JPWO2020053811A5 - - Google Patents

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Publication number
JPWO2020053811A5
JPWO2020053811A5 JP2021514019A JP2021514019A JPWO2020053811A5 JP WO2020053811 A5 JPWO2020053811 A5 JP WO2020053811A5 JP 2021514019 A JP2021514019 A JP 2021514019A JP 2021514019 A JP2021514019 A JP 2021514019A JP WO2020053811 A5 JPWO2020053811 A5 JP WO2020053811A5
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JP
Japan
Prior art keywords
compound
alkyl
hydrogen
methyl
pharmaceutical composition
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JP2021514019A
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English (en)
Japanese (ja)
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JP7361766B2 (ja
JP2022500425A (ja
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Priority claimed from PCT/IB2019/057710 external-priority patent/WO2020053811A1/fr
Publication of JP2022500425A publication Critical patent/JP2022500425A/ja
Publication of JPWO2020053811A5 publication Critical patent/JPWO2020053811A5/ja
Application granted granted Critical
Publication of JP7361766B2 publication Critical patent/JP7361766B2/ja
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JP2021514019A 2018-09-14 2019-09-12 ヒト免疫不全ウイルス複製の阻害剤 Active JP7361766B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862731196P 2018-09-14 2018-09-14
US62/731,196 2018-09-14
US201862733259P 2018-09-19 2018-09-19
US62/733,259 2018-09-19
PCT/IB2019/057710 WO2020053811A1 (fr) 2018-09-14 2019-09-12 Inhibiteurs de la réplication du virus de l'immunodéficience humaine

Publications (3)

Publication Number Publication Date
JP2022500425A JP2022500425A (ja) 2022-01-04
JPWO2020053811A5 true JPWO2020053811A5 (fr) 2022-08-09
JP7361766B2 JP7361766B2 (ja) 2023-10-16

Family

ID=68240777

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021514019A Active JP7361766B2 (ja) 2018-09-14 2019-09-12 ヒト免疫不全ウイルス複製の阻害剤

Country Status (4)

Country Link
US (1) US20220089598A1 (fr)
EP (1) EP3849982A1 (fr)
JP (1) JP7361766B2 (fr)
WO (1) WO2020053811A1 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7398448B2 (ja) 2018-10-24 2023-12-14 ヴィーブ ヘルスケア ユーケー(ナンバー5)リミテッド ヒト免疫不全ウイルス複製の阻害剤
UA128041C2 (uk) 2019-01-25 2024-03-20 Браун Юніверсіті Спосіб лікування пов'язаного з віком запалення у пацієнта
JPWO2021107066A1 (fr) 2019-11-28 2021-06-03

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102464654B (zh) 2010-11-12 2016-01-13 上海泓博智源医药技术有限公司 抗病毒化合物
PT2729448E (pt) 2011-07-06 2015-12-02 Gilead Sciences Inc Compostos para o tratamento de vih
CN102863512B (zh) 2011-07-07 2016-04-20 上海泓博智源医药技术有限公司 抗病毒化合物
TW201443037A (zh) 2013-01-09 2014-11-16 Gilead Sciences Inc 治療用化合物
AU2014205317B2 (en) 2013-01-09 2016-11-24 Gilead Sciences, Inc. 5-membered heteroaryls and their use as antiviral agents
ES2642265T3 (es) 2013-01-09 2017-11-16 Gilead Sciences, Inc. Compuestos terapéuticos para el tratamiento de infecciones virales
TWI694071B (zh) 2013-03-01 2020-05-21 美商基利科學股份有限公司 治療反轉錄病毒科(Retroviridae)病毒感染之治療性化合物
WO2015130966A1 (fr) 2014-02-28 2015-09-03 Gilead Sciences, Inc. Agents antiviraux
US10202353B2 (en) 2014-02-28 2019-02-12 Gilead Sciences, Inc. Therapeutic compounds
WO2016033243A1 (fr) 2014-08-29 2016-03-03 Gilead Sciences, Inc. Agents antirétroviraux
CN109890808B (zh) 2016-08-19 2020-08-07 吉利德科学公司 用于预防性或治疗性治疗hiv病毒感染的治疗性化合物
TW201906834A (zh) 2017-05-02 2019-02-16 英商Viiv醫療保健英國(No.5)有限公司 人類免疫不全病毒複製之抑制劑
JP7083398B2 (ja) 2018-02-15 2022-06-10 ギリアード サイエンシーズ, インコーポレイテッド ピリジン誘導体およびhiv感染を処置するためのその使用
CA3175384A1 (fr) 2018-02-16 2019-08-22 Gilead Sciences, Inc. Methodes et intermediaires pour preparer des composes therapeutiques utiles dans le traitement d'une infection virale des retroviridae
ES2962736T3 (es) 2018-04-11 2024-05-24 Viiv Healthcare Uk No 5 Ltd Compuestos de 4-oxo-3,4-dihidroquinazolina como inhibidores de la replicación del virus de la inmunodeficiencia humana
BR112021001617A2 (pt) 2018-08-09 2021-04-27 VIIV Healthcare UK (No.5) Limited inibidores de replicação do vírus da imunodeficiência humana

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