JP4098985B2 - テトラヒドロピペリンならびにその類似体および誘導体を用いて栄養素および薬剤調製物の生体利用能を高める方法 - Google Patents
テトラヒドロピペリンならびにその類似体および誘導体を用いて栄養素および薬剤調製物の生体利用能を高める方法 Download PDFInfo
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- JP4098985B2 JP4098985B2 JP2001585813A JP2001585813A JP4098985B2 JP 4098985 B2 JP4098985 B2 JP 4098985B2 JP 2001585813 A JP2001585813 A JP 2001585813A JP 2001585813 A JP2001585813 A JP 2001585813A JP 4098985 B2 JP4098985 B2 JP 4098985B2
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- Prior art keywords
- tetrahydropiperine
- piperine
- test
- skin
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
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Classifications
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/22—Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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| PCT/US2001/016070 WO2001089571A2 (en) | 2000-05-19 | 2001-05-21 | Method of increased bioavailability of nutrients and pharmaceutical preparations with tetrahydropiperine and its analogues and derivatives |
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| CA2489947A1 (en) * | 2002-06-24 | 2003-12-31 | Research Development Foundation | Treatment of human multiple myeloma by curcumin |
| WO2004067018A1 (en) * | 2003-01-30 | 2004-08-12 | Council Of Scientific And Industrial Research | Bioavailability enhancing activity of carum carvi extracts and fractions thereof |
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| US20050163873A1 (en) * | 2004-01-14 | 2005-07-28 | Robert Ritch | Methods and formulations for treating glaucoma |
| JP5254616B2 (ja) | 2004-09-13 | 2013-08-07 | クロノ セラピューティクス、インコーポレイテッド | 生物学的同調性(biosynchronous)経皮的薬物送達 |
| US8252321B2 (en) | 2004-09-13 | 2012-08-28 | Chrono Therapeutics, Inc. | Biosynchronous transdermal drug delivery for longevity, anti-aging, fatigue management, obesity, weight loss, weight management, delivery of nutraceuticals, and the treatment of hyperglycemia, alzheimer's disease, sleep disorders, parkinson's disease, aids, epilepsy, attention deficit disorder, nicotine addiction, cancer, headache and pain control, asthma, angina, hypertension, depression, cold, flu and the like |
| US20060130675A1 (en) * | 2004-11-30 | 2006-06-22 | Crawford David S | Transdermal nutritional supplement delivery patch |
| US8372040B2 (en) | 2005-05-24 | 2013-02-12 | Chrono Therapeutics, Inc. | Portable drug delivery device including a detachable and replaceable administration or dosing element |
| US20070237735A1 (en) * | 2006-03-31 | 2007-10-11 | Laboratoires Dermo-Cosmetik Inc. | Anti-aging composition, kit and method of use |
| US20080138417A1 (en) * | 2006-11-22 | 2008-06-12 | Charles Grigsby | Topical Composition And Method Of Forming |
| US20130017259A1 (en) | 2011-07-06 | 2013-01-17 | The Parkinson's Institute | Compositions and Methods for Treatment of Symptoms in Parkinson's Disease Patients |
| US10105487B2 (en) | 2013-01-24 | 2018-10-23 | Chrono Therapeutics Inc. | Optimized bio-synchronous bioactive agent delivery system |
| JP2018511355A (ja) | 2015-01-28 | 2018-04-26 | クロノ セラピューティクス インコーポレイテッドChrono Therapeutics Inc. | 薬剤送達方法及びシステム |
| AU2016228779A1 (en) | 2015-03-12 | 2017-09-07 | Chrono Therapeutics Inc. | Craving input and support system |
| WO2017020125A1 (en) * | 2015-07-31 | 2017-02-09 | Delivra Inc. | Transdermal formulations for delivery of capsaicinoids |
| KR102655937B1 (ko) * | 2016-09-27 | 2024-04-11 | (주)아모레퍼시픽 | 코스모페린을 포함하는 항스트레스 조성물 |
| WO2018069938A1 (en) * | 2016-10-14 | 2018-04-19 | Cipla Limited | Pharmaceutical compositions comprising rifaximin |
| EP3565617A1 (en) | 2017-01-06 | 2019-11-13 | Chrono Therapeutics Inc. | Transdermal drug delivery devices and methods |
| WO2019058386A1 (en) * | 2017-09-19 | 2019-03-28 | Cipla Limited | COMPOSITIONS COMPRISING IBRUTINIB AND AN ALKALOID HAVING IMPROVED BIOAVAILABILITY |
| EP3801732A4 (en) | 2018-05-29 | 2022-04-27 | Morningside Venture Investments Limited | METHODS AND SYSTEMS FOR DRUG DELIVERY |
| US12397141B2 (en) | 2018-11-16 | 2025-08-26 | Morningside Venture Investments Limited | Thermally regulated transdermal drug delivery system |
| US20200179362A1 (en) * | 2018-12-05 | 2020-06-11 | James E. Beecham | Dietary supplement comprising glucuronidation inhibition assist for healthful daily synergy of anti-inflammation, cellular anti-oxidant boost, cellular protein clean-up boost |
| JP7163261B2 (ja) * | 2019-09-27 | 2022-10-31 | 富士フイルム株式会社 | 水中油型乳化組成物、及び皮膚外用剤 |
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| EP0650728B1 (en) * | 1993-10-29 | 2002-02-27 | Council of Scientific and Industrial Research | Pharmaceutical compositions containing piperine and an antituberculosis or antileprosydrug |
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- 2001-05-21 GB GB0229561A patent/GB2380675B/en not_active Expired - Lifetime
- 2001-05-21 JP JP2001585813A patent/JP4098985B2/ja not_active Expired - Lifetime
- 2001-05-21 US US09/860,816 patent/US6849645B2/en not_active Expired - Lifetime
- 2001-05-21 AU AU2001278849A patent/AU2001278849A1/en not_active Abandoned
- 2001-05-21 WO PCT/US2001/016070 patent/WO2001089571A2/en not_active Ceased
- 2001-05-21 DE DE10196213.4A patent/DE10196213B4/de not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| US6849645B2 (en) | 2005-02-01 |
| WO2001089571A2 (en) | 2001-11-29 |
| DE10196213T1 (de) | 2003-04-30 |
| JP2003534295A (ja) | 2003-11-18 |
| DE10196213B4 (de) | 2020-12-17 |
| GB0229561D0 (en) | 2003-01-22 |
| WO2001089571A3 (en) | 2002-03-07 |
| GB2380675B (en) | 2004-11-03 |
| GB2380675A (en) | 2003-04-16 |
| AU2001278849A1 (en) | 2001-12-03 |
| US20020058695A1 (en) | 2002-05-16 |
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