JPWO2020111268A5 - - Google Patents
Download PDFInfo
- Publication number
- JPWO2020111268A5 JPWO2020111268A5 JP2020557880A JP2020557880A JPWO2020111268A5 JP WO2020111268 A5 JPWO2020111268 A5 JP WO2020111268A5 JP 2020557880 A JP2020557880 A JP 2020557880A JP 2020557880 A JP2020557880 A JP 2020557880A JP WO2020111268 A5 JPWO2020111268 A5 JP WO2020111268A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutical composition
- compound
- composition according
- edema
- crystalline form
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2018224434 | 2018-11-30 | ||
| JP2018224434 | 2018-11-30 | ||
| PCT/JP2019/046893 WO2020111268A1 (ja) | 2018-11-30 | 2019-11-29 | (3s)-3-[2-(6-アミノ-2-フルオロピリジン-3-イル)-4-フルオロ-1h-イミダゾール-5-イル]-7-[5-クロロ-2-(1h-テトラゾール-1-イル)フェニル]-2,3-ジヒドロインドリジン-5(1h)-オンの新規結晶 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2020111268A1 JPWO2020111268A1 (ja) | 2021-10-14 |
| JPWO2020111268A5 true JPWO2020111268A5 (https=) | 2022-08-12 |
| JP7196931B2 JP7196931B2 (ja) | 2022-12-27 |
Family
ID=70853323
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020557880A Active JP7196931B2 (ja) | 2018-11-30 | 2019-11-29 | (3s)-3-[2-(6-アミノ-2-フルオロピリジン-3-イル)-4-フルオロ-1h-イミダゾール-5-イル]-7-[5-クロロ-2-(1h-テトラゾール-1-イル)フェニル]-2,3-ジヒドロインドリジン-5(1h)-オンの新規結晶 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20210395250A1 (https=) |
| EP (1) | EP3888653A4 (https=) |
| JP (1) | JP7196931B2 (https=) |
| KR (1) | KR20210097119A (https=) |
| CN (1) | CN113226312A (https=) |
| AU (1) | AU2019390094A1 (https=) |
| BR (1) | BR112021010476A2 (https=) |
| CA (1) | CA3121447A1 (https=) |
| IL (1) | IL283481A (https=) |
| MX (1) | MX2021006147A (https=) |
| NZ (1) | NZ776666A (https=) |
| PH (1) | PH12021551219A1 (https=) |
| SG (1) | SG11202105697SA (https=) |
| TW (1) | TWI826599B (https=) |
| WO (1) | WO2020111268A1 (https=) |
| ZA (1) | ZA202103692B (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2022125869A1 (en) * | 2020-12-11 | 2022-06-16 | Board Of Regents, The University Of Texas System | Compositions and methods of making cocrystals using dielectric heating with dispersive and distributive mixing |
| JP2024125436A (ja) * | 2021-07-20 | 2024-09-19 | 小野薬品工業株式会社 | イミダゾール化合物の製造方法 |
| TWI833610B (zh) * | 2022-03-21 | 2024-02-21 | 大陸商上海濟煜醫藥科技有限公司 | 三并環類化合物製備方法及其中間體 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2630677C2 (ru) * | 2011-12-21 | 2017-09-12 | Оно Фармасьютикал Ко., Лтд. | Соединения |
| JP2016093285A (ja) | 2014-11-13 | 2016-05-26 | 株式会社ユニバーサルエンターテインメント | 遊技機 |
| MX385021B (es) * | 2014-12-10 | 2025-03-14 | Ono Pharmaceutical Co | Derivado de dihidroindolizinona. |
| JP6992284B2 (ja) * | 2016-06-06 | 2022-01-13 | 小野薬品工業株式会社 | ジヒドロインドリジノン誘導体を含有する医薬組成物 |
-
2019
- 2019-11-29 NZ NZ776666A patent/NZ776666A/en unknown
- 2019-11-29 TW TW108143720A patent/TWI826599B/zh not_active IP Right Cessation
- 2019-11-29 EP EP19888537.8A patent/EP3888653A4/en not_active Withdrawn
- 2019-11-29 MX MX2021006147A patent/MX2021006147A/es unknown
- 2019-11-29 KR KR1020217016005A patent/KR20210097119A/ko not_active Abandoned
- 2019-11-29 BR BR112021010476-3A patent/BR112021010476A2/pt not_active Application Discontinuation
- 2019-11-29 SG SG11202105697SA patent/SG11202105697SA/en unknown
- 2019-11-29 WO PCT/JP2019/046893 patent/WO2020111268A1/ja not_active Ceased
- 2019-11-29 AU AU2019390094A patent/AU2019390094A1/en not_active Abandoned
- 2019-11-29 US US17/297,649 patent/US20210395250A1/en not_active Abandoned
- 2019-11-29 CA CA3121447A patent/CA3121447A1/en active Pending
- 2019-11-29 CN CN201980079268.XA patent/CN113226312A/zh active Pending
- 2019-11-29 JP JP2020557880A patent/JP7196931B2/ja active Active
-
2021
- 2021-05-26 IL IL283481A patent/IL283481A/en unknown
- 2021-05-27 PH PH12021551219A patent/PH12021551219A1/en unknown
- 2021-05-28 ZA ZA2021/03692A patent/ZA202103692B/en unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JPWO2020111268A5 (https=) | ||
| RU2018139276A (ru) | Полиморфные модификации n-[(3-фтор-4-метоксипиридин-2-ил)метил]-3-(метоксиметил)-1-({ 4-[(2-оксопиридин-1-ил)метил]фенил} метил)пиразол-4-карбоксамида и их соли | |
| RU2020121152A (ru) | Твердые формы ингибитора калликреина плазмы и их соли | |
| JP2015528798A5 (https=) | ||
| RU2020121150A (ru) | Твердые формы ингибитора калликреина плазмы и его солей | |
| AU2018201060B2 (en) | 7,8-dihydoxyflavone and 7,8-substituted flavone derivatives, compositions, and methods related thereto | |
| JP2014502641A5 (https=) | ||
| JP2015524443A5 (https=) | ||
| JP2019059760A5 (https=) | ||
| JP2019518779A5 (https=) | ||
| JP2004534825A5 (https=) | ||
| JP2017526727A5 (https=) | ||
| RU2009107921A (ru) | ТЕРАПЕВТИЧЕСКИЕ СПОСОБЫ ЛЕЧЕНИЯ ВАСКУЛЯРНЫХ ЗАБОЛЕВАНИЙ ГЛАЗ АНТАГОНИСТАМИ Dll4 | |
| JP2012532112A5 (https=) | ||
| JP2011510014A5 (https=) | ||
| JP2016512505A5 (https=) | ||
| JP2012533570A5 (https=) | ||
| JP2015520151A5 (https=) | ||
| JP2014511891A5 (https=) | ||
| JP2016539180A5 (https=) | ||
| JP2014507455A5 (https=) | ||
| JP2015500223A5 (https=) | ||
| JP2016505071A5 (https=) | ||
| JP2010516700A5 (https=) | ||
| EA201100462A1 (ru) | Серосвязанные соединения для лечения офтальмологических заболеваний и расстройств |