JP6359456B2 - 7−(1h−イミダゾール−4−イルメチル)−5,6,7,8−テトラヒドロキノリンを含む肌の疾患および状態を治療するための医薬組成物 - Google Patents

7−(1h−イミダゾール−4−イルメチル)−5,6,7,8−テトラヒドロキノリンを含む肌の疾患および状態を治療するための医薬組成物 Download PDF

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Publication number
JP6359456B2
JP6359456B2 JP2014541225A JP2014541225A JP6359456B2 JP 6359456 B2 JP6359456 B2 JP 6359456B2 JP 2014541225 A JP2014541225 A JP 2014541225A JP 2014541225 A JP2014541225 A JP 2014541225A JP 6359456 B2 JP6359456 B2 JP 6359456B2
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skin
pharmaceutical composition
ylmethyl
imidazol
tetrahydroquinoline
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JP2014533271A (ja
JP2014533271A5 (enExample
Inventor
モハメッド アイ ディーバス
モハメッド アイ ディーバス
エドワード シー シア
エドワード シー シア
ジョン イー ドネッロ
ジョン イー ドネッロ
ダニエル ダブリュ ギル
ダニエル ダブリュ ギル
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Allergan Inc
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Allergan Inc
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/14Decongestants or antiallergics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner

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  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Medicinal Preparation (AREA)
JP2014541225A 2011-11-10 2012-11-08 7−(1h−イミダゾール−4−イルメチル)−5,6,7,8−テトラヒドロキノリンを含む肌の疾患および状態を治療するための医薬組成物 Active JP6359456B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161558104P 2011-11-10 2011-11-10
US61/558,104 2011-11-10
PCT/US2012/064075 WO2013070861A1 (en) 2011-11-10 2012-11-08 Pharmaceutical compositions comprising 7-(1h-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinoline for treating skin diseases and conditions

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017092572A Division JP6526737B2 (ja) 2011-11-10 2017-05-08 7−(1h−イミダゾール−4−イルメチル)−5,6,7,8−テトラヒドロキノリンを含む肌の疾患および状態を治療するための医薬組成物

Publications (3)

Publication Number Publication Date
JP2014533271A JP2014533271A (ja) 2014-12-11
JP2014533271A5 JP2014533271A5 (enExample) 2016-01-07
JP6359456B2 true JP6359456B2 (ja) 2018-07-18

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Family Applications (2)

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JP2014541225A Active JP6359456B2 (ja) 2011-11-10 2012-11-08 7−(1h−イミダゾール−4−イルメチル)−5,6,7,8−テトラヒドロキノリンを含む肌の疾患および状態を治療するための医薬組成物
JP2017092572A Active JP6526737B2 (ja) 2011-11-10 2017-05-08 7−(1h−イミダゾール−4−イルメチル)−5,6,7,8−テトラヒドロキノリンを含む肌の疾患および状態を治療するための医薬組成物

Family Applications After (1)

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JP2017092572A Active JP6526737B2 (ja) 2011-11-10 2017-05-08 7−(1h−イミダゾール−4−イルメチル)−5,6,7,8−テトラヒドロキノリンを含む肌の疾患および状態を治療するための医薬組成物

Country Status (22)

Country Link
US (4) US20130123303A1 (enExample)
EP (3) EP2776034B1 (enExample)
JP (2) JP6359456B2 (enExample)
KR (1) KR102004563B1 (enExample)
CN (1) CN104136029A (enExample)
AR (1) AR088845A1 (enExample)
AU (2) AU2012335803B2 (enExample)
BR (1) BR112014011336A2 (enExample)
CA (1) CA2855005C (enExample)
CL (1) CL2014001242A1 (enExample)
DK (1) DK2776034T3 (enExample)
ES (1) ES2635421T3 (enExample)
IL (3) IL232483B (enExample)
MX (1) MX350662B (enExample)
MY (1) MY182553A (enExample)
PH (1) PH12014501051A1 (enExample)
RU (2) RU2630978C2 (enExample)
SG (3) SG11201402246RA (enExample)
TW (3) TW202014189A (enExample)
UA (1) UA109359C2 (enExample)
WO (1) WO2013070861A1 (enExample)
ZA (1) ZA201403396B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10201535B2 (en) 2011-11-10 2019-02-12 Allergan, Inc. Pharmaceutical compositions comprising 7-(1H-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinoline for treating skin diseases and conditions

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AU2014262960A1 (en) * 2013-05-06 2015-11-26 Allergan, Inc. Alpha adrenergic agonists for the treatment of tissue trauma
FR3061434B1 (fr) * 2017-01-04 2019-07-12 Pierre Fabre Dermo-Cosmetique Composition cosmetique comprenant une association d'huile de pongamia et de pentylene glycol 4-t-butylcyclohexanol pour lutter contre la rosacee
RU2727695C1 (ru) * 2020-02-13 2020-07-22 Мурад Умарович Магомедов Способ комплексного лечения ринофимы

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WO2004073708A1 (en) * 1998-12-17 2004-09-02 Dean Thomas R Brinzolamide and brimonidine for treating ocular conditions
US20010049369A1 (en) * 2000-02-10 2001-12-06 Jablonski Monica M. Brimonidine compositions and methods for retinal degeneration
US6468989B1 (en) 2000-07-13 2002-10-22 Dow Pharmaceutical Sciences Gel compositions containing metronidazole
US6387383B1 (en) 2000-08-03 2002-05-14 Dow Pharmaceutical Sciences Topical low-viscosity gel composition
US20020198209A1 (en) 2001-05-03 2002-12-26 Allergan Sales Inc. Compositions having enhanced pharmacokinetic characteristics
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US7030149B2 (en) * 2002-04-19 2006-04-18 Allergan, Inc. Combination of brimonidine timolol for topical ophthalmic use
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ZA200604403B (en) * 2003-11-20 2007-09-26 Othera Pharmaceuticals Inc Amelioration of macular degeneration and other ophthalmic diseases
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US7323477B2 (en) * 2006-02-02 2008-01-29 Allergan, Inc. 7-((1H-imidazol-4-yl)methyl)-5,6,7,8-tetrahydroquinoline
RU2321399C1 (ru) * 2006-06-01 2008-04-10 Федеральное государственное учреждение "Нижегородский научно-исследовательский кожно-венерологический институт Федерального агентства по здравоохранению и социальному развитию" Способ лечения больных розацеа
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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10201535B2 (en) 2011-11-10 2019-02-12 Allergan, Inc. Pharmaceutical compositions comprising 7-(1H-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinoline for treating skin diseases and conditions

Also Published As

Publication number Publication date
AU2012335803A1 (en) 2014-05-29
AU2016216627A1 (en) 2016-09-08
KR20140107237A (ko) 2014-09-04
TW201713338A (zh) 2017-04-16
NZ624771A (en) 2016-11-25
EP3763370A1 (en) 2021-01-13
JP2017149767A (ja) 2017-08-31
SG11201402246RA (en) 2014-06-27
SG10201609145PA (en) 2016-12-29
US9308201B2 (en) 2016-04-12
PH12014501051A1 (en) 2022-11-02
TWI708604B (zh) 2020-11-01
RU2667645C1 (ru) 2018-09-21
TWI580424B (zh) 2017-05-01
IL261269A (en) 2018-10-31
EP3184110B1 (en) 2020-10-07
CA2855005A1 (en) 2013-05-16
MX350662B (es) 2017-09-13
CL2014001242A1 (es) 2014-11-14
JP2014533271A (ja) 2014-12-11
SG10201809506TA (en) 2018-11-29
EP3184110A1 (en) 2017-06-28
MY182553A (en) 2021-01-25
EP2776034B1 (en) 2017-03-22
RU2014122758A (ru) 2015-12-20
MX2014005640A (es) 2014-09-22
KR102004563B1 (ko) 2019-07-26
US20150231128A1 (en) 2015-08-20
CA2855005C (en) 2016-11-22
AU2012335803B2 (en) 2016-05-26
AR088845A1 (es) 2014-07-10
EP2776034A1 (en) 2014-09-17
RU2630978C2 (ru) 2017-09-15
JP6526737B2 (ja) 2019-06-05
TW202014189A (zh) 2020-04-16
US20130123303A1 (en) 2013-05-16
WO2013070861A1 (en) 2013-05-16
UA109359C2 (xx) 2015-08-10
IL268757A (en) 2019-10-31
ES2635421T3 (es) 2017-10-03
CN104136029A (zh) 2014-11-05
DK2776034T3 (en) 2017-07-10
TW201328694A (zh) 2013-07-16
IL232483A0 (en) 2014-06-30
IL232483B (en) 2018-10-31
US20170095466A1 (en) 2017-04-06
BR112014011336A2 (pt) 2017-05-02
AU2016216627B2 (en) 2017-10-19
ZA201403396B (en) 2015-07-29
US20160051534A1 (en) 2016-02-25

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