JPWO2021014166A5 - - Google Patents
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- Publication number
- JPWO2021014166A5 JPWO2021014166A5 JP2022504089A JP2022504089A JPWO2021014166A5 JP WO2021014166 A5 JPWO2021014166 A5 JP WO2021014166A5 JP 2022504089 A JP2022504089 A JP 2022504089A JP 2022504089 A JP2022504089 A JP 2022504089A JP WO2021014166 A5 JPWO2021014166 A5 JP WO2021014166A5
- Authority
- JP
- Japan
- Prior art keywords
- hydroxy
- compound
- carboxamide
- acetyl
- pyridine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB1910607.9A GB201910607D0 (en) | 2019-07-24 | 2019-07-24 | Compounds |
| GB1910607.9 | 2019-07-24 | ||
| GB2005739.4 | 2020-04-20 | ||
| GBGB2005739.4A GB202005739D0 (en) | 2020-04-20 | 2020-04-20 | Compounds |
| PCT/GB2020/051778 WO2021014166A1 (en) | 2019-07-24 | 2020-07-24 | Pyridine derivatives as tmem16a modulators for use in the treatment of respiratory conditions |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022541311A JP2022541311A (ja) | 2022-09-22 |
| JPWO2021014166A5 true JPWO2021014166A5 (enExample) | 2023-07-25 |
| JP7583022B2 JP7583022B2 (ja) | 2024-11-13 |
Family
ID=71948615
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022504089A Active JP7583022B2 (ja) | 2019-07-24 | 2020-07-24 | 呼吸器症状の治療における使用のためのtmem16aモジュレータとしてのピリジン誘導体 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20220235006A1 (enExample) |
| EP (1) | EP4003516A1 (enExample) |
| JP (1) | JP7583022B2 (enExample) |
| KR (1) | KR20220063162A (enExample) |
| CN (1) | CN114616226B (enExample) |
| AU (1) | AU2020317036A1 (enExample) |
| BR (1) | BR112022001164A2 (enExample) |
| CA (1) | CA3145120A1 (enExample) |
| CL (1) | CL2022000147A1 (enExample) |
| CO (1) | CO2022002022A2 (enExample) |
| CR (1) | CR20220072A (enExample) |
| IL (1) | IL290035A (enExample) |
| MX (1) | MX2022000841A (enExample) |
| PE (1) | PE20221441A1 (enExample) |
| PH (1) | PH12022550181A1 (enExample) |
| WO (1) | WO2021014166A1 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE20221441A1 (es) * | 2019-07-24 | 2022-09-21 | Tmem16A Ltd | Derivados de piridina como moduladores de tmem16a para su uso en el tratamiento de afecciones respiratorias |
| KR20260025059A (ko) * | 2024-08-13 | 2026-02-23 | 전남대학교산학협력단 | 신규한 치환된 피리딘 유도체 화합물, 이의 제조방법, 및 이를 유효성분으로 포함하는 호흡기 질환의 예방 또는 치료용 약학적 조성물 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050176767A1 (en) * | 2003-10-30 | 2005-08-11 | Laval Chan Chun Kong | Pyridine carboxamide and methods for inhibiting HIV integrase |
| EP3612180B1 (en) * | 2017-04-17 | 2023-10-11 | The Regents of the University of California | Substituted 2-acylamino-cycloalkylthiophene-3-carboxylic acid arylamides as inhibitors of calcium-activated chloride channel tmem16a |
| GB201801355D0 (en) * | 2018-01-26 | 2018-03-14 | Enterprise Therapeutics Ltd | Compounds |
| PE20221441A1 (es) * | 2019-07-24 | 2022-09-21 | Tmem16A Ltd | Derivados de piridina como moduladores de tmem16a para su uso en el tratamiento de afecciones respiratorias |
-
2020
- 2020-07-24 PE PE2022000119A patent/PE20221441A1/es unknown
- 2020-07-24 EP EP20751234.4A patent/EP4003516A1/en active Pending
- 2020-07-24 KR KR1020227006371A patent/KR20220063162A/ko not_active Ceased
- 2020-07-24 BR BR112022001164A patent/BR112022001164A2/pt not_active Application Discontinuation
- 2020-07-24 CN CN202080053192.6A patent/CN114616226B/zh active Active
- 2020-07-24 PH PH1/2022/550181A patent/PH12022550181A1/en unknown
- 2020-07-24 CR CR20220072A patent/CR20220072A/es unknown
- 2020-07-24 WO PCT/GB2020/051778 patent/WO2021014166A1/en not_active Ceased
- 2020-07-24 AU AU2020317036A patent/AU2020317036A1/en not_active Abandoned
- 2020-07-24 JP JP2022504089A patent/JP7583022B2/ja active Active
- 2020-07-24 CA CA3145120A patent/CA3145120A1/en active Pending
- 2020-07-24 MX MX2022000841A patent/MX2022000841A/es unknown
-
2022
- 2022-01-21 US US17/581,504 patent/US20220235006A1/en active Pending
- 2022-01-21 CL CL2022000147A patent/CL2022000147A1/es unknown
- 2022-01-23 IL IL290035A patent/IL290035A/en unknown
- 2022-02-24 CO CONC2022/0002022A patent/CO2022002022A2/es unknown
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