JPS6027676B2 - ピリミジノアミノメチルエルゴリン誘導体の製法 - Google Patents

ピリミジノアミノメチルエルゴリン誘導体の製法

Info

Publication number
JPS6027676B2
JPS6027676B2 JP49144603A JP14460374A JPS6027676B2 JP S6027676 B2 JPS6027676 B2 JP S6027676B2 JP 49144603 A JP49144603 A JP 49144603A JP 14460374 A JP14460374 A JP 14460374A JP S6027676 B2 JPS6027676 B2 JP S6027676B2
Authority
JP
Japan
Prior art keywords
dimethyl
formula
carbon atoms
group
pyrimidinoaminomethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP49144603A
Other languages
English (en)
Japanese (ja)
Other versions
JPS5095299A (US08066781-20111129-C00013.png
Inventor
アルカリ ジユリアナ
ベルナルデイ ルイジ
ボシシオ ジエルマノ
グレ−セル アルフレド
テムペリリ アルデミオ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Publication of JPS5095299A publication Critical patent/JPS5095299A/ja
Publication of JPS6027676B2 publication Critical patent/JPS6027676B2/ja
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/02Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hydrocarbon or substituted hydrocarbon radicals, attached in position 8
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Coloring (AREA)
JP49144603A 1973-12-21 1974-12-18 ピリミジノアミノメチルエルゴリン誘導体の製法 Expired JPS6027676B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT5453373 1973-12-21
IT54533/73 1973-12-21

Publications (2)

Publication Number Publication Date
JPS5095299A JPS5095299A (US08066781-20111129-C00013.png) 1975-07-29
JPS6027676B2 true JPS6027676B2 (ja) 1985-06-29

Family

ID=11287369

Family Applications (1)

Application Number Title Priority Date Filing Date
JP49144603A Expired JPS6027676B2 (ja) 1973-12-21 1974-12-18 ピリミジノアミノメチルエルゴリン誘導体の製法

Country Status (15)

Country Link
JP (1) JPS6027676B2 (US08066781-20111129-C00013.png)
AT (1) AT345997B (US08066781-20111129-C00013.png)
BE (1) BE823715A (US08066781-20111129-C00013.png)
CA (1) CA1033725A (US08066781-20111129-C00013.png)
CH (1) CH609345A5 (US08066781-20111129-C00013.png)
DE (1) DE2459630C3 (US08066781-20111129-C00013.png)
DK (1) DK138895B (US08066781-20111129-C00013.png)
FR (1) FR2255072B1 (US08066781-20111129-C00013.png)
GB (1) GB1436820A (US08066781-20111129-C00013.png)
HU (1) HU168767B (US08066781-20111129-C00013.png)
NL (1) NL7416120A (US08066781-20111129-C00013.png)
SE (1) SE417966B (US08066781-20111129-C00013.png)
SU (1) SU604492A3 (US08066781-20111129-C00013.png)
YU (1) YU335774A (US08066781-20111129-C00013.png)
ZA (1) ZA748053B (US08066781-20111129-C00013.png)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1192260B (it) * 1977-07-05 1988-03-31 Simes Derivati di ergoline-2-tioeteri e loro solfossidi
GB2112382B (en) * 1981-11-06 1985-03-06 Erba Farmitalia Ergoline derivatives
GB2120242A (en) * 1982-04-30 1983-11-30 Erba Farmitalia Ergoline derivatives
PH21123A (en) * 1983-04-28 1987-07-27 Erba Farmitalia Ergoline derivatives

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4862800U (US08066781-20111129-C00013.png) * 1971-11-18 1973-08-09

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE792188A (fr) * 1971-12-02 1973-06-01 Farmaceutici Italia Derives de l'ergoline

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4862800U (US08066781-20111129-C00013.png) * 1971-11-18 1973-08-09

Also Published As

Publication number Publication date
CA1033725A (en) 1978-06-27
JPS5095299A (US08066781-20111129-C00013.png) 1975-07-29
AU7659174A (en) 1976-06-24
GB1436820A (en) 1976-05-26
DK138895B (da) 1978-11-13
SE417966B (sv) 1981-04-27
FR2255072A1 (US08066781-20111129-C00013.png) 1975-07-18
ATA1010974A (de) 1978-02-15
CH609345A5 (en) 1979-02-28
FR2255072B1 (US08066781-20111129-C00013.png) 1978-07-28
AT345997B (de) 1978-10-10
BE823715A (fr) 1975-06-20
ZA748053B (en) 1976-01-28
DK664474A (US08066781-20111129-C00013.png) 1975-09-08
DE2459630A1 (de) 1975-07-03
DK138895C (US08066781-20111129-C00013.png) 1979-04-30
SE7416084L (US08066781-20111129-C00013.png) 1975-06-23
YU335774A (en) 1982-05-31
DE2459630C3 (de) 1981-05-07
NL7416120A (nl) 1975-06-24
HU168767B (US08066781-20111129-C00013.png) 1976-07-28
DE2459630B2 (de) 1980-07-10
SU604492A3 (ru) 1978-04-25

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