JPWO2014178229A1 - 放射性ガリウム結合部位を有するポリペプチド、及び、その放射性ガリウム錯体 - Google Patents
放射性ガリウム結合部位を有するポリペプチド、及び、その放射性ガリウム錯体 Download PDFInfo
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- JPWO2014178229A1 JPWO2014178229A1 JP2015514773A JP2015514773A JPWO2014178229A1 JP WO2014178229 A1 JPWO2014178229 A1 JP WO2014178229A1 JP 2015514773 A JP2015514773 A JP 2015514773A JP 2015514773 A JP2015514773 A JP 2015514773A JP WO2014178229 A1 JPWO2014178229 A1 JP WO2014178229A1
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- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0474—Organic compounds complexes or complex-forming compounds, i.e. wherein a radioactive metal (e.g. 111In3+) is complexed or chelated by, e.g. a N2S2, N3S, NS3, N4 chelating group
- A61K51/0478—Organic compounds complexes or complex-forming compounds, i.e. wherein a radioactive metal (e.g. 111In3+) is complexed or chelated by, e.g. a N2S2, N3S, NS3, N4 chelating group complexes from non-cyclic ligands, e.g. EDTA, MAG3
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/57563—Vasoactive intestinal peptide [VIP]; Related peptides
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JP2010515732A (ja) * | 2007-01-11 | 2010-05-13 | イミューノメディクス、インコーポレイテッド | タンパク質、ペプチドおよび他の分子の改善されたf−18標識化のための方法および組成物 |
JP2011507863A (ja) * | 2007-12-19 | 2011-03-10 | イミューノメディクス、インコーポレイテッド | タンパク質、ペプチド、および他の分子のf−18標識のための改良された方法および組成物 |
WO2012046845A1 (ja) * | 2010-10-08 | 2012-04-12 | 国立大学法人京都大学 | ペプチド誘導体及びその使用 |
WO2012108476A1 (ja) * | 2011-02-09 | 2012-08-16 | 国立大学法人京都大学 | 放射性標識されたポリペプチドの製造方法 |
-
2013
- 2013-09-26 TW TW102134720A patent/TW201440791A/zh unknown
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2014
- 2014-03-12 WO PCT/JP2014/056553 patent/WO2014178229A1/ja active Application Filing
- 2014-03-12 JP JP2015514773A patent/JPWO2014178229A1/ja active Pending
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JP2010515732A (ja) * | 2007-01-11 | 2010-05-13 | イミューノメディクス、インコーポレイテッド | タンパク質、ペプチドおよび他の分子の改善されたf−18標識化のための方法および組成物 |
JP2011507863A (ja) * | 2007-12-19 | 2011-03-10 | イミューノメディクス、インコーポレイテッド | タンパク質、ペプチド、および他の分子のf−18標識のための改良された方法および組成物 |
WO2012046845A1 (ja) * | 2010-10-08 | 2012-04-12 | 国立大学法人京都大学 | ペプチド誘導体及びその使用 |
WO2012108476A1 (ja) * | 2011-02-09 | 2012-08-16 | 国立大学法人京都大学 | 放射性標識されたポリペプチドの製造方法 |
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