JP5393700B2 - 治療化合物 - Google Patents
治療化合物 Download PDFInfo
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- JP5393700B2 JP5393700B2 JP2010543201A JP2010543201A JP5393700B2 JP 5393700 B2 JP5393700 B2 JP 5393700B2 JP 2010543201 A JP2010543201 A JP 2010543201A JP 2010543201 A JP2010543201 A JP 2010543201A JP 5393700 B2 JP5393700 B2 JP 5393700B2
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- compound according
- pharmaceutically acceptable
- acceptable salt
- intraocular pressure
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Ophthalmology & Optometry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Cosmetics (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2228208P | 2008-01-18 | 2008-01-18 | |
| US61/022,282 | 2008-01-18 | ||
| US12/352,995 | 2009-01-13 | ||
| US12/352,995 US7964595B2 (en) | 2008-01-18 | 2009-01-13 | Thiophenyl prostaglandin derivatives for treating glaucoma and ocular hypertension |
| PCT/US2009/030895 WO2009091765A1 (en) | 2008-01-18 | 2009-01-14 | Therapeutic compounds |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011522775A JP2011522775A (ja) | 2011-08-04 |
| JP2011522775A5 JP2011522775A5 (https=) | 2012-03-01 |
| JP5393700B2 true JP5393700B2 (ja) | 2014-01-22 |
Family
ID=40876973
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010543201A Expired - Fee Related JP5393700B2 (ja) | 2008-01-18 | 2009-01-14 | 治療化合物 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7964595B2 (https=) |
| EP (1) | EP2240462B1 (https=) |
| JP (1) | JP5393700B2 (https=) |
| AU (1) | AU2009205478B2 (https=) |
| BR (1) | BRPI0906879A2 (https=) |
| CA (1) | CA2712192C (https=) |
| DK (1) | DK2240462T3 (https=) |
| ES (1) | ES2434963T3 (https=) |
| WO (1) | WO2009091765A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG193840A1 (en) * | 2008-09-04 | 2013-10-30 | Santen Pharmaceutical Co Ltd | HAIR GROWTH PROMOTING AGENT CONTAINING 15,15-DIFLUOROPROSTAGLANDIN F2a DERIVATIVE AS ACTIVE INGREDIENT |
| WO2013180229A1 (ja) * | 2012-05-30 | 2013-12-05 | 旭硝子株式会社 | 育毛用組成物 |
| US9540357B1 (en) | 2014-07-31 | 2017-01-10 | Allergan, Inc. | 15-aryl prostaglandins as EP4 agonists, and methods of use thereof |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4543353A (en) * | 1981-11-27 | 1985-09-24 | Farmitalia Carlo Erba S.P.A. | Ester and amide derivatives of 13,14-didehydro prostaglandins |
| JPH0692305B2 (ja) * | 1987-05-15 | 1994-11-16 | 株式会社上野製薬応用研究所 | 体温上昇剤 |
| US5688819A (en) | 1992-09-21 | 1997-11-18 | Allergan | Cyclopentane heptanoic acid, 2-cycloalkyl or arylalkyl derivatives as therapeutic agents |
| WO2000051977A1 (en) * | 1999-03-05 | 2000-09-08 | The Procter & Gamble Company | Aldehyde intermediates for the preparation of prostaglandin derivatives |
| JP4834224B2 (ja) * | 1999-03-05 | 2011-12-14 | デューク ユニバーシティ | Ｃ１６不飽和ｆｐ−選択的プロスタグランジン類縁体 |
| US7166730B2 (en) | 2000-01-27 | 2007-01-23 | Fine Tech Laboratories, Ltd | Process for the preparation of prostaglandin derivatives |
| IL143477A (en) | 2001-05-31 | 2009-07-20 | Finetech Pharmaceutical Ltd | Process for the preparation of 17-phenyl-18,19,20-trinor-pgf2?? and its derivatives |
| US7101904B2 (en) * | 2004-08-10 | 2006-09-05 | Allergan, Inc. | Cyclopentane heptan(ENE)OIC acid, 2-heteroarylalkenyl derivatives as therapeutic agents |
| US7427685B2 (en) * | 2005-12-06 | 2008-09-23 | Allergan, Inc. | Therapeutic substituted cyclopentanes |
| US20070254920A1 (en) * | 2006-04-26 | 2007-11-01 | Aerie Pharmaceuticals, Inc. | Prodrug derivatives of acids using alcohols with homotopic hydroxy groups and methods for their preparation and use |
-
2009
- 2009-01-13 US US12/352,995 patent/US7964595B2/en active Active
- 2009-01-14 BR BRPI0906879-1A patent/BRPI0906879A2/pt not_active IP Right Cessation
- 2009-01-14 EP EP09702525.8A patent/EP2240462B1/en not_active Not-in-force
- 2009-01-14 ES ES09702525T patent/ES2434963T3/es active Active
- 2009-01-14 WO PCT/US2009/030895 patent/WO2009091765A1/en not_active Ceased
- 2009-01-14 CA CA2712192A patent/CA2712192C/en not_active Expired - Fee Related
- 2009-01-14 DK DK09702525.8T patent/DK2240462T3/da active
- 2009-01-14 AU AU2009205478A patent/AU2009205478B2/en not_active Ceased
- 2009-01-14 JP JP2010543201A patent/JP5393700B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009091765A1 (en) | 2009-07-23 |
| AU2009205478B2 (en) | 2014-01-16 |
| JP2011522775A (ja) | 2011-08-04 |
| CA2712192A1 (en) | 2009-07-23 |
| CA2712192C (en) | 2016-06-14 |
| EP2240462B1 (en) | 2013-08-21 |
| BRPI0906879A2 (pt) | 2015-07-07 |
| DK2240462T3 (da) | 2013-10-28 |
| EP2240462A1 (en) | 2010-10-20 |
| US20090186885A1 (en) | 2009-07-23 |
| US7964595B2 (en) | 2011-06-21 |
| ES2434963T3 (es) | 2013-12-18 |
| AU2009205478A1 (en) | 2009-07-23 |
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