JPWO2020246528A1 - - Google Patents
Info
- Publication number
- JPWO2020246528A1 JPWO2020246528A1 JP2021524890A JP2021524890A JPWO2020246528A1 JP WO2020246528 A1 JPWO2020246528 A1 JP WO2020246528A1 JP 2021524890 A JP2021524890 A JP 2021524890A JP 2021524890 A JP2021524890 A JP 2021524890A JP WO2020246528 A1 JPWO2020246528 A1 JP WO2020246528A1
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Physical Education & Sports Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Inorganic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025010012A JP2025061775A (ja) | 2019-06-04 | 2025-01-23 | 痛風又は高尿酸血症の治療薬 |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2019104534 | 2019-06-04 | ||
| PCT/JP2020/022039 WO2020246528A1 (ja) | 2019-06-04 | 2020-06-04 | 痛風又は高尿酸血症の治療薬 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025010012A Division JP2025061775A (ja) | 2019-06-04 | 2025-01-23 | 痛風又は高尿酸血症の治療薬 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPWO2020246528A1 true JPWO2020246528A1 (https=) | 2020-12-10 |
Family
ID=73653292
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021524890A Pending JPWO2020246528A1 (https=) | 2019-06-04 | 2020-06-04 | |
| JP2025010012A Pending JP2025061775A (ja) | 2019-06-04 | 2025-01-23 | 痛風又は高尿酸血症の治療薬 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025010012A Pending JP2025061775A (ja) | 2019-06-04 | 2025-01-23 | 痛風又は高尿酸血症の治療薬 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20220323441A1 (https=) |
| EP (1) | EP3981469B1 (https=) |
| JP (2) | JPWO2020246528A1 (https=) |
| KR (1) | KR20220016861A (https=) |
| CN (1) | CN113924145A (https=) |
| AU (1) | AU2020287549B2 (https=) |
| CA (1) | CA3149714A1 (https=) |
| WO (1) | WO2020246528A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN121648131A (zh) * | 2020-12-08 | 2026-03-13 | 学校法人东日本学园 | 细胞内atp增强剂 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005121153A1 (ja) * | 2004-06-14 | 2005-12-22 | Nippon Chemiphar Co., Ltd. | 縮合ピリミジン誘導体、及びキサンチンオキシダーゼ阻害剤 |
| JP2016520133A (ja) * | 2013-05-31 | 2016-07-11 | タケダ ファーマシューティカルズ ユー.エス.エー. インコーポレイティド | キサンチンオキシダーゼ阻害剤を用いた治療方法及びそれを含む組成物 |
| WO2019107412A1 (ja) * | 2017-11-28 | 2019-06-06 | 静岡県公立大学法人 | 固体分散体 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2019104534A (ja) | 2017-12-13 | 2019-06-27 | 大日本印刷株式会社 | ロール体梱包箱 |
| JP2021127289A (ja) * | 2018-04-27 | 2021-09-02 | 日本ケミファ株式会社 | 縮合ピリミジン誘導体 |
-
2020
- 2020-06-04 WO PCT/JP2020/022039 patent/WO2020246528A1/ja not_active Ceased
- 2020-06-04 EP EP20817851.7A patent/EP3981469B1/en active Active
- 2020-06-04 CN CN202080040395.1A patent/CN113924145A/zh active Pending
- 2020-06-04 KR KR1020217040180A patent/KR20220016861A/ko active Pending
- 2020-06-04 CA CA3149714A patent/CA3149714A1/en active Pending
- 2020-06-04 JP JP2021524890A patent/JPWO2020246528A1/ja active Pending
- 2020-06-04 AU AU2020287549A patent/AU2020287549B2/en active Active
- 2020-06-04 US US17/615,611 patent/US20220323441A1/en active Pending
-
2025
- 2025-01-23 JP JP2025010012A patent/JP2025061775A/ja active Pending
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005121153A1 (ja) * | 2004-06-14 | 2005-12-22 | Nippon Chemiphar Co., Ltd. | 縮合ピリミジン誘導体、及びキサンチンオキシダーゼ阻害剤 |
| JP2016520133A (ja) * | 2013-05-31 | 2016-07-11 | タケダ ファーマシューティカルズ ユー.エス.エー. インコーポレイティド | キサンチンオキシダーゼ阻害剤を用いた治療方法及びそれを含む組成物 |
| WO2019107412A1 (ja) * | 2017-11-28 | 2019-06-06 | 静岡県公立大学法人 | 固体分散体 |
Non-Patent Citations (3)
| Title |
|---|
| 丹野 史枝: "固体分散体キャリヤとしての添加剤HPMCAS(ヒプロメロース酢酸エステルコハク酸エステル)の物性に関する考察", 薬剤学, vol. 73, no. 4, JPN6019003583, 2013, pages 214 - 222, ISSN: 0005601447 * |
| 尾上誠良: "第3章 非晶質固体分散体", 難水溶性薬物の経口製剤化技術最前線(監修 川上亘作), JPN6020028038, 6 July 2016 (2016-07-06), pages 127 - 135, ISSN: 0005601446 * |
| 柏原俊夫ほか: "第4章 経口投与製剤の設計と開発のストラテジー", 経口投与製剤の設計と評価(編集者 橋田充), JPN6020028036, 1995, pages 47 - 67, ISSN: 0005601445 * |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2020246528A1 (ja) | 2020-12-10 |
| AU2020287549B2 (en) | 2026-01-29 |
| CA3149714A1 (en) | 2020-12-10 |
| KR20220016861A (ko) | 2022-02-10 |
| AU2020287549A1 (en) | 2022-01-27 |
| JP2025061775A (ja) | 2025-04-11 |
| EP3981469A1 (en) | 2022-04-13 |
| EP3981469B1 (en) | 2024-11-20 |
| US20220323441A1 (en) | 2022-10-13 |
| EP3981469A4 (en) | 2023-06-21 |
| CN113924145A (zh) | 2022-01-11 |
Similar Documents
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| A621 | Written request for application examination |
Free format text: JAPANESE INTERMEDIATE CODE: A621 Effective date: 20230526 |
|
| A131 | Notification of reasons for refusal |
Free format text: JAPANESE INTERMEDIATE CODE: A131 Effective date: 20240604 |
|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20240724 |
|
| A02 | Decision of refusal |
Free format text: JAPANESE INTERMEDIATE CODE: A02 Effective date: 20241105 |
|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20250123 |
|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A821 Effective date: 20250123 |