JPWO2021030379A5 - - Google Patents

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Publication number
JPWO2021030379A5
JPWO2021030379A5 JP2022508918A JP2022508918A JPWO2021030379A5 JP WO2021030379 A5 JPWO2021030379 A5 JP WO2021030379A5 JP 2022508918 A JP2022508918 A JP 2022508918A JP 2022508918 A JP2022508918 A JP 2022508918A JP WO2021030379 A5 JPWO2021030379 A5 JP WO2021030379A5
Authority
JP
Japan
Prior art keywords
carboxamide
isopropylamino
hydroxy
methylbutyl
pyridazine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022508918A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022545364A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/045831 external-priority patent/WO2021030379A1/en
Publication of JP2022545364A publication Critical patent/JP2022545364A/ja
Publication of JPWO2021030379A5 publication Critical patent/JPWO2021030379A5/ja
Pending legal-status Critical Current

Links

JP2022508918A 2019-08-13 2020-08-12 Irak4阻害剤として有用な二環ヘテロアリール化合物 Pending JP2022545364A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962885852P 2019-08-13 2019-08-13
US62/885,852 2019-08-13
PCT/US2020/045831 WO2021030379A1 (en) 2019-08-13 2020-08-12 Bicyclic heteroaryl compounds useful as irak4 inhibitors

Publications (2)

Publication Number Publication Date
JP2022545364A JP2022545364A (ja) 2022-10-27
JPWO2021030379A5 true JPWO2021030379A5 (es) 2023-08-10

Family

ID=72243202

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022508918A Pending JP2022545364A (ja) 2019-08-13 2020-08-12 Irak4阻害剤として有用な二環ヘテロアリール化合物

Country Status (6)

Country Link
US (1) US20220380372A1 (es)
EP (1) EP4013758A1 (es)
JP (1) JP2022545364A (es)
KR (1) KR20220047305A (es)
CN (1) CN114206874A (es)
WO (1) WO2021030379A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CR20210477A (es) 2019-03-19 2022-01-06 Boehringer Ingelheim Animal Health Usa Inc Compuestos de aza-benzotiofeno y aza-benzofurano como antihelmínticos
BR112022024156A2 (pt) 2020-05-29 2023-02-14 Boehringer Ingelheim Animal Health Usa Inc Compostos heterocílicos antelmínticos
CA3236894A1 (en) 2021-11-01 2023-05-04 Boehringer Ingelheim Vetmedica Gmbh Anthelmintic pyrrolopyridazine compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011014817A1 (en) * 2009-07-31 2011-02-03 Biocryst Pharmaceuticals, Inc. Pyrrolo [1, 2-b] pyridazine derivatives as janus kinase inhibitors
EP2686321B1 (en) * 2011-03-17 2016-11-16 Bristol-Myers Squibb Company Pyrrolopyridazine jak3 inhibitors and their use for the treatment of inflammatory and autoimmune diseases
WO2012129258A1 (en) * 2011-03-22 2012-09-27 Merck Sharp & Dohme Corp. Amidopyrazole inhibitors of interleukin receptor-associated kinases
US10155765B2 (en) * 2015-03-12 2018-12-18 Merck Sharp & Dohme Corp. Carboxamide inhibitors of IRAK4 activity

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