JPS61145160A - 光学活性なプロピオン酸誘導体の製造法 - Google Patents

光学活性なプロピオン酸誘導体の製造法

Info

Publication number
JPS61145160A
JPS61145160A JP59267436A JP26743684A JPS61145160A JP S61145160 A JPS61145160 A JP S61145160A JP 59267436 A JP59267436 A JP 59267436A JP 26743684 A JP26743684 A JP 26743684A JP S61145160 A JPS61145160 A JP S61145160A
Authority
JP
Japan
Prior art keywords
formula
compound
methoxyphenyl
propionic acid
epoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP59267436A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0461867B2 (US07714131-20100511-C00001.png
Inventor
Masatoshi Hayashi
正敏 林
Masao Yamamoto
雅夫 山本
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Nippon Chemiphar Co Ltd
Original Assignee
Nippon Chemiphar Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nippon Chemiphar Co Ltd filed Critical Nippon Chemiphar Co Ltd
Priority to JP59267436A priority Critical patent/JPS61145160A/ja
Publication of JPS61145160A publication Critical patent/JPS61145160A/ja
Publication of JPH0461867B2 publication Critical patent/JPH0461867B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP59267436A 1984-12-20 1984-12-20 光学活性なプロピオン酸誘導体の製造法 Granted JPS61145160A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP59267436A JPS61145160A (ja) 1984-12-20 1984-12-20 光学活性なプロピオン酸誘導体の製造法

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP59267436A JPS61145160A (ja) 1984-12-20 1984-12-20 光学活性なプロピオン酸誘導体の製造法

Publications (2)

Publication Number Publication Date
JPS61145160A true JPS61145160A (ja) 1986-07-02
JPH0461867B2 JPH0461867B2 (US07714131-20100511-C00001.png) 1992-10-02

Family

ID=17444814

Family Applications (1)

Application Number Title Priority Date Filing Date
JP59267436A Granted JPS61145160A (ja) 1984-12-20 1984-12-20 光学活性なプロピオン酸誘導体の製造法

Country Status (1)

Country Link
JP (1) JPS61145160A (US07714131-20100511-C00001.png)

Cited By (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0338893A2 (fr) * 1988-04-19 1989-10-25 Synthelabo Procédé de préparation de (+)-(2S,3S) (Amino-2 phényl) thio-3 hydroxy-2 (methoxy-4 phényl)-3 propionates de méthyle
EP0342904A2 (en) * 1988-05-18 1989-11-23 MARION LABORATORIES, INC. (a Delaware corporation) 2-Hydroxy-3-(4-methoxyphenyl)-3-(2-aminophenylthio)propionic acid, 8'-phenylmenthyl ester, especially for diltiazem
EP0342902A2 (en) * 1988-05-18 1989-11-23 MARION LABORATORIES, INC. (a Delaware corporation) 2-Hydroxy-propanoic acid acyclic alkyl esters for benzothiazepines
EP0343474A2 (en) * 1988-05-24 1989-11-29 F. Hoffmann-La Roche Ag Process for the preparation of optically pure aminophenylthio- and aminoaphthalenylthio-propanoic acids
US5008411A (en) * 1988-05-24 1991-04-16 Hoffmann-La Roche Inc. Glycidic acid ester and process of preparation
US5013835A (en) * 1989-01-11 1991-05-07 Synthelabo Method of preparing (+)-(2S,3S)-3-hydroxy-2-(4-methoxyphenyl)2,3-dihydro-5H-1,5-benzothiazepine-4-one
AU616517B2 (en) * 1988-05-18 1991-10-31 Aventis Pharmaceuticals Inc. Improved resolution of 3-(4-methoxyphenyl)glycidic acid with in situ conversion to alkyl esters
US5081277A (en) * 1988-10-03 1992-01-14 Synthelabo Process for the preparation of propionic acid derivatives
US5296618A (en) * 1992-05-14 1994-03-22 Orion-Yhtyma Oy Fermion Method for the manufacture of the derivatives of propionic acid
USRE34935E (en) * 1989-01-11 1995-05-09 Synthelabo Method for preparing (+)-(2S,3S)-3-hydroxy-2-(4-methoxyphenyl)-2,3-dihydro-5H-1,5-benzothiazepine-4-one and chlorinated derivatives thereof

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57136581A (en) * 1981-02-18 1982-08-23 Nippon Kayaku Co Ltd Preparation of 1,5-benzothiazepin derivative

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57136581A (en) * 1981-02-18 1982-08-23 Nippon Kayaku Co Ltd Preparation of 1,5-benzothiazepin derivative

Cited By (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5008434A (en) * 1988-04-19 1991-04-16 Synthelabo Process for the preparation of methyl (+)-(2S,3S)-3-[(2-aminophenyl)thio]-2-hydroxy-3-(4-methoxyphenyl)-propionates
EP0338893A2 (fr) * 1988-04-19 1989-10-25 Synthelabo Procédé de préparation de (+)-(2S,3S) (Amino-2 phényl) thio-3 hydroxy-2 (methoxy-4 phényl)-3 propionates de méthyle
AU616517B2 (en) * 1988-05-18 1991-10-31 Aventis Pharmaceuticals Inc. Improved resolution of 3-(4-methoxyphenyl)glycidic acid with in situ conversion to alkyl esters
EP0342902A3 (en) * 1988-05-18 1991-01-30 MARION LABORATORIES, INC. (a Delaware corporation) 2-hydroxy-propanoic acid acyclic alkyl esters for benzothiazepines
EP0342902A2 (en) * 1988-05-18 1989-11-23 MARION LABORATORIES, INC. (a Delaware corporation) 2-Hydroxy-propanoic acid acyclic alkyl esters for benzothiazepines
EP0342904A2 (en) * 1988-05-18 1989-11-23 MARION LABORATORIES, INC. (a Delaware corporation) 2-Hydroxy-3-(4-methoxyphenyl)-3-(2-aminophenylthio)propionic acid, 8'-phenylmenthyl ester, especially for diltiazem
EP0343474A2 (en) * 1988-05-24 1989-11-29 F. Hoffmann-La Roche Ag Process for the preparation of optically pure aminophenylthio- and aminoaphthalenylthio-propanoic acids
EP0343474A3 (en) * 1988-05-24 1991-01-23 F. Hoffmann-La Roche Ag Process for the preparation of optically pure aminophenylthio- and aminoaphthalenylthio-propanoic acids
US5008411A (en) * 1988-05-24 1991-04-16 Hoffmann-La Roche Inc. Glycidic acid ester and process of preparation
US5081277A (en) * 1988-10-03 1992-01-14 Synthelabo Process for the preparation of propionic acid derivatives
US5013835A (en) * 1989-01-11 1991-05-07 Synthelabo Method of preparing (+)-(2S,3S)-3-hydroxy-2-(4-methoxyphenyl)2,3-dihydro-5H-1,5-benzothiazepine-4-one
US5102998A (en) * 1989-01-11 1992-04-07 Synthelabo Method for preparing (+)-(2s,3s)-3-hydroxy-2-(4-methoxyphenyl)-2,3-dihydro-5h-1,5-benzothiazepine-4-one and chlorinated derivatives thereof
USRE34935E (en) * 1989-01-11 1995-05-09 Synthelabo Method for preparing (+)-(2S,3S)-3-hydroxy-2-(4-methoxyphenyl)-2,3-dihydro-5H-1,5-benzothiazepine-4-one and chlorinated derivatives thereof
US5296618A (en) * 1992-05-14 1994-03-22 Orion-Yhtyma Oy Fermion Method for the manufacture of the derivatives of propionic acid

Also Published As

Publication number Publication date
JPH0461867B2 (US07714131-20100511-C00001.png) 1992-10-02

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