JP5671537B2 - ４−アミノブタ−２−エノリド類の新規調製方法 - Google Patents
４−アミノブタ−２−エノリド類の新規調製方法 Download PDFInfo
- Publication number
- JP5671537B2 JP5671537B2 JP2012525066A JP2012525066A JP5671537B2 JP 5671537 B2 JP5671537 B2 JP 5671537B2 JP 2012525066 A JP2012525066 A JP 2012525066A JP 2012525066 A JP2012525066 A JP 2012525066A JP 5671537 B2 JP5671537 B2 JP 5671537B2
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- chloro
- acid
- formula
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/66—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Furan Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP09168068 | 2009-08-18 | ||
| EP09168068.6 | 2009-08-18 | ||
| US23587809P | 2009-08-21 | 2009-08-21 | |
| US61/235,878 | 2009-08-21 | ||
| PCT/EP2010/004800 WO2011020564A1 (de) | 2009-08-18 | 2010-08-05 | Neues verfahren zur herstellung von 4-aminobut-2-enoliden |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013502385A JP2013502385A (ja) | 2013-01-24 |
| JP5671537B2 true JP5671537B2 (ja) | 2015-02-18 |
Family
ID=41226872
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012525066A Active JP5671537B2 (ja) | 2009-08-18 | 2010-08-05 | ４−アミノブタ−２−エノリド類の新規調製方法 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US8314242B2 (enExample) |
| EP (1) | EP2467374B1 (enExample) |
| JP (1) | JP5671537B2 (enExample) |
| KR (1) | KR20120059555A (enExample) |
| CN (1) | CN102471315B (enExample) |
| BR (1) | BR112012003225A2 (enExample) |
| DK (1) | DK2467374T3 (enExample) |
| ES (1) | ES2421394T3 (enExample) |
| IL (1) | IL217460A0 (enExample) |
| IN (1) | IN2012DN01461A (enExample) |
| MX (1) | MX2012001727A (enExample) |
| TW (1) | TW201111370A (enExample) |
| WO (1) | WO2011020564A1 (enExample) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN113896679B (zh) * | 2021-11-18 | 2024-03-01 | 合肥利夫生物科技有限公司 | 一种吡咯吡啶激酶抑制剂关键中间体的合成方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH503722A (de) | 1969-05-28 | 1971-02-28 | Lonza Ag | Verfahren zur Herstellung von Tetronsäure |
| DE3311003A1 (de) | 1983-03-25 | 1984-09-27 | Bayer Ag, 5090 Leverkusen | Chromon- und thiochromonsubstituierte 1,4-dihydropyridinlactone, mehrere verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln |
| CH658056A5 (de) | 1984-02-09 | 1986-10-15 | Lonza Ag | Verfahren zur herstellung von tetronsaeure. |
| WO1992000964A1 (fr) | 1990-07-05 | 1992-01-23 | Nippon Soda Co., Ltd. | Derive d'amine |
| US5252741A (en) * | 1990-08-10 | 1993-10-12 | Reilly Industries, Inc. | Processes for the synthesis of imines, aldehydes, and unsymmetrical secondary amines |
| DE102006015467A1 (de) * | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| EP2039678A1 (de) | 2007-09-18 | 2009-03-25 | Bayer CropScience AG | Verfahren zum Herstellen von 4-Aminobut-2-enoliden |
| EP2042496A1 (de) * | 2007-09-18 | 2009-04-01 | Bayer CropScience AG | Verfahren zur Herstellung von 4-Aminobut-2-enoliden |
-
2010
- 2010-07-30 TW TW099125236A patent/TW201111370A/zh unknown
- 2010-08-05 EP EP10742759.3A patent/EP2467374B1/de active Active
- 2010-08-05 WO PCT/EP2010/004800 patent/WO2011020564A1/de not_active Ceased
- 2010-08-05 ES ES10742759T patent/ES2421394T3/es active Active
- 2010-08-05 JP JP2012525066A patent/JP5671537B2/ja active Active
- 2010-08-05 MX MX2012001727A patent/MX2012001727A/es active IP Right Grant
- 2010-08-05 CN CN201080035042.9A patent/CN102471315B/zh active Active
- 2010-08-05 DK DK10742759.3T patent/DK2467374T3/da active
- 2010-08-05 IN IN1461DEN2012 patent/IN2012DN01461A/en unknown
- 2010-08-05 BR BR112012003225A patent/BR112012003225A2/pt not_active Application Discontinuation
- 2010-08-05 KR KR1020127006802A patent/KR20120059555A/ko not_active Withdrawn
- 2010-08-17 US US12/858,031 patent/US8314242B2/en active Active
-
2012
- 2012-01-10 IL IL217460A patent/IL217460A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20110054182A1 (en) | 2011-03-03 |
| CN102471315B (zh) | 2014-05-28 |
| DK2467374T3 (da) | 2013-08-05 |
| US8314242B2 (en) | 2012-11-20 |
| WO2011020564A1 (de) | 2011-02-24 |
| MX2012001727A (es) | 2012-04-02 |
| BR112012003225A2 (pt) | 2015-09-22 |
| KR20120059555A (ko) | 2012-06-08 |
| EP2467374B1 (de) | 2013-05-01 |
| CN102471315A (zh) | 2012-05-23 |
| ES2421394T3 (es) | 2013-09-02 |
| TW201111370A (en) | 2011-04-01 |
| IL217460A0 (en) | 2012-03-01 |
| IN2012DN01461A (enExample) | 2015-06-05 |
| EP2467374A1 (de) | 2012-06-27 |
| JP2013502385A (ja) | 2013-01-24 |
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