JPWO2020111268A5 - - Google Patents

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Publication number
JPWO2020111268A5
JPWO2020111268A5 JP2020557880A JP2020557880A JPWO2020111268A5 JP WO2020111268 A5 JPWO2020111268 A5 JP WO2020111268A5 JP 2020557880 A JP2020557880 A JP 2020557880A JP 2020557880 A JP2020557880 A JP 2020557880A JP WO2020111268 A5 JPWO2020111268 A5 JP WO2020111268A5
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JP
Japan
Prior art keywords
pharmaceutical composition
compound
composition according
edema
crystalline form
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020557880A
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English (en)
Japanese (ja)
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JPWO2020111268A1 (ja
JP7196931B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/JP2019/046893 external-priority patent/WO2020111268A1/ja
Publication of JPWO2020111268A1 publication Critical patent/JPWO2020111268A1/ja
Publication of JPWO2020111268A5 publication Critical patent/JPWO2020111268A5/ja
Application granted granted Critical
Publication of JP7196931B2 publication Critical patent/JP7196931B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2020557880A 2018-11-30 2019-11-29 (3s)-3-[2-(6-アミノ-2-フルオロピリジン-3-イル)-4-フルオロ-1h-イミダゾール-5-イル]-7-[5-クロロ-2-(1h-テトラゾール-1-イル)フェニル]-2,3-ジヒドロインドリジン-5(1h)-オンの新規結晶 Active JP7196931B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2018224434 2018-11-30
JP2018224434 2018-11-30
PCT/JP2019/046893 WO2020111268A1 (ja) 2018-11-30 2019-11-29 (3s)-3-[2-(6-アミノ-2-フルオロピリジン-3-イル)-4-フルオロ-1h-イミダゾール-5-イル]-7-[5-クロロ-2-(1h-テトラゾール-1-イル)フェニル]-2,3-ジヒドロインドリジン-5(1h)-オンの新規結晶

Publications (3)

Publication Number Publication Date
JPWO2020111268A1 JPWO2020111268A1 (ja) 2021-10-14
JPWO2020111268A5 true JPWO2020111268A5 (https=) 2022-08-12
JP7196931B2 JP7196931B2 (ja) 2022-12-27

Family

ID=70853323

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020557880A Active JP7196931B2 (ja) 2018-11-30 2019-11-29 (3s)-3-[2-(6-アミノ-2-フルオロピリジン-3-イル)-4-フルオロ-1h-イミダゾール-5-イル]-7-[5-クロロ-2-(1h-テトラゾール-1-イル)フェニル]-2,3-ジヒドロインドリジン-5(1h)-オンの新規結晶

Country Status (16)

Country Link
US (1) US20210395250A1 (https=)
EP (1) EP3888653A4 (https=)
JP (1) JP7196931B2 (https=)
KR (1) KR20210097119A (https=)
CN (1) CN113226312A (https=)
AU (1) AU2019390094A1 (https=)
BR (1) BR112021010476A2 (https=)
CA (1) CA3121447A1 (https=)
IL (1) IL283481A (https=)
MX (1) MX2021006147A (https=)
NZ (1) NZ776666A (https=)
PH (1) PH12021551219A1 (https=)
SG (1) SG11202105697SA (https=)
TW (1) TWI826599B (https=)
WO (1) WO2020111268A1 (https=)
ZA (1) ZA202103692B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4259143A4 (en) * 2020-12-11 2024-11-13 Board of Regents, The University of Texas System COMPOSITIONS AND METHODS FOR MANUFACTURING COCRYSTALS BY DIELECTRIC HEATING WITH DISPERSIVE AND DISTRIBUTIVE MIXTURE
JP2024125436A (ja) * 2021-07-20 2024-09-19 小野薬品工業株式会社 イミダゾール化合物の製造方法
WO2023179624A1 (zh) * 2022-03-21 2023-09-28 上海济煜医药科技有限公司 三并环类化合物制备方法及其中间体

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9732085B2 (en) 2011-12-21 2017-08-15 Ono Pharmaceutical Co., Ltd. Pyridinone and pyrimidinone derivatives as factor Xia
JP2016093285A (ja) 2014-11-13 2016-05-26 株式会社ユニバーサルエンターテインメント 遊技機
BR112017012146B1 (pt) * 2014-12-10 2023-11-21 Ono Pharmaceutical Co., Ltd Composto derivado de di-hidroindolizinona, seu uso, composição farmacêutica e inibidor de fxia
JP6992284B2 (ja) * 2016-06-06 2022-01-13 小野薬品工業株式会社 ジヒドロインドリジノン誘導体を含有する医薬組成物

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