JP6541687B2 - 中鎖グリセリドを含有する即時放出フィルムコーティング、及びそれによってコーティングされている基材 - Google Patents

中鎖グリセリドを含有する即時放出フィルムコーティング、及びそれによってコーティングされている基材 Download PDF

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JP6541687B2
JP6541687B2 JP2016565103A JP2016565103A JP6541687B2 JP 6541687 B2 JP6541687 B2 JP 6541687B2 JP 2016565103 A JP2016565103 A JP 2016565103A JP 2016565103 A JP2016565103 A JP 2016565103A JP 6541687 B2 JP6541687 B2 JP 6541687B2
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film coating
coating composition
composition according
medium chain
weight
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Japanese (ja)
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JP2017509691A5 (enExample
JP2017509691A (ja
Inventor
テッコー，ジェーソン
ジェイ． プルサク，ブラッドリー
ジェイ． プルサク，ブラッドリー
アール． ギンベル，ジェフリー
アール． ギンベル，ジェフリー
トゥー，ダニエル
Original Assignee
ビーピーエスアイ ホールディングス， エルエルシー
ビーピーエスアイ ホールディングス， エルエルシー
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/282—Organic compounds, e.g. fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2813—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2893—Tablet coating processes
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08J—WORKING-UP; GENERAL PROCESSES OF COMPOUNDING; AFTER-TREATMENT NOT COVERED BY SUBCLASSES C08B, C08C, C08F, C08G or C08H
    • C08J3/00—Processes of treating or compounding macromolecular substances
    • C08J3/02—Making solutions, dispersions, lattices or gels by other methods than by solution, emulsion or suspension polymerisation techniques
    • C08J3/03—Making solutions, dispersions, lattices or gels by other methods than by solution, emulsion or suspension polymerisation techniques in aqueous media

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Inorganic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Polymers & Plastics (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Application Of Or Painting With Fluid Materials (AREA)
  • Paints Or Removers (AREA)
JP2016565103A 2014-01-21 2015-01-14 中鎖グリセリドを含有する即時放出フィルムコーティング、及びそれによってコーティングされている基材 Active JP6541687B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461929735P 2014-01-21 2014-01-21
US61/929,735 2014-01-21
PCT/US2015/011422 WO2015112400A1 (en) 2014-01-21 2015-01-14 Immediate release film coatings containing medium chain glycerides and substrates coated therewith

Publications (3)

Publication Number Publication Date
JP2017509691A JP2017509691A (ja) 2017-04-06
JP2017509691A5 JP2017509691A5 (enExample) 2018-02-01
JP6541687B2 true JP6541687B2 (ja) 2019-07-10

Family

ID=53543848

Family Applications (1)

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JP2016565103A Active JP6541687B2 (ja) 2014-01-21 2015-01-14 中鎖グリセリドを含有する即時放出フィルムコーティング、及びそれによってコーティングされている基材

Country Status (14)

Country Link
US (2) US9504654B2 (enExample)
EP (1) EP3096891B1 (enExample)
JP (1) JP6541687B2 (enExample)
KR (1) KR102287342B1 (enExample)
CN (1) CN105916598B (enExample)
AU (1) AU2015209674B2 (enExample)
BR (1) BR112016016623B1 (enExample)
CA (1) CA2933202C (enExample)
ES (1) ES2802156T3 (enExample)
HU (1) HUE049598T2 (enExample)
MX (1) MX378845B (enExample)
PL (1) PL3096891T3 (enExample)
RU (1) RU2686183C2 (enExample)
WO (1) WO2015112400A1 (enExample)

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KR102158339B1 (ko) * 2016-02-05 2020-09-21 삼진제약주식회사 인습성이 개선된 카르베딜롤 속방성 제제
US10232045B2 (en) * 2016-08-04 2019-03-19 Bpsi Holdings Llc Easy to swallow coatings and substrates coated therewith
US20180338922A1 (en) * 2017-05-26 2018-11-29 Esperion Therapeutics, Inc. Fixed dose formulations
TR201721437A2 (tr) * 2017-12-25 2019-07-22 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Fesoterodi̇ni̇n modi̇fi̇ye salim sağlayan formülasyonlari
KR102103530B1 (ko) 2018-06-29 2020-04-22 주식회사 코피텍 필름 코팅용 조성물 및 이를 코팅한 정제
KR102265977B1 (ko) 2018-07-16 2021-06-16 주식회사 코피텍 방습성이 개선된 필름 코팅용 조성물 및 이를 코팅한 정제
EP4417220A4 (en) * 2021-10-11 2025-10-08 Towa Pharmaceutical Co Ltd METHOD FOR PRODUCING A LIQUID MIXTURE, LIQUID MIXTURE AND SOLID COMPOSITION

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JPS59193831A (ja) * 1983-04-18 1984-11-02 Sankyo Co Ltd 腸溶性製剤の製造法
US6248363B1 (en) * 1999-11-23 2001-06-19 Lipocine, Inc. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
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IL162293A0 (en) * 2001-12-19 2005-11-20 Alza Corp Formulation and dosage form for increasing oral bioavailability of hydrophilic macromolecules
FR2838647B1 (fr) * 2002-04-23 2006-02-17 Particules enrobees a liberation prolongee, leur procede de preparation et comprimes les contenant
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Also Published As

Publication number Publication date
BR112016016623B1 (pt) 2022-02-01
EP3096891B1 (en) 2020-04-08
CA2933202C (en) 2022-05-31
AU2015209674B2 (en) 2018-11-08
WO2015112400A1 (en) 2015-07-30
US20170035697A1 (en) 2017-02-09
HUE049598T2 (hu) 2020-09-28
MX378845B (es) 2025-03-10
KR102287342B1 (ko) 2021-08-06
RU2686183C2 (ru) 2019-04-24
EP3096891A1 (en) 2016-11-30
CN105916598B (zh) 2020-07-17
BR112016016623A2 (enExample) 2017-08-08
CN105916598A (zh) 2016-08-31
EP3096891A4 (en) 2017-10-04
KR20160111375A (ko) 2016-09-26
RU2016133221A3 (enExample) 2018-07-17
US20150202160A1 (en) 2015-07-23
ES2802156T3 (es) 2021-01-15
US9504654B2 (en) 2016-11-29
RU2016133221A (ru) 2018-03-02
CA2933202A1 (en) 2015-07-30
AU2015209674A1 (en) 2016-06-23
US9789067B2 (en) 2017-10-17
PL3096891T3 (pl) 2020-08-24
MX2016008583A (es) 2017-02-02
JP2017509691A (ja) 2017-04-06

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