JP7395480B2 - フェニルスルホンアミドを含む薬学的組成物、及びそれらの治療的適用 - Google Patents

フェニルスルホンアミドを含む薬学的組成物、及びそれらの治療的適用 Download PDF

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JP7395480B2
JP7395480B2 JP2020538987A JP2020538987A JP7395480B2 JP 7395480 B2 JP7395480 B2 JP 7395480B2 JP 2020538987 A JP2020538987 A JP 2020538987A JP 2020538987 A JP2020538987 A JP 2020538987A JP 7395480 B2 JP7395480 B2 JP 7395480B2
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デウジ ナズニーン
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クラ セラピューティクス, エルエルシー
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/18Sulfonamides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/63Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents

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  • Pharmacology & Pharmacy (AREA)
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  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
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  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Psychology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2020538987A 2018-01-10 2019-01-08 フェニルスルホンアミドを含む薬学的組成物、及びそれらの治療的適用 Active JP7395480B2 (ja)

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JP2023144990A JP2023182589A (ja) 2018-01-10 2023-09-07 フェニルスルホンアミドを含む薬学的組成物、及びそれらの治療的適用
JP2025165134A JP2026021312A (ja) 2018-01-10 2025-10-01 フェニルスルホンアミドを含む薬学的組成物、及びそれらの治療的適用

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US201862615869P 2018-01-10 2018-01-10
US62/615,869 2018-01-10
PCT/US2019/012608 WO2019139869A1 (en) 2018-01-10 2019-01-08 Pharmaceutical compositions comprising phenylsulfonamides, and their therapeutic applications

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JPWO2019139869A5 JPWO2019139869A5 (https=) 2022-01-18
JP2021510168A5 JP2021510168A5 (https=) 2022-01-18
JP7395480B2 true JP7395480B2 (ja) 2023-12-11

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JP2023144990A Pending JP2023182589A (ja) 2018-01-10 2023-09-07 フェニルスルホンアミドを含む薬学的組成物、及びそれらの治療的適用
JP2025165134A Pending JP2026021312A (ja) 2018-01-10 2025-10-01 フェニルスルホンアミドを含む薬学的組成物、及びそれらの治療的適用

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JP2025165134A Pending JP2026021312A (ja) 2018-01-10 2025-10-01 フェニルスルホンアミドを含む薬学的組成物、及びそれらの治療的適用

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US (3) US11701334B2 (https=)
EP (1) EP3737382A1 (https=)
JP (3) JP7395480B2 (https=)
AU (2) AU2019207491A1 (https=)
CA (1) CA3087856A1 (https=)
TW (2) TWI823890B (https=)
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JP7395480B2 (ja) 2018-01-10 2023-12-11 クラ セラピューティクス, エルエルシー フェニルスルホンアミドを含む薬学的組成物、及びそれらの治療的適用
EP3997068A1 (en) * 2019-07-11 2022-05-18 Cura Therapeutics, LLC Sulfone compounds and pharmaceutical compositions thereof, and their therapeutic applications for the treatment of neurodegenerative diseases
CA3146159A1 (en) * 2019-07-11 2021-01-14 Cura Therapeutics, Llc Phenyl compounds and pharmaceutical compositions thereof, and their therapeutic applications

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