-19
EP22196417 2022-09-19
PCT/JP2023/001552 WO2023140329A1 (ja) 2022-01-21 2023-01-19 がんの治療または予防用医薬

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024135111A Division JP2024161461A (ja) 2022-01-21 2024-08-13 がんの治療または予防用医薬

Publications (3)

Publication Number Publication Date
JPWO2023140329A1 JPWO2023140329A1 (https=) 2023-07-27
JPWO2023140329A5 true JPWO2023140329A5 (https=) 2024-08-06
JP7540104B2 JP7540104B2 (ja) 2024-08-26

Family

ID=87348318

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2023575297A Active JP7540104B2 (ja) 2022-01-21 2023-01-19 がんの治療または予防用医薬
JP2024135111A Pending JP2024161461A (ja) 2022-01-21 2024-08-13 がんの治療または予防用医薬

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024135111A Pending JP2024161461A (ja) 2022-01-21 2024-08-13 がんの治療または予防用医薬

Country Status (8)

Country Link
EP (1) EP4467154A4 (https=)
JP (2) JP7540104B2 (https=)
KR (2) KR20250135911A (https=)
AU (1) AU2023208566A1 (https=)
IL (1) IL313434A (https=)
MX (1) MX2024008358A (https=)
TW (1) TW202339786A (https=)
WO (1) WO2023140329A1 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112022007535A2 (pt) 2019-11-07 2022-07-12 Chugai Pharmaceutical Co Ltd Composto peptídico cíclico tendo ação inibitória de kras
US12312379B2 (en) 2021-05-07 2025-05-27 Chugai Seiyaku Kabushiki Kaisha Methods for producing cyclic compounds comprising N-substituted amino acid residues
JP7823181B2 (ja) 2022-05-06 2026-03-03 中外製薬株式会社 Hrasおよびnrasに対して選択的なkras阻害作用を有する環状化合物
US20250049810A1 (en) 2023-08-07 2025-02-13 Revolution Medicines, Inc. Methods of treating a ras protein-related disease or disorder
AU2024360465A1 (en) 2023-10-12 2026-04-09 Revolution Medicines, Inc. Macrocyclic ras inhibitors
WO2025171296A1 (en) 2024-02-09 2025-08-14 Revolution Medicines, Inc. Ras inhibitors
TW202547461A (zh) 2024-05-17 2025-12-16 美商銳新醫藥公司 Ras抑制劑
WO2025255438A1 (en) 2024-06-07 2025-12-11 Revolution Medicines, Inc. Methods of treating a ras protein-related disease or disorder
WO2025265060A1 (en) 2024-06-21 2025-12-26 Revolution Medicines, Inc. Therapeutic compositions and methods for managing treatment-related effects
WO2026006747A1 (en) 2024-06-28 2026-01-02 Revolution Medicines, Inc. Ras inhibitors
WO2026015801A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2026015790A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2026015796A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2026015825A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Use of ras inhibitor for treating pancreatic cancer
WO2026050446A1 (en) 2024-08-29 2026-03-05 Revolution Medicines, Inc. Ras inhibitors
WO2026072904A2 (en) 2024-09-26 2026-04-02 Revolution Medicines, Inc. Compositions and methods for treating lung cancer

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20230523T1 (hr) 2013-09-06 2023-08-04 Taiho Pharmaceutical Co., Ltd. Antitumorski agens i sredstvo za poboljšavanje antitumorskog efekta
JP7377679B2 (ja) * 2018-11-19 2023-11-10 アムジエン・インコーポレーテツド がん治療のためのkrasg12c阻害剤及び1種以上の薬学的に活性な追加の薬剤を含む併用療法
US20220152026A1 (en) * 2019-02-12 2022-05-19 Novartis Ag Pharmaceutical combination comprising tno155 and a krasg12c inhibitor
BR112021018739A2 (pt) * 2019-03-29 2022-05-03 Dicerna Pharmaceuticals Inc Composições e métodos para o tratamento de doenças ou distúrbios associados a kras
EP4017454A4 (en) 2019-08-19 2023-09-20 Savvybaby Pty Ltd. BABY BOTTLE AND ASSOCIATED VALVE SYSTEM
JP2021063014A (ja) 2019-10-10 2021-04-22 国立大学法人 東京大学 白血病治療薬
BR112022007535A2 (pt) * 2019-11-07 2022-07-12 Chugai Pharmaceutical Co Ltd Composto peptídico cíclico tendo ação inibitória de kras
AR121078A1 (es) 2020-01-22 2022-04-13 Chugai Pharmaceutical Co Ltd Derivados de arilamida con actividad antitumoral

Similar Documents

Publication Publication Date Title
JPWO2023140329A5 (https=)
JP2024526155A5 (https=)
Zhao et al. Combining neratinib with CDK4/6, mTOR, and MEK inhibitors in models of HER2-positive cancer
TW202339786A (zh) 癌症之治療或預防用醫藥
CN108601787B (zh) 用于治疗恶性肿瘤的组合疗法
WO2021243280A2 (en) Methods of treating cancer in patients with an anomalous kras gene or deletions within chromosome 9
JP2018518529A5 (https=)
JP2024526135A (ja) Erk1/2阻害剤とkras g12c阻害剤の併用療法
US12281085B2 (en) Bisfluoroalkyl-1,4-benzodiazepinone compounds and methods of use thereof
JP2024505680A5 (https=)
JP2025024064A (ja) 癌治療
TWI906448B (zh) Kras g12c抑制劑在治療癌症中之用途
JP2021536507A (ja) Her駆動性がんを治療または予防するための化合物、組成物、及び方法
US12233072B2 (en) Compositions comprising bisfluoroalkyl-1,4-benzodiazepinone compounds for treating Adenoid Cystic Carcinoma
BR112020023204A2 (pt) composições que compreendem compostos de bisfluoroalquil-1,4-benzodiazepinona e métodos de uso dos mesmos
Arora et al. Evaluation of NUC-1031: a first-in-class ProTide in biliary tract cancer
TW201618785A (zh) 使用erk抑制劑的治療方法
JP2016106092A (ja) 組合せ
JP2022529824A5 (https=)
SG11202112061RA (en) Bisfluoroalkyl-1,4-benzodiazepin one compounds for treating notch-activated breast cancer
Guan et al. Individualized drug screening based on next generation sequencing and patient derived xenograft model for pancreatic cancer with bone metastasis
JP6148320B2 (ja) 組合せ
KR20210113314A (ko) 골수이형성 증후군을 치료하기 위한 alk5 억제제
JP2024507221A5 (https=)
CN116159062A (zh) 药物组合物及其用途