JP5857008B2 - C−4”位置換マクロライド誘導体を含有する医薬 - Google Patents
C−4”位置換マクロライド誘導体を含有する医薬 Download PDFInfo
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- JP5857008B2 JP5857008B2 JP2013169941A JP2013169941A JP5857008B2 JP 5857008 B2 JP5857008 B2 JP 5857008B2 JP 2013169941 A JP2013169941 A JP 2013169941A JP 2013169941 A JP2013169941 A JP 2013169941A JP 5857008 B2 JP5857008 B2 JP 5857008B2
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- 0 C*(C)N(*)C(C1)C1(COC1(C2)C(C[C@@]([C@@](C)[C@@](*[C@@](C3)OC4(CC4)CC3(C3)C3N(C)C)[C@@](C3)*3CCC*[C@](*)C[C@](C)C3([C@](C)C3C)O3)C4(CC4)C3=O)C1)[C@]2OC Chemical compound C*(C)N(*)C(C1)C1(COC1(C2)C(C[C@@]([C@@](C)[C@@](*[C@@](C3)OC4(CC4)CC3(C3)C3N(C)C)[C@@](C3)*3CCC*[C@](*)C[C@](C)C3([C@](C)C3C)O3)C4(CC4)C3=O)C1)[C@]2OC 0.000 description 3
- NLJHLCBDUOXJQK-UHFFFAOYSA-N C(C1)C11CC2(CC2)OC2(CC2)C1 Chemical compound C(C1)C11CC2(CC2)OC2(CC2)C1 NLJHLCBDUOXJQK-UHFFFAOYSA-N 0.000 description 1
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Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
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JP2013169941A JP5857008B2 (ja) | 2012-08-20 | 2013-08-19 | C−4”位置換マクロライド誘導体を含有する医薬 |
Applications Claiming Priority (3)
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JP2012181339 | 2012-08-20 | ||
JP2012181339 | 2012-08-20 | ||
JP2013169941A JP5857008B2 (ja) | 2012-08-20 | 2013-08-19 | C−4”位置換マクロライド誘導体を含有する医薬 |
Publications (3)
Publication Number | Publication Date |
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JP2014058509A JP2014058509A (ja) | 2014-04-03 |
JP2014058509A5 JP2014058509A5 (ru) | 2014-07-17 |
JP5857008B2 true JP5857008B2 (ja) | 2016-02-10 |
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JP2013169941A Expired - Fee Related JP5857008B2 (ja) | 2012-08-20 | 2013-08-19 | C−4”位置換マクロライド誘導体を含有する医薬 |
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JP (1) | JP5857008B2 (ru) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR102810A1 (es) | 2014-08-18 | 2017-03-29 | Taisho Pharmaceutical Co Ltd | Derivado de macrólido sustituido en la posición c-4 |
CN104592057B (zh) * | 2015-01-12 | 2017-05-10 | 中国科学院上海有机化学研究所 | 一种三硝基乙基氨基甲酸酯的合成方法 |
WO2017142002A1 (ja) * | 2016-02-17 | 2017-08-24 | 大正製薬株式会社 | C-4"位置換マクロライド化合物フリー体及び塩の結晶形並びにそれらの製造方法 |
CN106748905B (zh) * | 2016-12-14 | 2018-04-13 | 河南省化工研究所有限责任公司 | 一种制备2‑氨基乙基磺酰胺盐酸盐的方法 |
CN106928294A (zh) * | 2017-03-22 | 2017-07-07 | 上海启雁实业有限公司 | 制备酮内酯大环内酯类抗生素的方法 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1998009978A1 (en) * | 1996-09-04 | 1998-03-12 | Abbott Laboratories | 6-o-substituted ketolides having antibacterial activity |
HN1998000074A (es) * | 1997-06-11 | 1999-01-08 | Pfizer Prod Inc | Derivados de macrolidos c-4 sustituidos |
WO2008143729A2 (en) * | 2007-02-28 | 2008-11-27 | Rib-X Pharmaceuticals, Inc. | Macrolide compounds and methods of making and using the same |
AR085286A1 (es) * | 2011-02-21 | 2013-09-18 | Taisho Pharmaceutical Co Ltd | Derivado de macrolido sustituido en la posicion c-4 |
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2013
- 2013-08-19 JP JP2013169941A patent/JP5857008B2/ja not_active Expired - Fee Related
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JP2014058509A (ja) | 2014-04-03 |
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