CN105916598B - 含有中链甘油酯的即释型膜包衣及用其包被的基质 - Google Patents

含有中链甘油酯的即释型膜包衣及用其包被的基质 Download PDF

Info

Publication number
CN105916598B
CN105916598B CN201580005058.8A CN201580005058A CN105916598B CN 105916598 B CN105916598 B CN 105916598B CN 201580005058 A CN201580005058 A CN 201580005058A CN 105916598 B CN105916598 B CN 105916598B
Authority
CN
China
Prior art keywords
film coating
coating composition
medium chain
glycerides
chain glycerides
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
CN201580005058.8A
Other languages
English (en)
Chinese (zh)
Other versions
CN105916598A (zh
Inventor
J·特克伊
B·J·普鲁萨克
J·R·金贝儿
D·杜
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BPSI Holdings LLC
Original Assignee
BPSI Holdings LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BPSI Holdings LLC filed Critical BPSI Holdings LLC
Publication of CN105916598A publication Critical patent/CN105916598A/zh
Application granted granted Critical
Publication of CN105916598B publication Critical patent/CN105916598B/zh
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2813—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/282—Organic compounds, e.g. fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2893—Tablet coating processes
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08J—WORKING-UP; GENERAL PROCESSES OF COMPOUNDING; AFTER-TREATMENT NOT COVERED BY SUBCLASSES C08B, C08C, C08F, C08G or C08H
    • C08J3/00—Processes of treating or compounding macromolecular substances
    • C08J3/02—Making solutions, dispersions, lattices or gels by other methods than by solution, emulsion or suspension polymerisation techniques
    • C08J3/03—Making solutions, dispersions, lattices or gels by other methods than by solution, emulsion or suspension polymerisation techniques in aqueous media

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Inorganic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Polymers & Plastics (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Application Of Or Painting With Fluid Materials (AREA)
  • Paints Or Removers (AREA)
CN201580005058.8A 2014-01-21 2015-01-14 含有中链甘油酯的即释型膜包衣及用其包被的基质 Active CN105916598B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461929735P 2014-01-21 2014-01-21
US61/929,735 2014-01-21
PCT/US2015/011422 WO2015112400A1 (en) 2014-01-21 2015-01-14 Immediate release film coatings containing medium chain glycerides and substrates coated therewith

Publications (2)

Publication Number Publication Date
CN105916598A CN105916598A (zh) 2016-08-31
CN105916598B true CN105916598B (zh) 2020-07-17

Family

ID=53543848

Family Applications (1)

Application Number Title Priority Date Filing Date
CN201580005058.8A Active CN105916598B (zh) 2014-01-21 2015-01-14 含有中链甘油酯的即释型膜包衣及用其包被的基质

Country Status (14)

Country Link
US (2) US9504654B2 (enExample)
EP (1) EP3096891B1 (enExample)
JP (1) JP6541687B2 (enExample)
KR (1) KR102287342B1 (enExample)
CN (1) CN105916598B (enExample)
AU (1) AU2015209674B2 (enExample)
BR (1) BR112016016623B1 (enExample)
CA (1) CA2933202C (enExample)
ES (1) ES2802156T3 (enExample)
HU (1) HUE049598T2 (enExample)
MX (1) MX378845B (enExample)
PL (1) PL3096891T3 (enExample)
RU (1) RU2686183C2 (enExample)
WO (1) WO2015112400A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102158339B1 (ko) * 2016-02-05 2020-09-21 삼진제약주식회사 인습성이 개선된 카르베딜롤 속방성 제제
US10232045B2 (en) * 2016-08-04 2019-03-19 Bpsi Holdings Llc Easy to swallow coatings and substrates coated therewith
US20180338922A1 (en) * 2017-05-26 2018-11-29 Esperion Therapeutics, Inc. Fixed dose formulations
TR201721437A2 (tr) * 2017-12-25 2019-07-22 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Fesoterodi̇ni̇n modi̇fi̇ye salim sağlayan formülasyonlari
KR102103530B1 (ko) 2018-06-29 2020-04-22 주식회사 코피텍 필름 코팅용 조성물 및 이를 코팅한 정제
KR102265977B1 (ko) 2018-07-16 2021-06-16 주식회사 코피텍 방습성이 개선된 필름 코팅용 조성물 및 이를 코팅한 정제
EP4417220A4 (en) * 2021-10-11 2025-10-08 Towa Pharmaceutical Co Ltd METHOD FOR PRODUCING A LIQUID MIXTURE, LIQUID MIXTURE AND SOLID COMPOSITION

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102421421A (zh) * 2009-05-12 2012-04-18 Bpsi控股有限责任公司 含有抗黏性剂细微颗粒的包衣和覆有该包衣的基体

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57171428A (en) * 1981-04-13 1982-10-22 Sankyo Co Ltd Preparation of coated solid preparation
DE3220434A1 (de) 1982-05-29 1983-12-01 Robert Bosch Gmbh, 7000 Stuttgart Verfahren zur ueberwachung einer messgroesse
JPS5973529A (ja) 1982-10-12 1984-04-25 Sankyo Co Ltd 被覆固形製剤の製造法
JPS59193831A (ja) * 1983-04-18 1984-11-02 Sankyo Co Ltd 腸溶性製剤の製造法
US6248363B1 (en) * 1999-11-23 2001-06-19 Lipocine, Inc. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
US6448323B1 (en) * 1999-07-09 2002-09-10 Bpsi Holdings, Inc. Film coatings and film coating compositions based on polyvinyl alcohol
KR100425226B1 (ko) * 2001-07-03 2004-03-30 주식회사 팜트리 아세클로페낙을 함유하는 경제적인 경구용 제제의 조성 및제법
IL162293A0 (en) * 2001-12-19 2005-11-20 Alza Corp Formulation and dosage form for increasing oral bioavailability of hydrophilic macromolecules
FR2838647B1 (fr) * 2002-04-23 2006-02-17 Particules enrobees a liberation prolongee, leur procede de preparation et comprimes les contenant
DE10311585A1 (de) * 2003-03-14 2004-09-23 Basf Ag Wirkstoffhaltige Adsorbate
EP1729742A1 (en) * 2004-03-31 2006-12-13 BPSI Holdings, Inc. Enteric coatings for orally ingestible substrates
TWI415635B (zh) * 2004-05-28 2013-11-21 必治妥施貴寶公司 加衣錠片調製物及製備彼之方法
US20080096979A1 (en) * 2004-11-08 2008-04-24 Rubicon Research Pvt. Ltd. Aqueous Pharmaceutical Coating
WO2006111980A2 (en) * 2005-04-20 2006-10-26 Ideal Cures Pvt. Ltd. Pva based film coating and film coating compositions
JP2007217390A (ja) * 2006-02-20 2007-08-30 Hitoshi Ichihashi カプリロカプロイルマクロゴール−８グリセリドを含む医薬組成物
US20080181928A1 (en) 2006-12-22 2008-07-31 Miv Therapeutics, Inc. Coatings for implantable medical devices for liposome delivery
US8883176B2 (en) 2008-09-25 2014-11-11 Isp Investments Inc. Smooth, high solids tablet coating composition
TWI438012B (zh) 2008-12-25 2014-05-21 Toray Industries 固態製劑用之塗覆劑及使用其之固態製劑
WO2010112965A1 (en) * 2009-03-30 2010-10-07 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi Isolation coating of diclofenac tablets
WO2010122583A2 (en) 2009-04-24 2010-10-28 Rubicon Research Private Limited Oral pharmaceutical compositions of acid labile substances
MX2011011919A (es) * 2009-05-12 2012-01-27 Bpsi Holdings Llc Sistemas de recubrimiento de pelicula de liberacion inmediata con barrera contra humedad mejorada y sustratos recubiertos con dichos sistemas.
CN102655858B (zh) * 2009-12-22 2015-11-25 Abbvie公司 Abt-263胶囊
EP2544546A4 (en) * 2010-03-08 2014-10-15 Sensient Colors Inc FOOD-SPIRITUAL DRYING COATING COMPOSITION AND METHOD FOR THE PRODUCTION AND USE THEREOF
WO2012120364A2 (en) * 2011-03-09 2012-09-13 Ideal Cures Pvt. Ltd. Novel immediate release film coating compositions
WO2014090859A1 (en) * 2012-12-12 2014-06-19 Leo Laboratories Limited Gel compositions
WO2014096983A1 (en) * 2012-12-21 2014-06-26 Wockhardt Limited Stable pharmaceutical compositions of saxagliptin or salts thereof
GB201319792D0 (en) * 2013-11-08 2013-12-25 Sigmoid Pharma Ltd Formulations

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102421421A (zh) * 2009-05-12 2012-04-18 Bpsi控股有限责任公司 含有抗黏性剂细微颗粒的包衣和覆有该包衣的基体

Also Published As

Publication number Publication date
BR112016016623B1 (pt) 2022-02-01
EP3096891B1 (en) 2020-04-08
CA2933202C (en) 2022-05-31
AU2015209674B2 (en) 2018-11-08
WO2015112400A1 (en) 2015-07-30
US20170035697A1 (en) 2017-02-09
HUE049598T2 (hu) 2020-09-28
MX378845B (es) 2025-03-10
KR102287342B1 (ko) 2021-08-06
RU2686183C2 (ru) 2019-04-24
EP3096891A1 (en) 2016-11-30
BR112016016623A2 (enExample) 2017-08-08
CN105916598A (zh) 2016-08-31
EP3096891A4 (en) 2017-10-04
KR20160111375A (ko) 2016-09-26
RU2016133221A3 (enExample) 2018-07-17
US20150202160A1 (en) 2015-07-23
JP6541687B2 (ja) 2019-07-10
ES2802156T3 (es) 2021-01-15
US9504654B2 (en) 2016-11-29
RU2016133221A (ru) 2018-03-02
CA2933202A1 (en) 2015-07-30
AU2015209674A1 (en) 2016-06-23
US9789067B2 (en) 2017-10-17
PL3096891T3 (pl) 2020-08-24
MX2016008583A (es) 2017-02-02
JP2017509691A (ja) 2017-04-06

Similar Documents

Publication Publication Date Title
CN105916598B (zh) 含有中链甘油酯的即释型膜包衣及用其包被的基质
EP2429505B1 (en) Enhanced moisture barrier immediate release film coating systems and substrates coated therewith
AU2014223658B2 (en) Delayed release film coatings containing calcium silicate and substrates coated therewith
EP2429504A1 (en) Film coatings containing fine particle size detackifiers and substrates coated therewith
CA3031671C (en) EASY-TO-SWALLOW COATINGS AND SUBSTRATES COATED WITH THESE

Legal Events

Date Code Title Description
C06 Publication
PB01 Publication
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
GR01 Patent grant
GR01 Patent grant