JP6158180B2 - 乳がんの処置 - Google Patents

乳がんの処置 Download PDF

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Publication number
JP6158180B2
JP6158180B2 JP2014523048A JP2014523048A JP6158180B2 JP 6158180 B2 JP6158180 B2 JP 6158180B2 JP 2014523048 A JP2014523048 A JP 2014523048A JP 2014523048 A JP2014523048 A JP 2014523048A JP 6158180 B2 JP6158180 B2 JP 6158180B2
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JP
Japan
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substituted
alkyl
heterocyclic
alkenyl
alkynyl
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JP2014523048A
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English (en)
Japanese (ja)
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JP2014524934A (ja
JP2014524934A5 (OSRAM
Inventor
アンドリュー エー． プロッター，
アンドリュー エー． プロッター，
ジェニファー リッチャー，
ジェニファー リッチャー，
ドーン コックレン，
ドーン コックレン，
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University of Colorado System
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University of Colorado System
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48192564&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JP6158180(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by University of Colorado System filed Critical University of Colorado System
Publication of JP2014524934A publication Critical patent/JP2014524934A/ja
Publication of JP2014524934A5 publication Critical patent/JP2014524934A5/ja
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2014523048A 2011-07-29 2012-07-27 乳がんの処置 Active JP6158180B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161513361P 2011-07-29 2011-07-29
US61/513,361 2011-07-29
PCT/US2012/048471 WO2013066440A1 (en) 2011-07-29 2012-07-27 Treatment of breast cancer

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017072819A Division JP2017141269A (ja) 2011-07-29 2017-03-31 乳がんの処置

Publications (3)

Publication Number Publication Date
JP2014524934A JP2014524934A (ja) 2014-09-25
JP2014524934A5 JP2014524934A5 (OSRAM) 2015-08-27
JP6158180B2 true JP6158180B2 (ja) 2017-07-05

Family

ID=48192564

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2014523048A Active JP6158180B2 (ja) 2011-07-29 2012-07-27 乳がんの処置
JP2017072819A Pending JP2017141269A (ja) 2011-07-29 2017-03-31 乳がんの処置

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2017072819A Pending JP2017141269A (ja) 2011-07-29 2017-03-31 乳がんの処置

Country Status (18)

Country Link
US (4) US9517229B2 (OSRAM)
EP (4) EP3610731A1 (OSRAM)
JP (2) JP6158180B2 (OSRAM)
KR (1) KR101923250B1 (OSRAM)
CN (1) CN103997894B (OSRAM)
BR (1) BR112014002200A2 (OSRAM)
CA (1) CA2843417C (OSRAM)
CY (1) CY1121038T1 (OSRAM)
DK (1) DK2739153T3 (OSRAM)
EA (1) EA028452B1 (OSRAM)
ES (1) ES2696074T3 (OSRAM)
HU (1) HUE040524T2 (OSRAM)
MX (1) MX359664B (OSRAM)
PH (1) PH12014500248B1 (OSRAM)
PL (1) PL2739153T3 (OSRAM)
PT (1) PT2739153T (OSRAM)
SI (1) SI2739153T1 (OSRAM)
WO (1) WO2013066440A1 (OSRAM)

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JP2017141269A (ja) * 2011-07-29 2017-08-17 メディベイション プロステイト セラピューティクス， インコーポレイテッド 乳がんの処置

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UA115805C2 (uk) * 2013-04-17 2017-12-26 Сігнал Фармасьютікалз, Елелсі Комбінована терапія, яка включає сполуку дигідропіразинопіразину й антагоніст рецептора андрогену, для лікування раку простати
JP6945587B2 (ja) * 2013-11-07 2021-10-06 デシフェラ ファーマシューティカルズ，エルエルシー ガンの処置に有用なｔｉｅ２キナーゼの阻害方法
CA2929715A1 (en) * 2013-11-07 2015-05-14 Deciphera Pharmaceuticals, Llc Methods for inhibiting tie2 kinase useful in the treatment of cancer
WO2015184145A1 (en) * 2014-05-28 2015-12-03 Eisai R&D Management Co., Ltd. Use of eribulin and poly (adp ribose) polymerase (parp) inhibitors as combination therapy for the treatment of cancer
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CN104857517B (zh) * 2015-05-14 2018-04-27 南京海纳医药科技股份有限公司 一种恩杂鲁胺软胶囊及其制备方法
US9963433B2 (en) * 2016-01-29 2018-05-08 Wayne State University Anticancer drugs including the chemical structures of an androgen receptor ligand and a histone deacetylase inhibitor
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CN107987055A (zh) * 2017-12-19 2018-05-04 刘秀云 硫代咪唑二酮类雄激素受体拮抗剂及其用途
WO2019152711A1 (en) 2018-01-31 2019-08-08 Diciphera Pharmaceuticals Llc. Combination therapy for the treatment of gastrointestinal stromal tumors
KR102708050B1 (ko) 2018-01-31 2024-09-24 데시페라 파마슈티칼스, 엘엘씨. 비만 세포증의 치료를 위한 병용 요법
US11292782B2 (en) 2018-11-30 2022-04-05 Nuvation Bio Inc. Diarylhydantoin compounds and methods of use thereof
AU2019387370A1 (en) 2018-11-30 2021-06-10 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
TWI878335B (zh) 2019-08-12 2025-04-01 美商迪賽孚爾製藥有限公司 治療胃腸道基質瘤方法
CA3150433A1 (en) 2019-08-12 2021-02-18 Deciphera Pharmaceuticals, Llc Ripretinib for treating gastrointestinal stromal tumors
FI4084778T3 (fi) 2019-12-30 2023-12-18 Deciphera Pharmaceuticals Llc Amorfisia kinaasi-inhibiittoriformulaatioita ja menetelmiä niiden käyttämiseksi
CN115243681B (zh) 2019-12-30 2024-08-16 德西费拉制药有限责任公司 1-(4-溴-5-(1-乙基-7-(甲氨基)-2-侧氧基-1,2-二氢-1,6-萘啶-3-基)-2-氟苯基)-3-苯基脲的组合物
KR20230058410A (ko) * 2020-08-03 2023-05-03 온코사이트 코포레이션 종양의 분류 및 반응성 예측
US11779572B1 (en) 2022-09-02 2023-10-10 Deciphera Pharmaceuticals, Llc Methods of treating gastrointestinal stromal tumors

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Publication number Priority date Publication date Assignee Title
JP2017141269A (ja) * 2011-07-29 2017-08-17 メディベイション プロステイト セラピューティクス， インコーポレイテッド 乳がんの処置

Also Published As

Publication number Publication date
SI2739153T1 (sl) 2018-12-31
BR112014002200A2 (pt) 2017-03-07
HK1201413A1 (en) 2015-09-04
CN103997894A (zh) 2014-08-20
JP2014524934A (ja) 2014-09-25
CN103997894B (zh) 2016-08-24
US20210069154A1 (en) 2021-03-11
CA2843417C (en) 2018-08-21
HK1198867A1 (en) 2015-06-19
EA028452B1 (ru) 2017-11-30
EP2739153B1 (en) 2018-08-22
US20140296312A1 (en) 2014-10-02
DK2739153T3 (en) 2018-12-03
ES2696074T3 (es) 2019-01-14
US10111861B2 (en) 2018-10-30
WO2013066440A9 (en) 2013-07-18
PH12014500248A1 (en) 2014-03-17
JP2017141269A (ja) 2017-08-17
HUE040524T2 (hu) 2019-03-28
EP3610731A1 (en) 2020-02-19
PT2739153T (pt) 2018-11-28
PH12014500248B1 (en) 2018-08-31
PL2739153T3 (pl) 2019-04-30
EP2739153A4 (en) 2015-03-11
KR101923250B1 (ko) 2018-11-28
US20190262315A1 (en) 2019-08-29
MX359664B (es) 2018-10-05
US9517229B2 (en) 2016-12-13
CA2843417A1 (en) 2013-05-10
EP3791724A1 (en) 2021-03-17
EP3430907A1 (en) 2019-01-23
CY1121038T1 (el) 2019-12-11
EP2739153A1 (en) 2014-06-11
MX2014001218A (es) 2014-08-22
US20170087132A1 (en) 2017-03-30
KR20140107174A (ko) 2014-09-04
WO2013066440A1 (en) 2013-05-10
EA201400178A1 (ru) 2014-11-28

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