JPS62103058A - 安息香酸エステル類 - Google Patents

安息香酸エステル類

Info

Publication number
JPS62103058A
JPS62103058A JP61172627A JP17262786A JPS62103058A JP S62103058 A JPS62103058 A JP S62103058A JP 61172627 A JP61172627 A JP 61172627A JP 17262786 A JP17262786 A JP 17262786A JP S62103058 A JPS62103058 A JP S62103058A
Authority
JP
Japan
Prior art keywords
group
acid
formula
compound
kbr
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP61172627A
Other languages
English (en)
Japanese (ja)
Inventor
Setsuo Fujii
藤井　節郎
Eizo Hattori
服部　英三
Mitsuteru Hirata
平田　光輝
Koichiro Watanabe
渡辺　好一郎
Tomio Ota
大田　富夫
Nobuo Yokoo
横尾　信夫
Masahiko Nagakura
永倉　正彦
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kowa Co Ltd
Original Assignee
Kowa Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to US06/886,046 priority Critical patent/US4746737A/en
Priority to AU60328/86A priority patent/AU6032886A/en
Application filed by Kowa Co Ltd filed Critical Kowa Co Ltd
Priority to EP86110154A priority patent/EP0214429A1/en
Publication of JPS62103058A publication Critical patent/JPS62103058A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/18—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
    • C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
    • C07D207/27—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/08—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP61172627A 1985-07-26 1986-07-22 安息香酸エステル類 Pending JPS62103058A (ja)

Priority Applications (3)

Application Number Priority Date Filing Date Title
US06/886,046 US4746737A (en) 1985-07-26 1986-07-16 Phenyl guanidinobenzoate derivatives which have protease inhibitory activity
AU60328/86A AU6032886A (en) 1985-07-26 1986-07-18 Guanidinobenzoyl esters
EP86110154A EP0214429A1 (en) 1985-07-26 1986-07-23 Benzoyl esters

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP60-165236 1985-07-26
JP16523685 1985-07-26

Publications (1)

Publication Number Publication Date
JPS62103058A true JPS62103058A (ja) 1987-05-13

Family

ID=15808446

Family Applications (1)

Application Number Title Priority Date Filing Date
JP61172627A Pending JPS62103058A (ja) 1985-07-26 1986-07-22 安息香酸エステル類

Country Status (6)

Country Link
JP (1) JPS62103058A (da)
KR (1) KR870001154A (da)
CN (1) CN86105509A (da)
DK (1) DK353786A (da)
ES (1) ES2009208A6 (da)
HU (1) HU196590B (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2848561C (en) * 2011-09-15 2019-04-02 Astellas Pharma Inc. Guanidinobenzoic acid compound

Also Published As

Publication number Publication date
HUT41378A (en) 1987-04-28
HU196590B (en) 1988-12-28
DK353786A (da) 1987-01-27
DK353786D0 (da) 1986-07-25
ES2009208A6 (es) 1989-09-16
CN86105509A (zh) 1987-02-11
KR870001154A (ko) 1987-03-11

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