JPS55100377A - Intermediate for prostaglandim analog and its preparation - Google Patents
Intermediate for prostaglandim analog and its preparationInfo
- Publication number
- JPS55100377A JPS55100377A JP655579A JP655579A JPS55100377A JP S55100377 A JPS55100377 A JP S55100377A JP 655579 A JP655579 A JP 655579A JP 655579 A JP655579 A JP 655579A JP S55100377 A JPS55100377 A JP S55100377A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- tetrahydropyran
- analog
- compound
- prostaglandim
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Pyrane Compounds (AREA)
Abstract
NEW MATERIAL:A prostaglandin analog of formula I (R1 is H, tetrahydropyran- 2-yl, etc.; R2 is H, trityl, etc.; R3 is formyl, etc.; R4 is benzyl, etc.; THP is tetrahydropyran-2-yl, etc.; X is ethylene, etc.; n is 0 or an integer 1W5; R1 and R2 are not H when R3 is formyl).
EXAMPLE: (EZ)-2α-(5-Hydroxy-2-pentenyl)-3β-(1-methoxy-1-methyl)-ethoxymethyl-4α-(tetrahydropyran-2-yloxy)cyclopentan-1-α-ol.
USE: An intermediate for prostaglandin useful as medicines or drugs for animals, or preparing analogs thereof.
PROCESS: A compound of formula I is subjected to the witting reaction with a ylide of a phosphonium compound of formula III (X is halogen; R5 is H, etc.) in a solvent, e.g. THF, to give the objective compound of formula IV.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (10)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP655579A JPS55100377A (en) | 1979-01-25 | 1979-01-25 | Intermediate for prostaglandim analog and its preparation |
HU80142A HU183068B (en) | 1979-01-25 | 1980-01-23 | Process for preparing prostaglandin e down 1 analogues |
GB8002207A GB2045745B (en) | 1979-01-25 | 1980-01-23 | Intermediates for prostaglandin analogues |
SE8000545A SE452157B (en) | 1979-01-25 | 1980-01-23 | INTERMEDIATES FOR THE MANUFACTURING OF TRANS- DELTA? 722-PROSTAGLANDIN-E? 711-ANALOGS AND PROCEDURES FOR PRODUCING THESE |
IT19399/80A IT1149877B (en) | 1979-01-25 | 1980-01-23 | INTERMEDIATE PRODUCTS FOR ANALOGS OF PROSTAGLANDINA |
CA000344233A CA1154441A (en) | 1979-01-25 | 1980-01-23 | Intermediates for prostaglandin analogues |
NL8000428A NL8000428A (en) | 1979-01-25 | 1980-01-23 | INTERMEDIATES FOR THE PREPARATION OF PROSTAGLANDINE ANALOGS, METHODS FOR PREPARING THEM AND THEIR USE IN THE PREPARATION OF PROSTAGLANDINE ANALOGS. |
DK027780A DK165111C (en) | 1979-01-25 | 1980-01-23 | CYCLOPENTAND DERIVATIVES AND PROCEDURES FOR PREPARING THEREOF |
FR8001501A FR2447374A1 (en) | 1979-01-25 | 1980-01-24 | INTERMEDIATES FOR THE PREPARATION OF 2TRANS-PROSTAGLANDIN E1 ANALOGS |
CH57680A CH644360A5 (en) | 1979-01-25 | 1980-01-24 | INTERMEDIATES FOR THE PREPARATION OF TRANS-PROSTAGLANDIN ANALOGS HAVING A DOUBLE LINK BETWEEN CARBON ATOMS 13 AND 14 AND 2 AND 3. |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP655579A JPS55100377A (en) | 1979-01-25 | 1979-01-25 | Intermediate for prostaglandim analog and its preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS55100377A true JPS55100377A (en) | 1980-07-31 |
Family
ID=11641571
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP655579A Pending JPS55100377A (en) | 1979-01-25 | 1979-01-25 | Intermediate for prostaglandim analog and its preparation |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS55100377A (en) |
-
1979
- 1979-01-25 JP JP655579A patent/JPS55100377A/en active Pending
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ES8302616A1 (en) | Process for the preparation of ethylene glycol. | |
JPS55100377A (en) | Intermediate for prostaglandim analog and its preparation | |
JPS572242A (en) | Preparation of 2-bromo-2-nitro-1,3-propanediol | |
JPS5559121A (en) | 1-halo-3-decyne compound | |
FR2295045A1 (en) | PROCESS FOR THE PREPARATION OF VINYL HALOGENIDES WITH LOW VINYL HALOGENIDE WHICH HAVE NOT REACTED | |
JPS57131780A (en) | Novel 6-oxabicyclo(3.2.1)octan-7-one derivative | |
JPS5430144A (en) | Preparation of isocamphane | |
JPS57131792A (en) | Novel 2-oxabicyclo(2.2.2)octan-3-one derivative | |
JPS5281396A (en) | Preparation of curable resins | |
JPS5236649A (en) | Process for preparation of prostaglandin analogs and pharmceutical com position containing the compounds as effetual components | |
JPS51138650A (en) | Process for preparing optically active trans-cyclopentene-3,5,-diolmon oester | |
JPS57183728A (en) | Preparation of methyl-norbornene derivative | |
JPS5772997A (en) | Novel oligomannoside and its preparation | |
JPS52111509A (en) | Preparation of unsaturated compounds | |
JPS5225724A (en) | Process for preparation of pure m-alkyltoluene | |
JPS53111002A (en) | Preparation of squalane | |
JPS5424883A (en) | Prostaglandin analogues and their preparation | |
JPS5536443A (en) | Phenoxybutyramide derivative | |
JPS5625175A (en) | Preparation of antispasmolytic agent | |
JPS5673033A (en) | 1-halo-4-decyne compound | |
JPS51125046A (en) | Process for preparing prostaglandin analogues | |
JPS5239665A (en) | Process for preparing perfluorolactones | |
JPS55124778A (en) | 6-(2,2-ethylenedioxyethyl)fulvene derivative | |
JPS5536444A (en) | Thiocarbostyril derivative | |
JPS5257132A (en) | Process for preparation of thioanisole |