JPWO2022196797A1 - - Google Patents
Info
- Publication number
- JPWO2022196797A1 JPWO2022196797A1 JP2023507198A JP2023507198A JPWO2022196797A1 JP WO2022196797 A1 JPWO2022196797 A1 JP WO2022196797A1 JP 2023507198 A JP2023507198 A JP 2023507198A JP 2023507198 A JP2023507198 A JP 2023507198A JP WO2022196797 A1 JPWO2022196797 A1 JP WO2022196797A1
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
- C07K1/062—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for alpha- or omega-carboxy functions
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/46—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/68—One oxygen atom attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/96—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/02—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length in solution
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/02—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length in solution
- C07K1/026—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length in solution by fragment condensation in solution
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
- C07K1/063—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for alpha-amino functions
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
- C07K1/064—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for omega-amino or -guanidino functions
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
- C07K5/101—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms, e.g. Val, Ile, Leu
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Analytical Chemistry (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021045625 | 2021-03-19 | ||
| PCT/JP2022/012551 WO2022196797A1 (ja) | 2021-03-19 | 2022-03-18 | アミノ酸又はペプチドの製造方法、保護基形成用試薬、及び、化合物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPWO2022196797A1 true JPWO2022196797A1 (https=) | 2022-09-22 |
| JPWO2022196797A5 JPWO2022196797A5 (https=) | 2024-02-26 |
Family
ID=83320476
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023507198A Pending JPWO2022196797A1 (https=) | 2021-03-19 | 2022-03-18 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20240002432A1 (https=) |
| EP (1) | EP4310094A4 (https=) |
| JP (1) | JPWO2022196797A1 (https=) |
| CN (1) | CN116997559A (https=) |
| TW (1) | TW202302620A (https=) |
| WO (1) | WO2022196797A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2025110921A (ja) * | 2024-01-17 | 2025-07-30 | 富士フイルム株式会社 | ペプチドの製造方法、化合物、及びペプチド合成試薬 |
Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016140232A1 (ja) * | 2015-03-04 | 2016-09-09 | Jitsubo株式会社 | ペプチド合成方法 |
| JP2018508531A (ja) * | 2015-03-06 | 2018-03-29 | ステルス バイオセラピューティックス コープ | 薬学的に適切なペプチドを調製するための方法 |
| WO2019231760A1 (en) * | 2018-05-31 | 2019-12-05 | Gap Peptides Llc | Method for solution-phase peptide synthesis and protecting strategies therefore |
| WO2020175472A1 (ja) * | 2019-02-28 | 2020-09-03 | 富士フイルム株式会社 | ペプチド化合物の製造方法、保護基形成用試薬、及び、縮合多環芳香族炭化水素化合物 |
| WO2020175473A1 (ja) * | 2019-02-28 | 2020-09-03 | 富士フイルム株式会社 | ペプチド化合物の製造方法、保護基形成用試薬、及び、芳香族複素環化合物 |
| WO2020262258A1 (ja) * | 2019-06-28 | 2020-12-30 | 富士フイルム株式会社 | ペプチド化合物の製造方法、保護基形成用試薬、及び、縮合多環芳香族炭化水素化合物 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE136551T1 (de) | 1988-05-10 | 1996-04-15 | Alpha 1 Biomedicals Inc | Festphase-verfahren zur gewinnung von thymosin- alpha-1 |
| JPH04360899A (ja) | 1991-06-04 | 1992-12-14 | Tanabe Seiyaku Co Ltd | 生理活性ペンタペプチドの製造法 |
| AU5059800A (en) * | 1999-04-08 | 2000-11-14 | Deutsches Krebsforschungszentrum Stiftung Des Offentlichen Rechts | Nucleoside derivatives with photo-unstable protective groups |
| JP5609815B2 (ja) * | 2010-08-26 | 2014-10-22 | 信越化学工業株式会社 | ポジ型化学増幅レジスト材料及びパターン形成方法 |
| JP5454458B2 (ja) * | 2010-11-25 | 2014-03-26 | 信越化学工業株式会社 | ポジ型レジスト材料及びパターン形成方法 |
| GB201310921D0 (en) * | 2013-06-19 | 2013-07-31 | Chemical & Biopharmaceutical Lab Of Patras S A | Peptide-resin conjugate and use thereof |
| WO2020189621A1 (ja) * | 2019-03-15 | 2020-09-24 | 日産化学株式会社 | ペプチド化合物の製造方法 |
| JP7301965B2 (ja) | 2019-06-28 | 2023-07-03 | 富士フイルム株式会社 | ペプチド化合物の製造方法、保護基形成用試薬、及び、縮合多環化合物 |
-
2022
- 2022-03-18 WO PCT/JP2022/012551 patent/WO2022196797A1/ja not_active Ceased
- 2022-03-18 JP JP2023507198A patent/JPWO2022196797A1/ja active Pending
- 2022-03-18 CN CN202280022201.4A patent/CN116997559A/zh active Pending
- 2022-03-18 EP EP22771542.2A patent/EP4310094A4/en active Pending
- 2022-03-18 TW TW111110043A patent/TW202302620A/zh unknown
-
2023
- 2023-09-18 US US18/468,937 patent/US20240002432A1/en active Pending
Patent Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016140232A1 (ja) * | 2015-03-04 | 2016-09-09 | Jitsubo株式会社 | ペプチド合成方法 |
| JP2018508531A (ja) * | 2015-03-06 | 2018-03-29 | ステルス バイオセラピューティックス コープ | 薬学的に適切なペプチドを調製するための方法 |
| WO2019231760A1 (en) * | 2018-05-31 | 2019-12-05 | Gap Peptides Llc | Method for solution-phase peptide synthesis and protecting strategies therefore |
| WO2020175472A1 (ja) * | 2019-02-28 | 2020-09-03 | 富士フイルム株式会社 | ペプチド化合物の製造方法、保護基形成用試薬、及び、縮合多環芳香族炭化水素化合物 |
| WO2020175473A1 (ja) * | 2019-02-28 | 2020-09-03 | 富士フイルム株式会社 | ペプチド化合物の製造方法、保護基形成用試薬、及び、芳香族複素環化合物 |
| WO2020262258A1 (ja) * | 2019-06-28 | 2020-12-30 | 富士フイルム株式会社 | ペプチド化合物の製造方法、保護基形成用試薬、及び、縮合多環芳香族炭化水素化合物 |
Non-Patent Citations (1)
| Title |
|---|
| J. ORG. CHEM., vol. 39, no. 23, JPN6026005611, 1974, pages 3441 - 3442, ISSN: 0005796909 * |
Also Published As
| Publication number | Publication date |
|---|---|
| EP4310094A4 (en) | 2024-10-16 |
| CN116997559A (zh) | 2023-11-03 |
| EP4310094A1 (en) | 2024-01-24 |
| US20240002432A1 (en) | 2024-01-04 |
| WO2022196797A1 (ja) | 2022-09-22 |
| TW202302620A (zh) | 2023-01-16 |
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