JP6403780B2 - 押出成形された持続放出性乱用抑止性丸剤 - Google Patents
押出成形された持続放出性乱用抑止性丸剤 Download PDFInfo
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- JP6403780B2 JP6403780B2 JP2016540580A JP2016540580A JP6403780B2 JP 6403780 B2 JP6403780 B2 JP 6403780B2 JP 2016540580 A JP2016540580 A JP 2016540580A JP 2016540580 A JP2016540580 A JP 2016540580A JP 6403780 B2 JP6403780 B2 JP 6403780B2
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Images
Classifications
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
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- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
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- Health & Medical Sciences (AREA)
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- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Neurology (AREA)
- Addiction (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Emergency Medicine (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (11)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361917120P | 2013-12-17 | 2013-12-17 | |
| US201361917074P | 2013-12-17 | 2013-12-17 | |
| US61/917,120 | 2013-12-17 | ||
| US61/917,074 | 2013-12-17 | ||
| US201461980259P | 2014-04-16 | 2014-04-16 | |
| US201461980254P | 2014-04-16 | 2014-04-16 | |
| US61/980,254 | 2014-04-16 | ||
| US61/980,259 | 2014-04-16 | ||
| US14/457,714 US10195153B2 (en) | 2013-08-12 | 2014-08-12 | Extruded immediate release abuse deterrent pill |
| US14/457,714 | 2014-08-12 | ||
| PCT/US2014/070942 WO2015095387A1 (en) | 2013-12-17 | 2014-12-17 | Extruded extended release abuse deterrent pill |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| JP2018169278A Division JP6678212B2 (ja) | 2013-12-17 | 2018-09-11 | 押出成形された持続放出性乱用抑止性丸剤 |
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| JP2017503780A JP2017503780A (ja) | 2017-02-02 |
| JP6403780B2 true JP6403780B2 (ja) | 2018-10-10 |
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| JP2018169278A Expired - Fee Related JP6678212B2 (ja) | 2013-12-17 | 2018-09-11 | 押出成形された持続放出性乱用抑止性丸剤 |
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| JP2018169278A Expired - Fee Related JP6678212B2 (ja) | 2013-12-17 | 2018-09-11 | 押出成形された持続放出性乱用抑止性丸剤 |
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| EP (1) | EP3082775A4 (enExample) |
| JP (2) | JP6403780B2 (enExample) |
| AU (3) | AU2014364800A1 (enExample) |
| CA (1) | CA2934078C (enExample) |
| WO (1) | WO2015095387A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2019001816A (ja) * | 2013-12-17 | 2019-01-10 | ファーマシューティカル マニュファクチュアリング リサーチ サービシズ，インコーポレーテッド | 押出成形された持続放出性乱用抑止性丸剤 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| IL273627B2 (en) | 2017-12-20 | 2025-03-01 | Purdue Pharma Lp | Morphine sulfate dosage forms for abuse deterrence |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| EP2065055A1 (en) * | 1996-06-26 | 2009-06-03 | Board of Regents, The University of Texas System | Holt-melt extrudable pharmaceutical formulation |
| FI1765303T4 (fi) * | 2004-07-01 | 2023-01-31 | Väärinkäytöltä suojattu oraalinen tabletti | |
| US20080152595A1 (en) * | 2004-11-24 | 2008-06-26 | Acura Pharmaceuticals, Inc. | Methods and compositions for deterring abuse of orally administered pharmaceutical products |
| DE102007011485A1 (de) * | 2007-03-07 | 2008-09-11 | Grünenthal GmbH | Darreichungsform mit erschwertem Missbrauch |
| GB0909680D0 (en) * | 2009-06-05 | 2009-07-22 | Euro Celtique Sa | Dosage form |
| EA201400172A1 (ru) * | 2011-07-29 | 2014-06-30 | Грюненталь Гмбх | Устойчивая к разрушению таблетка, которая обеспечивает немедленное высвобождение лекарственного средства |
| ES2644935T3 (es) * | 2012-04-18 | 2017-12-01 | Mallinckrodt Llc | Composiciones farmacéuticas de liberación inmediata con propiedades disuasorias del abuso |
| US9549899B2 (en) * | 2012-07-06 | 2017-01-24 | Egalet Ltd. | Abuse deterrent pharmaceutical compositions for controlled release |
| CA2919892C (en) * | 2013-08-12 | 2019-06-18 | Pharmaceutical Manufacturing Research Services, Inc. | Extruded immediate release abuse deterrent pill |
| AU2014364800A1 (en) * | 2013-12-17 | 2016-07-07 | Pharmaceutical Manufacturing Research Services, Inc. | Extruded extended release abuse deterrent pill |
-
2014
- 2014-12-17 AU AU2014364800A patent/AU2014364800A1/en not_active Abandoned
- 2014-12-17 EP EP14871095.7A patent/EP3082775A4/en not_active Withdrawn
- 2014-12-17 WO PCT/US2014/070942 patent/WO2015095387A1/en not_active Ceased
- 2014-12-17 CA CA2934078A patent/CA2934078C/en not_active Expired - Fee Related
- 2014-12-17 JP JP2016540580A patent/JP6403780B2/ja not_active Expired - Fee Related
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2018
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2019
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2019001816A (ja) * | 2013-12-17 | 2019-01-10 | ファーマシューティカル マニュファクチュアリング リサーチ サービシズ，インコーポレーテッド | 押出成形された持続放出性乱用抑止性丸剤 |
Also Published As
| Publication number | Publication date |
|---|---|
| CA2934078C (en) | 2019-08-06 |
| CA2934078A1 (en) | 2015-06-25 |
| AU2018253567A1 (en) | 2018-11-08 |
| AU2014364800A1 (en) | 2016-07-07 |
| AU2019216710A1 (en) | 2019-09-12 |
| WO2015095387A1 (en) | 2015-06-25 |
| JP2017503780A (ja) | 2017-02-02 |
| EP3082775A4 (en) | 2017-05-17 |
| JP6678212B2 (ja) | 2020-04-08 |
| JP2019001816A (ja) | 2019-01-10 |
| EP3082775A1 (en) | 2016-10-26 |
| AU2018253567B2 (en) | 2019-05-23 |
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