JP6531100B2 - キナーゼ阻害剤としての置換ニコチンアミド誘導体 - Google Patents
キナーゼ阻害剤としての置換ニコチンアミド誘導体 Download PDFInfo
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- JP6531100B2 JP6531100B2 JP2016538520A JP2016538520A JP6531100B2 JP 6531100 B2 JP6531100 B2 JP 6531100B2 JP 2016538520 A JP2016538520 A JP 2016538520A JP 2016538520 A JP2016538520 A JP 2016538520A JP 6531100 B2 JP6531100 B2 JP 6531100B2
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- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
- C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D411/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
- C07D411/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
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- Health & Medical Sciences (AREA)
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| US201361915186P | 2013-12-12 | 2013-12-12 | |
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| US61/915,209 | 2013-12-12 | ||
| PCT/US2014/069601 WO2015089220A1 (en) | 2013-12-12 | 2014-12-10 | Substituted nicotinamide derivatives as kinase inhibitors |
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| US10046649B2 (en) | 2012-06-28 | 2018-08-14 | Midtronics, Inc. | Hybrid and electric vehicle battery pack maintenance device |
| US20110300416A1 (en) | 2010-06-03 | 2011-12-08 | Bertness Kevin I | Battery pack maintenance for electric vehicle |
| US11740294B2 (en) | 2010-06-03 | 2023-08-29 | Midtronics, Inc. | High use battery pack maintenance |
| DE112012004706T5 (de) | 2011-11-10 | 2014-08-21 | Midtronics, Inc. | Batteriepack-Testvorrichtung |
| US11325479B2 (en) | 2012-06-28 | 2022-05-10 | Midtronics, Inc. | Hybrid and electric vehicle battery maintenance device |
| US10843574B2 (en) | 2013-12-12 | 2020-11-24 | Midtronics, Inc. | Calibration and programming of in-vehicle battery sensors |
| US10473555B2 (en) | 2014-07-14 | 2019-11-12 | Midtronics, Inc. | Automotive maintenance system |
| US10317468B2 (en) | 2015-01-26 | 2019-06-11 | Midtronics, Inc. | Alternator tester |
| US10608353B2 (en) | 2016-06-28 | 2020-03-31 | Midtronics, Inc. | Battery clamp |
| US12320857B2 (en) | 2016-10-25 | 2025-06-03 | Midtronics, Inc. | Electrical load for electronic battery tester and electronic battery tester including such electrical load |
| US11054480B2 (en) | 2016-10-25 | 2021-07-06 | Midtronics, Inc. | Electrical load for electronic battery tester and electronic battery tester including such electrical load |
| CN108456163A (zh) | 2017-02-20 | 2018-08-28 | 中国科学院上海药物研究所 | 含邻氨基杂芳环炔基的化合物及其制备方法和用途 |
| US11513160B2 (en) | 2018-11-29 | 2022-11-29 | Midtronics, Inc. | Vehicle battery maintenance device |
| CN111662227B (zh) * | 2019-03-06 | 2022-07-05 | 中国科学院上海药物研究所 | 邻氨基吡啶炔类化合物及其制备方法和用途 |
| US11566972B2 (en) | 2019-07-31 | 2023-01-31 | Midtronics, Inc. | Tire tread gauge using visual indicator |
| US11545839B2 (en) | 2019-11-05 | 2023-01-03 | Midtronics, Inc. | System for charging a series of connected batteries |
| US11668779B2 (en) | 2019-11-11 | 2023-06-06 | Midtronics, Inc. | Hybrid and electric vehicle battery pack maintenance device |
| US11474153B2 (en) | 2019-11-12 | 2022-10-18 | Midtronics, Inc. | Battery pack maintenance system |
| US11973202B2 (en) | 2019-12-31 | 2024-04-30 | Midtronics, Inc. | Intelligent module interface for battery maintenance device |
| DE102020216599A1 (de) | 2019-12-31 | 2021-07-01 | Midtronics, Inc. | Intelligente Modulschnittstelle für eine Batteriewartungsvorrichtung |
| US11486930B2 (en) | 2020-01-23 | 2022-11-01 | Midtronics, Inc. | Electronic battery tester with battery clamp storage holsters |
| US12330513B2 (en) | 2022-02-14 | 2025-06-17 | Midtronics, Inc. | Battery maintenance device with high voltage connector |
| US12392833B2 (en) | 2022-05-09 | 2025-08-19 | Midtronics, Inc. | Electronic battery tester |
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| US7915443B2 (en) * | 2006-11-16 | 2011-03-29 | Allergan, Inc. | Sulfoximines as kinase inhibitors |
| US8558002B2 (en) * | 2006-11-16 | 2013-10-15 | Allergan, Inc. | Sulfoximines as kinase inhibitors |
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| CA2932831A1 (en) | 2015-06-18 |
| BR112016013539A2 (pt) | 2020-10-27 |
| US20160194311A1 (en) | 2016-07-07 |
| AU2014362391B2 (en) | 2019-04-04 |
| CN105814021A (zh) | 2016-07-27 |
| CN105814021B (zh) | 2020-03-13 |
| US20150166518A1 (en) | 2015-06-18 |
| AU2014362391A1 (en) | 2016-06-16 |
| JP2016539995A (ja) | 2016-12-22 |
| US9567324B2 (en) | 2017-02-14 |
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