JPS6330312B2 - - Google Patents

Info

Publication number
JPS6330312B2
JPS6330312B2 JP57025821A JP2582182A JPS6330312B2 JP S6330312 B2 JPS6330312 B2 JP S6330312B2 JP 57025821 A JP57025821 A JP 57025821A JP 2582182 A JP2582182 A JP 2582182A JP S6330312 B2 JPS6330312 B2 JP S6330312B2
Authority
JP
Japan
Prior art keywords
alpha
penam
formula
acid
dioxide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP57025821A
Other languages
English (en)
Japanese (ja)
Other versions
JPS57154192A (en
Inventor
Aanesuto Baasu Uein
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Original Assignee
Pfizer Corp Belgium
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium filed Critical Pfizer Corp Belgium
Publication of JPS57154192A publication Critical patent/JPS57154192A/ja
Publication of JPS6330312B2 publication Critical patent/JPS6330312B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP57025821A 1981-02-20 1982-02-19 Bis-esters of alkanediol as antibacterial Granted JPS57154192A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/236,407 US4364957A (en) 1979-09-26 1981-02-20 Bis-esters of alkanediols as antibacterial agents

Publications (2)

Publication Number Publication Date
JPS57154192A JPS57154192A (en) 1982-09-22
JPS6330312B2 true JPS6330312B2 (en, 2012) 1988-06-17

Family

ID=22889370

Family Applications (1)

Application Number Title Priority Date Filing Date
JP57025821A Granted JPS57154192A (en) 1981-02-20 1982-02-19 Bis-esters of alkanediol as antibacterial

Country Status (11)

Country Link
US (1) US4364957A (en, 2012)
EP (1) EP0059046B1 (en, 2012)
JP (1) JPS57154192A (en, 2012)
AT (1) ATE15044T1 (en, 2012)
AU (1) AU527894B2 (en, 2012)
CA (1) CA1176242A (en, 2012)
DE (1) DE3265503D1 (en, 2012)
DK (1) DK72282A (en, 2012)
ES (1) ES8304992A1 (en, 2012)
GR (1) GR75173B (en, 2012)
IE (1) IE52902B1 (en, 2012)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4478748A (en) * 1981-02-20 1984-10-23 Pfizer Inc. Bis-esters of alkanediols
US4530792A (en) * 1982-11-01 1985-07-23 Pfizer Inc. Process and intermediates for preparation of 1,1-dioxopenicillanoyloxymethyl 6-beta-aminopenicillanate
US4462934A (en) 1983-03-31 1984-07-31 Pfizer Inc. Bis-esters of dicarboxylic acids with amoxicillin and certain hydroxymethylpenicillanate 1,1-dioxides
JPS60214792A (ja) * 1984-04-06 1985-10-28 Taiho Yakuhin Kogyo Kk ペナム酸エステル誘導体
CN104650119B (zh) * 2015-02-10 2017-04-05 中国科学院长春应用化学研究所 一种β‑内酰胺化合物的制备方法
IT202000031070A1 (it) 2020-12-16 2022-06-16 Paolo Bonomi Procedimento di sintesi di derivati ammidici dell’acido 8-idrossi penicillanico

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
BE881675A (fr) 1979-02-13 1980-08-12 Leo Pharm Prod Ltd B-lactames derives de l'acide penicillanique leur preparation et leurs utilisations therapeutiques
IL59257A (en) * 1979-02-13 1983-09-30 Rech Applications Therap 6-(n-(cyclic amino-substituted methylene)amino)penicillanates and salts thereof,their production and pharmaceutical compositions containing them
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4256733A (en) * 1979-09-26 1981-03-17 Pfizer Inc. Acetoxymethyl penam compounds as β-lactamase inhibitors

Also Published As

Publication number Publication date
ATE15044T1 (de) 1985-09-15
DE3265503D1 (en) 1985-09-26
JPS57154192A (en) 1982-09-22
EP0059046A1 (en) 1982-09-01
ES509782A0 (es) 1983-03-16
AU527894B2 (en) 1983-03-31
AU8062382A (en) 1982-11-04
DK72282A (da) 1982-08-21
CA1176242A (en) 1984-10-16
US4364957A (en) 1982-12-21
ES8304992A1 (es) 1983-03-16
IE820342L (en) 1982-08-20
IE52902B1 (en) 1988-04-13
EP0059046B1 (en) 1985-08-21
GR75173B (en, 2012) 1984-07-13

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