JPH0132225B2 - - Google Patents
Info
- Publication number
- JPH0132225B2 JPH0132225B2 JP51077992A JP7799276A JPH0132225B2 JP H0132225 B2 JPH0132225 B2 JP H0132225B2 JP 51077992 A JP51077992 A JP 51077992A JP 7799276 A JP7799276 A JP 7799276A JP H0132225 B2 JPH0132225 B2 JP H0132225B2
- Authority
- JP
- Japan
- Prior art keywords
- benzazepine
- pyrrolo
- dihydro
- cyano
- dimethylaminopropylidene
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/325—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
- C07D207/327—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/38—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to acyclic carbon atoms and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/24—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Anesthesiology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US59243675A | 1975-07-02 | 1975-07-02 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS527996A JPS527996A (en) | 1977-01-21 |
| JPH0132225B2 true JPH0132225B2 (cs) | 1989-06-29 |
Family
ID=24370639
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP51077992A Granted JPS527996A (en) | 1975-07-02 | 1976-07-02 | Pyroro *2*11b* *3** benzazepine |
Country Status (18)
| Country | Link |
|---|---|
| JP (1) | JPS527996A (cs) |
| AU (1) | AU499122B2 (cs) |
| BE (1) | BE843678A (cs) |
| CA (1) | CA1092105A (cs) |
| CH (5) | CH626366A5 (cs) |
| CY (1) | CY1091A (cs) |
| DE (2) | DE2629877A1 (cs) |
| ES (1) | ES449432A1 (cs) |
| FR (1) | FR2315935A1 (cs) |
| GB (1) | GB1499047A (cs) |
| GR (1) | GR60851B (cs) |
| HK (1) | HK60580A (cs) |
| HU (1) | HU177866B (cs) |
| MY (1) | MY8100227A (cs) |
| NL (1) | NL188287C (cs) |
| PT (1) | PT65295B (cs) |
| SE (1) | SE424076B (cs) |
| ZA (1) | ZA763990B (cs) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4148903A (en) * | 1977-07-28 | 1979-04-10 | Merck & Co., Inc. | Antipsychotic, antiserotonin and antihistaminic pyrrolo[2,1-b][3]benzazepines |
| JPH0487401U (cs) * | 1990-12-06 | 1992-07-29 | ||
| US6271392B1 (en) | 1994-10-07 | 2001-08-07 | Rhone-Poulenc Inc. | Intermediates useful for the synthesis of 1-arylpyrrole pesticides |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3428677A (en) * | 1962-09-24 | 1969-02-18 | Merck & Co Inc | Chemical compounds and methods of preparing same |
| US3499037A (en) * | 1966-05-31 | 1970-03-03 | Merck & Co Inc | Preparation of trifluoromethyl substituted dibenzocycloheptenes |
-
1976
- 1976-06-30 CA CA256,080A patent/CA1092105A/en not_active Expired
- 1976-06-30 PT PT65295A patent/PT65295B/pt unknown
- 1976-06-30 FR FR7619897A patent/FR2315935A1/fr active Granted
- 1976-07-01 GR GR51162A patent/GR60851B/el unknown
- 1976-07-01 ES ES449432A patent/ES449432A1/es not_active Expired
- 1976-07-01 GB GB27487/76A patent/GB1499047A/en not_active Expired
- 1976-07-01 BE BE168549A patent/BE843678A/xx not_active IP Right Cessation
- 1976-07-01 SE SE7607534A patent/SE424076B/xx not_active IP Right Cessation
- 1976-07-01 CY CY1091A patent/CY1091A/xx unknown
- 1976-07-01 AU AU15488/76A patent/AU499122B2/en not_active Expired
- 1976-07-01 CH CH844376A patent/CH626366A5/de not_active IP Right Cessation
- 1976-07-02 HU HU76ME2001A patent/HU177866B/hu unknown
- 1976-07-02 DE DE19762629877 patent/DE2629877A1/de active Granted
- 1976-07-02 JP JP51077992A patent/JPS527996A/ja active Granted
- 1976-07-02 NL NLAANVRAGE7607347,A patent/NL188287C/xx not_active IP Right Cessation
- 1976-07-02 DE DE2661014A patent/DE2661014C2/de not_active Expired
- 1976-07-02 ZA ZA00763990A patent/ZA763990B/xx unknown
-
1980
- 1980-05-16 CH CH386180A patent/CH626617A5/de not_active IP Right Cessation
- 1980-05-16 CH CH385980A patent/CH626893A5/de not_active IP Right Cessation
- 1980-05-16 CH CH386280A patent/CH626618A5/de not_active IP Right Cessation
- 1980-05-16 CH CH386080A patent/CH626616A5/de not_active IP Right Cessation
- 1980-10-30 HK HK605/80A patent/HK60580A/xx unknown
-
1981
- 1981-12-30 MY MY227/81A patent/MY8100227A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NL7607347A (nl) | 1977-01-04 |
| SE424076B (sv) | 1982-06-28 |
| PT65295A (en) | 1976-07-01 |
| HK60580A (en) | 1980-11-07 |
| DE2661014C2 (cs) | 1989-01-05 |
| JPS527996A (en) | 1977-01-21 |
| ZA763990B (en) | 1978-02-22 |
| CA1092105A (en) | 1980-12-23 |
| ES449432A1 (es) | 1977-12-16 |
| AU1548876A (en) | 1978-01-05 |
| DE2629877A1 (de) | 1977-01-20 |
| CH626618A5 (en) | 1981-11-30 |
| NL188287C (nl) | 1992-05-18 |
| DE2629877C2 (cs) | 1989-01-05 |
| CH626617A5 (en) | 1981-11-30 |
| FR2315935B1 (cs) | 1978-11-17 |
| CY1091A (en) | 1980-12-27 |
| FR2315935A1 (fr) | 1977-01-28 |
| SE7607534L (sv) | 1977-01-03 |
| CH626616A5 (en) | 1981-11-30 |
| CH626366A5 (en) | 1981-11-13 |
| GB1499047A (en) | 1978-01-25 |
| PT65295B (en) | 1978-05-10 |
| AU499122B2 (en) | 1979-04-05 |
| GR60851B (en) | 1978-08-31 |
| NL188287B (nl) | 1991-12-16 |
| HU177866B (en) | 1982-01-28 |
| DE2661014A1 (cs) | 1985-07-04 |
| BE843678A (fr) | 1977-01-03 |
| CH626893A5 (en) | 1981-12-15 |
| MY8100227A (en) | 1981-12-31 |
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