JPS5536444A - Thiocarbostyril derivative - Google Patents
Thiocarbostyril derivativeInfo
- Publication number
- JPS5536444A JPS5536444A JP11044378A JP11044378A JPS5536444A JP S5536444 A JPS5536444 A JP S5536444A JP 11044378 A JP11044378 A JP 11044378A JP 11044378 A JP11044378 A JP 11044378A JP S5536444 A JPS5536444 A JP S5536444A
- Authority
- JP
- Japan
- Prior art keywords
- thiocarbostyril
- derivative
- formula
- hydroxythiocarbostyril
- dihydrothiocarbostyril
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Abstract
NEW MATERIAL:Thiocarbostyril derivative of formula 1 (R1 is lower alkyl; R2 is cycloalkyl; the bond between the 3 and 4 positions in thiocarbostyril is double or single).
EXAMPLE: 6-[ 3-( N-Methyl-N-cyclohexylaminocarbonyl )propoxy ]-3, 4-dihydrothiocarbostyril.
USE: Antithrombosis, anti-inflammatory, antiulcerative, and antiasthmatic.
PREPARATION: A hydroxythiocarbostyril derivative of formula 2 and a haloamide of formula 3 (X is Cl, Br, I) are subjected to dehydrohalogenation reaction to give the compound of formula 1.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP11044378A JPS5536444A (en) | 1978-09-07 | 1978-09-07 | Thiocarbostyril derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP11044378A JPS5536444A (en) | 1978-09-07 | 1978-09-07 | Thiocarbostyril derivative |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5536444A true JPS5536444A (en) | 1980-03-14 |
JPS6148503B2 JPS6148503B2 (en) | 1986-10-24 |
Family
ID=14535842
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP11044378A Granted JPS5536444A (en) | 1978-09-07 | 1978-09-07 | Thiocarbostyril derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5536444A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1989010919A1 (en) | 1988-05-02 | 1989-11-16 | Otsuka Pharmaceutical Co., Ltd. | Carbostyril derivatives |
Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS51133277A (en) * | 1975-05-15 | 1976-11-18 | Otsuka Pharmaceut Co Ltd | A process for preparing novel carbostyril derivatives |
JPS51136676A (en) * | 1975-05-16 | 1976-11-26 | Otsuka Pharmaceut Co Ltd | Process for preparation of carbostyril derivatives |
JPS52125163A (en) * | 1976-04-14 | 1977-10-20 | Otsuka Pharmaceut Co Ltd | Novel benzcyclamide derivatives |
JPS5321177A (en) * | 1976-08-09 | 1978-02-27 | Otsuka Pharmaceut Co Ltd | Thiocarbostyryl derivatives |
-
1978
- 1978-09-07 JP JP11044378A patent/JPS5536444A/en active Granted
Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS51133277A (en) * | 1975-05-15 | 1976-11-18 | Otsuka Pharmaceut Co Ltd | A process for preparing novel carbostyril derivatives |
JPS51136676A (en) * | 1975-05-16 | 1976-11-26 | Otsuka Pharmaceut Co Ltd | Process for preparation of carbostyril derivatives |
JPS52125163A (en) * | 1976-04-14 | 1977-10-20 | Otsuka Pharmaceut Co Ltd | Novel benzcyclamide derivatives |
JPS5321177A (en) * | 1976-08-09 | 1978-02-27 | Otsuka Pharmaceut Co Ltd | Thiocarbostyryl derivatives |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1989010919A1 (en) | 1988-05-02 | 1989-11-16 | Otsuka Pharmaceutical Co., Ltd. | Carbostyril derivatives |
JPH0249768A (en) * | 1988-05-02 | 1990-02-20 | Otsuka Pharmaceut Co Ltd | Carbostyril derivative |
Also Published As
Publication number | Publication date |
---|---|
JPS6148503B2 (en) | 1986-10-24 |
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