JPWO2023027198A1 - - Google Patents

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Publication number
JPWO2023027198A1
JPWO2023027198A1 JP2022574839A JP2022574839A JPWO2023027198A1 JP WO2023027198 A1 JPWO2023027198 A1 JP WO2023027198A1 JP 2022574839 A JP2022574839 A JP 2022574839A JP 2022574839 A JP2022574839 A JP 2022574839A JP WO2023027198 A1 JPWO2023027198 A1 JP WO2023027198A1
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022574839A
Other versions
JPWO2023027198A5 (ja
JP7253866B1 (ja
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CN202211151791.9A external-priority patent/CN116514734A/zh
Application filed filed Critical
Publication of JPWO2023027198A1 publication Critical patent/JPWO2023027198A1/ja
Priority to JP2023048827A priority Critical patent/JP7466731B2/ja
Application granted granted Critical
Publication of JP7253866B1 publication Critical patent/JP7253866B1/ja
Publication of JPWO2023027198A5 publication Critical patent/JPWO2023027198A5/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/194—Carboxylic acids, e.g. valproic acid having two or more carboxyl groups, e.g. succinic, maleic or phthalic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Virology (AREA)
  • Biophysics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Biochemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
JP2022574839A 2021-11-24 2022-11-22 トリアジン誘導体を含有する経口投与する製剤 Active JP7253866B1 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023048827A JP7466731B2 (ja) 2021-11-24 2023-03-24 トリアジン誘導体を含有する経口投与する製剤

Applications Claiming Priority (19)

Application Number Priority Date Filing Date Title
JP2021189932 2021-11-24
JP2021189932 2021-11-24
JP2021191635 2021-11-26
JP2021191635 2021-11-26
JP2022006725 2022-01-19
JP2022006725 2022-01-19
JP2022012386 2022-01-28
JP2022012386 2022-01-28
JP2022017132 2022-02-07
JP2022017132 2022-02-07
JP2022027629 2022-02-25
JP2022027629 2022-02-25
JP2022046304 2022-03-23
JP2022046304 2022-03-23
JP2022142767 2022-09-08
JP2022142767 2022-09-08
CN202211151791.9 2022-09-21
CN202211151791.9A CN116514734A (zh) 2021-11-24 2022-09-21 三嗪衍生物的制造方法和含有三嗪衍生物的口服给与的制剂
PCT/JP2022/043092 WO2023027198A1 (ja) 2021-11-24 2022-11-22 トリアジン誘導体を含有する経口投与する製剤

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023048827A Division JP7466731B2 (ja) 2021-11-24 2023-03-24 トリアジン誘導体を含有する経口投与する製剤

Publications (3)

Publication Number Publication Date
JPWO2023027198A1 true JPWO2023027198A1 (ja) 2023-03-02
JP7253866B1 JP7253866B1 (ja) 2023-04-07
JPWO2023027198A5 JPWO2023027198A5 (ja) 2023-08-02

Family

ID=85321709

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022574839A Active JP7253866B1 (ja) 2021-11-24 2022-11-22 トリアジン誘導体を含有する経口投与する製剤
JP2023048827A Active JP7466731B2 (ja) 2021-11-24 2023-03-24 トリアジン誘導体を含有する経口投与する製剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023048827A Active JP7466731B2 (ja) 2021-11-24 2023-03-24 トリアジン誘導体を含有する経口投与する製剤

Country Status (6)

Country Link
US (1) US20240148741A1 (ja)
EP (1) EP4289432A1 (ja)
JP (2) JP7253866B1 (ja)
KR (1) KR20230119022A (ja)
AU (1) AU2022333823A1 (ja)
WO (1) WO2023027198A1 (ja)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI811812B (zh) 2020-10-16 2023-08-11 美商基利科學股份有限公司 磷脂化合物及其用途
EP4122926A4 (en) * 2021-04-14 2023-08-30 Shionogi & Co., Ltd TRIAZINE DERIVATIVE HAVING AN INHIBITOR EFFECT ON THE PROPAGATION OF VIRUSES, AND PHARMACEUTICAL COMPOSITION CONTAINING IT
KR20230119022A (ko) 2021-11-24 2023-08-14 시오노기 앤드 컴파니, 리미티드 트라이아진 유도체를 함유하는 경구 투여하는 제제
TW202339757A (zh) * 2022-01-19 2023-10-16 日商塩野義製藥股份有限公司 新型冠狀病毒感染症治療用醫藥
WO2023193818A1 (zh) * 2022-04-08 2023-10-12 湖北九康通生物医药有限公司 一种多取代三嗪烷类化合物的合成方法
CN116589410B (zh) * 2023-05-29 2024-05-03 济南国鼎医药科技有限公司 一种6-氯-2-甲基-2h-吲唑-5-胺的合成方法
CN116621817B (zh) * 2023-07-20 2023-09-29 爱斯特（成都）生物制药股份有限公司 一种富马酸恩赛特韦的晶型及其制备方法、药物组合物和用途

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2318362A1 (en) * 1998-01-13 1999-07-22 Sharon T. Cload Triazine antiviral compounds
PL2399910T3 (pl) 2009-02-13 2014-09-30 Shionogi & Co Pochodne triazyny jako antagoniści receptora p2x3 i/albo p2x2/3 i kompozycja farmaceutyczna zawierająca je
WO2012009258A2 (en) 2010-07-13 2012-01-19 Edward Roberts Peptidomimetic galanin receptor modulators
KR101867110B1 (ko) 2010-08-10 2018-06-12 시오노기 앤드 컴파니, 리미티드 트라이아진 유도체 및 그것을 함유하는 진통 작용을 갖는 의약 조성물
TW201331188A (zh) 2011-12-15 2013-08-01 Shionogi & Co 經取代之三□衍生物及含有其之醫藥組成物
TWI637949B (zh) 2013-06-14 2018-10-11 塩野義製藥股份有限公司 胺基三衍生物及含有其等之醫藥組合物
WO2019087884A1 (ja) * 2017-10-31 2019-05-09 富士フイルム株式会社 組成物、抗菌組成物、抗ウイルス用組成物、抗ノロウイルス用組成物、スプレー、ワイパー
AU2021253796B2 (en) 2020-04-05 2023-06-01 Pfizer Inc. Compounds and methods for the treatment of COVID-19
US11351149B2 (en) 2020-09-03 2022-06-07 Pfizer Inc. Nitrile-containing antiviral compounds
JPWO2022158528A1 (ja) * 2021-01-20 2022-07-28
EP4313097A1 (en) * 2021-03-29 2024-02-07 Shireen Nature Company for General Trading, Ltd. Willow extract and its use in treating coronavirus infection, inflammation, and associated medical conditions
EP4122926A4 (en) * 2021-04-14 2023-08-30 Shionogi & Co., Ltd TRIAZINE DERIVATIVE HAVING AN INHIBITOR EFFECT ON THE PROPAGATION OF VIRUSES, AND PHARMACEUTICAL COMPOSITION CONTAINING IT
CN113735838B (zh) 2021-09-27 2022-07-08 成都施贝康生物医药科技有限公司 二氢嘧啶类化合物、其制备方法及用途
CN113666914B (zh) 2021-09-27 2022-06-07 成都施贝康生物医药科技有限公司 二氢嘧啶类化合物及其制备方法和用途
CN113801097B (zh) 2021-09-27 2022-11-22 成都施贝康生物医药科技有限公司 二氢嘧啶类化合物、其制备方法及用途
CN113773300B (zh) 2021-09-27 2022-10-11 成都施贝康生物医药科技有限公司 磺酰胺类化合物、其制备方法及用途
CN113620888B (zh) 2021-09-27 2023-06-06 成都施贝康生物医药科技有限公司 二氢嘧啶类化合物及其制备方法和应用
KR20230119022A (ko) 2021-11-24 2023-08-14 시오노기 앤드 컴파니, 리미티드 트라이아진 유도체를 함유하는 경구 투여하는 제제

Also Published As

Publication number Publication date
EP4289432A1 (en) 2023-12-13
KR20230119022A (ko) 2023-08-14
AU2022333823A1 (en) 2024-05-02
JP7253866B1 (ja) 2023-04-07
US20240148741A1 (en) 2024-05-09
JP7466731B2 (ja) 2024-04-12
JP2023078413A (ja) 2023-06-06
WO2023027198A1 (ja) 2023-03-02

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