JP7794807B2 - 気道疾患の治療に使用するための（１ｒ，３ｓ）－３－（（５－シアノ－４－フェニルチアゾール－２－イル）カルバモイル）シクロペンタン－１－カルボン酸およびその誘導体 - Google Patents
気道疾患の治療に使用するための（１ｒ，３ｓ）－３－（（５－シアノ－４－フェニルチアゾール－２－イル）カルバモイル）シクロペンタン－１－カルボン酸およびその誘導体Info
- Publication number
- JP7794807B2 JP7794807B2 JP2023512647A JP2023512647A JP7794807B2 JP 7794807 B2 JP7794807 B2 JP 7794807B2 JP 2023512647 A JP2023512647 A JP 2023512647A JP 2023512647 A JP2023512647 A JP 2023512647A JP 7794807 B2 JP7794807 B2 JP 7794807B2
- Authority
- JP
- Japan
- Prior art keywords
- asthma
- compound
- treatment
- pharmaceutical composition
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP20382764.7 | 2020-08-21 | ||
| EP20382764.7A EP3957308A1 (en) | 2020-08-21 | 2020-08-21 | (1r,3s)-3-((5-cyano-4-phenylthiazol-2-yl)carbamoyl)cyclopentane-1-carboxylic acid and derivatives thereof for use in the treatment of airway diseases |
| PCT/EP2021/073133 WO2022038261A1 (en) | 2020-08-21 | 2021-08-20 | (1r,3s)-3-((5-cyano-4-phenylthiazol-2-yl)carbamoyl)cyclopentane-1-carboxylic acid and derivatives thereof for use in the treatment of airway diseases |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2023538419A JP2023538419A (ja) | 2023-09-07 |
| JPWO2022038261A5 JPWO2022038261A5 (https=) | 2024-07-29 |
| JP2023538419A5 JP2023538419A5 (https=) | 2024-07-29 |
| JP7794807B2 true JP7794807B2 (ja) | 2026-01-06 |
Family
ID=72234795
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023512647A Active JP7794807B2 (ja) | 2020-08-21 | 2021-08-20 | 気道疾患の治療に使用するための（１ｒ，３ｓ）－３－（（５－シアノ－４－フェニルチアゾール－２－イル）カルバモイル）シクロペンタン－１－カルボン酸およびその誘導体 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US20230321053A1 (https=) |
| EP (2) | EP3957308A1 (https=) |
| JP (1) | JP7794807B2 (https=) |
| KR (1) | KR20230054444A (https=) |
| CN (1) | CN115942933A (https=) |
| AU (1) | AU2021327728A1 (https=) |
| BR (1) | BR112023002778A2 (https=) |
| CA (1) | CA3190081A1 (https=) |
| DK (1) | DK4199922T3 (https=) |
| ES (1) | ES3001104T3 (https=) |
| FI (1) | FI4199922T3 (https=) |
| HR (1) | HRP20241621T1 (https=) |
| HU (1) | HUE069338T2 (https=) |
| LT (1) | LT4199922T (https=) |
| MX (1) | MX2023002156A (https=) |
| PL (1) | PL4199922T3 (https=) |
| PT (1) | PT4199922T (https=) |
| RS (1) | RS66263B1 (https=) |
| SI (1) | SI4199922T1 (https=) |
| WO (1) | WO2022038261A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102460040B1 (ko) | 2016-04-27 | 2022-11-01 | 애브비 인코포레이티드 | 항-il-13 항체를 이용한 il-13 활성이 유해한 질환의 치료 방법 |
| US12162940B2 (en) | 2021-05-05 | 2024-12-10 | Immatics Biotechnologies Gmbh | BMA031 antigen binding polypeptides |
Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009529539A (ja) | 2006-03-07 | 2009-08-20 | エンダセア， インコーポレイテッド | 呼吸器障害を治療するための方法および組成物 |
| JP2010540615A (ja) | 2007-10-02 | 2010-12-24 | パロビオファルマ，エス．エル． | アデノシンａ１レセプターアンタゴニストとしての新規化合物 |
| WO2016040007A1 (en) | 2014-09-08 | 2016-03-17 | Cephalon, Inc. | Use of reslizumab to treat moderate to severe eosinophilic asthma |
| JP2019203009A (ja) | 2013-10-15 | 2019-11-28 | アストラゼネカ アクチボラグ | ベンラリズマブを使用して慢性閉塞性肺疾患を治療するための方法 |
| JP2020505349A (ja) | 2017-01-20 | 2020-02-20 | パロビオファルマ、ソシエダッド、リミターダＰａｌｏｂｉｏｆａｒｍａ Ｓ．Ｌ | アデノシンａ３受容体の調節剤 |
| JP2020509066A (ja) | 2017-03-06 | 2020-03-26 | パロビオファルマ、ソシエダッド、リミターダＰａｌｏｂｉｏｆａｒｍａ Ｓ．Ｌ | （１ｒ，３ｓ）−３−（５−シアノ−４−フェニル−１，３−チアゾール−２−イルカルバモイル）シクロペンタンカルボン酸のアミン塩 |
-
2020
- 2020-08-21 EP EP20382764.7A patent/EP3957308A1/en not_active Withdrawn
-
2021
- 2021-08-20 RS RS20241285A patent/RS66263B1/sr unknown
- 2021-08-20 CA CA3190081A patent/CA3190081A1/en active Pending
- 2021-08-20 MX MX2023002156A patent/MX2023002156A/es unknown
- 2021-08-20 PL PL21765908.5T patent/PL4199922T3/pl unknown
- 2021-08-20 HU HUE21765908A patent/HUE069338T2/hu unknown
- 2021-08-20 FI FIEP21765908.5T patent/FI4199922T3/fi active
- 2021-08-20 DK DK21765908.5T patent/DK4199922T3/da active
- 2021-08-20 AU AU2021327728A patent/AU2021327728A1/en active Pending
- 2021-08-20 KR KR1020237009717A patent/KR20230054444A/ko active Pending
- 2021-08-20 CN CN202180051106.2A patent/CN115942933A/zh active Pending
- 2021-08-20 HR HRP20241621TT patent/HRP20241621T1/hr unknown
- 2021-08-20 LT LTEPPCT/EP2021/073133T patent/LT4199922T/lt unknown
- 2021-08-20 US US18/040,508 patent/US20230321053A1/en active Pending
- 2021-08-20 WO PCT/EP2021/073133 patent/WO2022038261A1/en not_active Ceased
- 2021-08-20 BR BR112023002778A patent/BR112023002778A2/pt unknown
- 2021-08-20 PT PT217659085T patent/PT4199922T/pt unknown
- 2021-08-20 EP EP21765908.5A patent/EP4199922B1/en active Active
- 2021-08-20 ES ES21765908T patent/ES3001104T3/es active Active
- 2021-08-20 JP JP2023512647A patent/JP7794807B2/ja active Active
- 2021-08-20 SI SI202130242T patent/SI4199922T1/sl unknown
Patent Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009529539A (ja) | 2006-03-07 | 2009-08-20 | エンダセア， インコーポレイテッド | 呼吸器障害を治療するための方法および組成物 |
| JP2010540615A (ja) | 2007-10-02 | 2010-12-24 | パロビオファルマ，エス．エル． | アデノシンａ１レセプターアンタゴニストとしての新規化合物 |
| JP2019203009A (ja) | 2013-10-15 | 2019-11-28 | アストラゼネカ アクチボラグ | ベンラリズマブを使用して慢性閉塞性肺疾患を治療するための方法 |
| WO2016040007A1 (en) | 2014-09-08 | 2016-03-17 | Cephalon, Inc. | Use of reslizumab to treat moderate to severe eosinophilic asthma |
| JP2020505349A (ja) | 2017-01-20 | 2020-02-20 | パロビオファルマ、ソシエダッド、リミターダＰａｌｏｂｉｏｆａｒｍａ Ｓ．Ｌ | アデノシンａ３受容体の調節剤 |
| JP2020509066A (ja) | 2017-03-06 | 2020-03-26 | パロビオファルマ、ソシエダッド、リミターダＰａｌｏｂｉｏｆａｒｍａ Ｓ．Ｌ | （１ｒ，３ｓ）−３−（５−シアノ−４−フェニル−１，３−チアゾール−２−イルカルバモイル）シクロペンタンカルボン酸のアミン塩 |
Non-Patent Citations (3)
| Title |
|---|
| Current Pharmaceutical Design，2019年，Vol. 25, No. 26，pp.2792-2807 |
| European journal of pharmacology，2006年，Vol. 551, No. 1-3，pp.116-124 |
| Trends in pharmacological sciences，2009年，Vol. 30, No. 10，pp.528-535 |
Also Published As
| Publication number | Publication date |
|---|---|
| US20230321053A1 (en) | 2023-10-12 |
| EP3957308A1 (en) | 2022-02-23 |
| RS66263B1 (sr) | 2024-12-31 |
| JP2023538419A (ja) | 2023-09-07 |
| EP4199922B1 (en) | 2024-09-25 |
| DK4199922T3 (da) | 2024-11-25 |
| SI4199922T1 (sl) | 2025-03-31 |
| HRP20241621T1 (hr) | 2025-01-31 |
| KR20230054444A (ko) | 2023-04-24 |
| PT4199922T (pt) | 2024-12-18 |
| BR112023002778A2 (pt) | 2023-03-14 |
| LT4199922T (lt) | 2025-01-10 |
| AU2021327728A1 (en) | 2023-03-09 |
| CA3190081A1 (en) | 2022-02-24 |
| FI4199922T3 (fi) | 2024-12-05 |
| HUE069338T2 (hu) | 2025-02-28 |
| WO2022038261A1 (en) | 2022-02-24 |
| EP4199922A1 (en) | 2023-06-28 |
| MX2023002156A (es) | 2023-03-01 |
| ES3001104T3 (es) | 2025-03-04 |
| CN115942933A (zh) | 2023-04-07 |
| PL4199922T3 (pl) | 2025-02-10 |
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